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Title:
トレプロスチニル誘導体化合物およびその使用方法
Document Type and Number:
Japanese Patent JP6561109
Kind Code:
B2
Abstract:
Compounds represented by formulae I, II, III, and IV including pro-drugs for treprostinil and prostacyclin analogs. Uses include treatment of pulmonary hypertension (PH) or pulmonary arterial hypertension (PAH). The structures of the compounds can be adapted to the particular application for suitable treatment dosage. Transdermal applications can be used.

Inventors:
Becker Cyrus Kay.
Liscourio Gwenaela
Pfister Jurgue
Benkatraman Minax
Chang Xiao Ming
Application Number:
JP2017500911A
Publication Date:
August 14, 2019
Filing Date:
July 16, 2014
Export Citation:
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Assignee:
Corsair Pharma Inc.
International Classes:
C07C69/712; A61K31/40; A61K31/421; A61K31/439; A61K31/445; A61K31/5375; A61K45/00; A61P7/02; A61P7/10; A61P9/00; A61P9/12; A61P11/00; A61P43/00; C07C235/20; C07D211/60; C07D257/06; C07D263/26; C07D265/30; C07D295/088; C07D321/00; C07D323/00; C07D453/02
Domestic Patent References:
JP2007501281A
Foreign References:
WO2013024052A1
US20030108512
WO2011153363A1
Attorney, Agent or Firm:
Hatsushi Shimizu
Masao Haruna
Hirotaka Yamaguchi
Toshi Gobe
Ryuichi Inoue
Toshimitsu Sato
Koichi Niimi
Tomohiko Kobayashi
Hideki Kodera
Masato Ozeki
Yoshihiro Igarashi
Kazuya Kawamoto