Title:
炎症性疾患および疼痛の治療における、β-アミノアルコールの使用
Document Type and Number:
Japanese Patent JP5174987
Kind Code:
B2
Abstract:
A compound for therapeutic use, of the formula wherein R1 is aryl or heteroaryl optionally substituted with R5; R2 is H, alkyl or CH2OH or forms part of a ring with R4; R3 is H, alkyl or CH2OH or forms part of a ring with R4; R4 is H, alkyl or (when forming part of a ring with R2 or R3) CH2; and R5 is alkyl, CF3, OH, Oalkyl, OCOalkyl, CONH2, CN, halogen, NH2, NO2, NHCHO, NHCONH2, NHSO2Me, CONH2, or SOMe; or a salt thereof.
Inventors:
Brew, John
Baxter, Andrew Douglas
Bannister, Robin Mark
Baxter, Andrew Douglas
Bannister, Robin Mark
Application Number:
JP2012224947A
Publication Date:
April 03, 2013
Filing Date:
October 10, 2012
Export Citation:
Assignee:
Biocopea Limited
International Classes:
A61P1/02; A61K31/137; A61P1/04; A61P9/00; A61P17/00; A61P17/04; A61P17/06; A61P19/02; A61P25/04; A61P25/06; A61P29/00; C07C225/06; C07C225/22
Domestic Patent References:
| JP2003529563A | ||||
| JP5811852B1 | ||||
| JP60132937A | ||||
| JP52131579A | ||||
| JP53112883A | ||||
| JP57154129A |
Foreign References:
| WO2005044809A1 | ||||
| FR8801566A1 | ||||
| US2900415 | ||||
| GB886035A | ||||
| DE152814C1 | ||||
| WO2002016327A1 | ||||
| WO2006092691A1 |
Other References:
Yingyong Huaxue,Vol.22, No.3,p.343-345 (2005).
Journal of Medicinal Chemistry,Vol.39, No.2,p.347-349 (1996).
Journal of Medicinal Chemistry,Vol.39, No.2,p.347-349 (1996).
Attorney, Agent or Firm:
Hidekazu Miyoshi
Masakazu Ito
Yuko Hara
Masakazu Ito
Yuko Hara