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Title:
2型糖尿病の防止および処置において使用することができる医薬品を調製するためのリモナバントの使用
Document Type and Number:
Japanese Patent JP2008530189
Kind Code:
A
Abstract:
Use of rimonabant and N-piperidino-5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-ethylpyrazole-3-carboxamide, as cannabinoids (CB1) receptor antagonists (I), for the preparation of drugs useful to treat and prevent type-II diabetes. An independent claim is included for a composition comprising (I) and an active ingredient of metformin and sulfonylurea. ACTIVITY : Antidiabetic. MECHANISM OF ACTION : Cannabinoids (CB1) receptor antagonist.

Inventors:
Anotan, Corinne
Lauzan's waig, pierre
Application Number:
JP2007555669A
Publication Date:
August 07, 2008
Filing Date:
February 20, 2006
Export Citation:
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Assignee:
Sanofui-Aventice
International Classes:
A61K31/454; A61K31/155; A61K45/00; A61P3/10; A61P9/00; A61P25/02; A61P27/02; C07D231/14
Attorney, Agent or Firm:
Yoshio Kawaguchi
Makoto Ono
Chihiro Watanabe
Kenkyo Kanayama
Katsuma Osaki
Mitsuaki Tsubokura