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Title:
ビタミンDレセプターモジュレーター
Document Type and Number:
Japanese Patent JP4594099
Kind Code:
B2
Abstract:
The present invention relates to novel, non-secosteroidal, diaryl compounds with vitamin D receptor (VDR) modulating activity that are less hypercalcemic than 1α,25 dihydroxy vitamin D3. These compounds are useful for treating bone disease and psoriasis.

Inventors:
Emilio Enrique Bonnell
Robert Peter Gajuski
Charles David Jones
Le Jeanlian
Ma Tianway
Sunil Nagpal
In Kwon Yi
Application Number:
JP2004555373A
Publication Date:
December 08, 2010
Filing Date:
November 20, 2003
Export Citation:
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Assignee:
Eli Lilly and Company
International Classes:
C07C235/34; A61K31/137; A61K31/165; A61K31/18; A61K31/192; A61K31/198; A61K31/235; A61K31/41; A61K31/426; A61K31/565; A61K31/60; A61K31/663; A61K35/04; A61K38/23; A61P3/10; A61P3/14; A61P17/00; A61P17/06; A61P19/00; A61P19/10; A61P21/04; A61P25/00; A61P25/28; A61P29/00; A61P35/00; A61P35/02; A61P43/00; C07C51/09; C07C51/367; C07C51/373; C07C59/48; C07C59/64; C07C59/66; C07C59/68; C07C59/90; C07C65/24; C07C65/34; C07C65/40; C07C67/36; C07C69/732; C07C69/734; C07C69/738; C07C69/76; C07C69/94; C07C231/02; C07C231/12; C07C231/14; C07C235/42; C07C311/51; C07C315/04; C07C317/28; C07D207/26; C07D207/27; C07D233/78; C07D257/04; C07D257/06; C07D261/12; C07D271/113; C07D277/34; C07D295/185; C07B53/00; C07B57/00; C07B61/00; C07D271/10
Domestic Patent References:
JP2002523388A
Attorney, Agent or Firm:
Kyousei Tamura
Samejima Mutsumi
Masahiro Nitta
Kure Hidenori