The benzo Okisabo roll derivative for bacterial infection medical treatment

Title:

The benzo Okisabo roll derivative for bacterial infection medical treatment

Document Type and Number:

Japanese Patent JP5952280

Kind Code:

B2

Abstract:

This invention relates to benzoxaborole compounds for formula (I) wherein R 3 is -CH 2 NH 2 ; R 4 is selected from the group consisting of halogen, methyl, ethyl, propyl, isopropyl, butyl, isobutyl, sec-butyl, methoxy, ethoxy, propoxy, isopropoxy, butoxy, isobutoxy, and sec-butoxy; Y is O; and R 5 is -(CH 2 ) a -R 12 wherein a is 2,3 or 4; and R 12 is selected from the group consisting of H, OH, NH 2 , methyl, ethyl, -NHS(O) 2 CH 3 , cyano, -NHC(O)CH 3 , -NHC(O)NHCH 2 CH 3 , -C(O)NH 2 , -C(O)OH, 4-(methoxy)phenyl, benzyl, benzoxy, -NHC(O)OCH 2 Ph, -C(O)NHCH 2 CH 2 OH and -C(NH 2 )(NH); or a salt, hydrate or solvate thereof, and their use for treating bacterial infections.

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Inventors:

Hernandez, Vincent, Es.
Ding, charles
Prattner, Jacob, J.
Ally, Michael Richard, Kevin
Rock, fernando
Chang, Suomin
Eason, Eric
Lee, Shan Feng
Butterfly, din

Application Number:

JP2013527375A

Publication Date:

July 13, 2016

Filing Date:

September 07, 2011

Export Citation:

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