Title:
【発明の名称】治療用化合物
Document Type and Number:
Japanese Patent JP2002501923
Kind Code:
A
Abstract:
This invention relates to novel structural analogues and derivatives of compounds with general analgesic or related pharmacological activity. In particular the invention relates to derivatives of opioid compounds, particularly morphine and related compounds, in which an opioid compound is linked via the nitrogen at position 17 to a spacer group, which in turn is linked to a charged group, or a pharmaceutically acceptable salt thereof. In particularly preferred embodiments the opioid compound is morphine, codeine, or buprenorphine.
Inventors:
Jackson, Roy, William
Sabasinfu, Kamani, Rupika
Baura, Alan, Lewis, Arthur
Sabasinfu, Kamani, Rupika
Baura, Alan, Lewis, Arthur
Application Number:
JP2000529336A
Publication Date:
January 22, 2002
Filing Date:
January 29, 1999
Export Citation:
Assignee:
Monash University
Polychip Pharmaceuticals Proprietary Limited
Polychip Pharmaceuticals Proprietary Limited
International Classes:
C07D221/26; A61K31/435; A61K31/445; A61K31/451; A61K31/472; A61K31/485; A61K47/48; A61P25/04; C07D211/32; C07D211/64; C07D221/28; C07D489/02; C07D489/04; C07D489/08; C07D489/12; (IPC1-7): C07D489/02; A61K31/435; A61K31/445; A61K31/472; A61K31/485; A61P25/04; C07D211/32; C07D211/64; C07D221/26; C07D221/28; C07D489/04; C07D489/08; C07D489/12
Attorney, Agent or Firm:
Akira Asamura (3 outside)