Title:
【発明の名称】癌治療において用いるためのグラニュラチミド誘導体
Document Type and Number:
Japanese Patent JP2002506868
Kind Code:
A
Abstract:
Novel granulatimide compounds and pharmaceutical formulations thereof are provided. Compounds of this invention have general formula (I) or (II) wherein are independently R or Z as defined below, or in combination F and F' is Ar1 as defined below; Ar1 is a monocyclic, bicyclic or tricyclic, fully or partially aromatic system containing five or six membered carbocyclic or, oxygen, nitrogen or sulphur containing heterocyclic rings, optionally substituted with R or Z; W is selected from the group consisting of formula (i); (ii) or (iii), wherein the structures are as described in: (i), (ii) and (iii). R and Z are optional substituents as defined in the application.
Inventors:
Anderson Raymond Jay.
Loberge michel
Sangella Justin Binder
Render
Pierce edward
Berlink Robert G. S.
Brighton robert
Loberge michel
Sangella Justin Binder
Render
Pierce edward
Berlink Robert G. S.
Brighton robert
Application Number:
JP2000536717A
Publication Date:
March 05, 2002
Filing Date:
March 11, 1999
Export Citation:
Assignee:
The University of British Columbia
Kinetech Pharmaceuticals, Inc.
Kinetech Pharmaceuticals, Inc.
International Classes:
A61K31/4188; A61K31/437; A61K31/553; A61K31/7042; A61K31/7052; A61K31/7056; A61P35/00; A61P43/00; C07D471/22; C07D487/04; C07D487/14; C07D487/22; C07D498/22; C07H9/06; C07H19/044; C07H19/23; (IPC1-7): C07D487/14; A61K31/4188; A61K31/437; A61K31/553; A61K31/7056; A61P35/00; A61P43/00; C07D471/22; C07D487/04; C07D487/22; C07D498/22; C07H19/23
Foreign References:
| WO1996011933A1 | 1996-04-25 | |||
| WO1996011933A1 | 1996-04-25 |
Other References:
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Attorney, Agent or Firm:
Shimizu Hatsushi (1 person outside)