Title:
抗菌薬および抗菌薬関連化合物の高透過性組成物またはプロドラッグ
Document Type and Number:
Japanese Patent JP2012529443
Kind Code:
A
Abstract:
High penetration comp1ositions (HPCs) or prodrugs (HPPs) of antimicrobials and antimicrobial-related compounds are provided. The HPCs/HPPs are capable of being converted to parent drugs or drug metabolites after crossing the biological barrier and thus can render treatments. Additionally, the HPCs/HPPs are capable of reaching areas that their parent drugs may not be able to access and rendering a sufficient concentration at the target areas and therefore render novel treatments.
Inventors:
You Chongshi
Shurina
Chen Yu Hua
Yang Bing Bing
Two Sea Cheung
Shurina
Chen Yu Hua
Yang Bing Bing
Two Sea Cheung
Application Number:
JP2012514336A
Publication Date:
November 22, 2012
Filing Date:
June 10, 2010
Export Citation:
Assignee:
Techfields Biochem Company Limited
International Classes:
C07D213/76; A61K31/429; A61K31/43; A61K31/431; A61K31/545; A61K31/546; A61K47/48; A61K49/00; A61P33/04; A61P33/10; A61P33/12; A61P43/00; C07D215/56; C07D471/04; C07D498/04; C07D499/46; C07D499/60; C07D499/62; C07D499/64; C07D499/86; C07D499/88; C07D499/897; C07D501/22; C07D501/34; C07D501/36; C07D501/59; C07F9/40; C07F9/6558
Domestic Patent References:
| JP2012511027A | 2012-05-17 | |||
| JPS52153992A | 1977-12-21 | |||
| JPS5419993A | 1979-02-15 | |||
| JP2012511027A | 2012-05-17 |
Foreign References:
| WO2008072032A1 | 2008-06-19 |
Other References:
JPN6014026636; Ｃｈｅｍｉｃａｌ Ａｂｓｔｒａｃｔｓ ６１：３３９３６
JPN6014026639; Ｄｅｒｍａｔｏｌｏｇｉｃａ （１９６７）， １３４（３）， １２９-３４
JPN6014026639; Ｄｅｒｍａｔｏｌｏｇｉｃａ （１９６７）， １３４（３）， １２９-３４
Attorney, Agent or Firm:
Koichi Tsujii
Sadao Kumakura
Atsushi Hakoda
Kenji Asai
Kazuo Yamazaki
Satsuki Ichikawa
Shimura
Sadao Kumakura
Atsushi Hakoda
Kenji Asai
Kazuo Yamazaki
Satsuki Ichikawa
Shimura