バイオアベイラビリティが高いアルボシジブプロドラッグ

Title:

バイオアベイラビリティが高いアルボシジブプロドラッグ

Document Type and Number:

Japanese Patent JP7133680

Kind Code:

B2

Abstract:

Compounds having the following structure (I):or a stereoisomer, tautomer or pharmaceutically acceptable salt thereof, wherein one of R¹, R² or R³ is -P(=O)(OH)₂, and the other two of R¹, R² and R³ are each H, are provided. Pharmaceutical compositions comprising the compounds, and methods for use of the compounds for treating diseases associated with overexpression of a cyclin-dependent kinase (CDK) are also provided.

More Like This:

JP5313883	Nitrogen-containing condensed ring derivative, pharmaceutical composition containing it, and its pharmaceutical use
JP2022009127	PRODRUG COMPOUND AND APPLICATION THEREOF
WO/2023/183618	PSYCHEDELIC COMPOSITIONS AND METHODS FOR FORMING THE SAME

Inventors:

Adam Siddiqui-Jane
David J. Bearth

Application Number:

JP2021079708A

Publication Date:

September 08, 2022

Filing Date:

May 10, 2021

Export Citation:

Click for automatic bibliography generation Help

Assignee:

Sumitomo Pharma Oncology, Incorporated

International Classes:

A61K31/675; A61K9/20; A61K9/48; A61K45/00; A61K47/04; A61K47/12; A61K47/26; A61K47/38; A61P35/00; A61P35/02; A61P43/00

Domestic Patent References:

JP2004529125A

Foreign References:

WO2006101846A1

Attorney, Agent or Firm:

Shusaku Yamamoto
Morishita Natsuki
Takatoshi Iida
Daisuke Ishikawa
Kensaku Yamamoto

Previous Patent: game machine

Next Patent: Lighting device, sensor unit, reading device and image forming device