Login| Sign Up| Help| Contact|

Patent Searching and Data


Title:
【発明の名称】プロテアーゼ阻害剤としての新規化合物及び組成物
Document Type and Number:
Japanese Patent JP2002539191
Kind Code:
A
Abstract:
The present invention relates to novel N-cyanomethyl amides which are cysteine protease inhibitors, the pharmaceutically acceptable salts and N-oxides thereof, their uses as therapeutic agents and the methods of their making.

Inventors:
Bryant, Clifford M.
Banin, Barley A.
Clinac, Erica A.
Patterson, John W.
Application Number:
JP2000605556A
Publication Date:
November 19, 2002
Filing Date:
March 15, 2000
Export Citation:
Click for automatic bibliography generation   Help
Assignee:
AXYS PHARMACEUTICALS, INC.
International Classes:
A61K31/275; A61K31/277; A61K31/341; A61K31/343; A61K31/36; A61K31/381; A61K31/395; A61K31/40; A61K31/404; A61K31/4045; A61K31/4164; A61K31/4166; A61K31/417; A61K31/426; A61K31/433; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4436; A61K31/4439; A61K31/445; A61K31/4453; A61K31/4468; A61K31/454; A61K31/455; A61K31/465; A61K31/47; A61K31/495; A61K31/496; A61K31/505; A61K31/535; A61K31/5375; A61K31/54; A61K31/663; A61K45/00; A61P3/10; A61P5/14; A61P9/00; A61P9/10; A61P11/00; A61P11/06; A61P17/00; A61P17/02; A61P19/02; A61P19/10; A61P21/04; A61P25/00; A61P25/28; A61P27/02; A61P29/00; A61P33/00; A61P35/00; A61P37/00; A61P37/02; A61P37/08; A61P43/00; C07C253/30; C07C255/29; C07C255/60; C07C269/06; C07C271/22; C07C273/18; C07C275/24; C07C303/40; C07C311/06; C07C311/09; C07C315/04; C07C317/50; C07C319/20; C07C323/52; C07C323/60; C07C323/62; C07D207/09; C07D207/14; C07D207/16; C07D209/06; C07D209/08; C07D209/14; C07D209/22; C07D209/26; C07D209/42; C07D209/52; C07D211/58; C07D211/60; C07D211/62; C07D213/30; C07D213/34; C07D213/40; C07D213/56; C07D295/12; C07D213/70; C07D213/71; C07D213/75; C07D213/81; C07D213/82; C07D215/54; C07D233/24; C07D233/26; C07D233/64; C07D233/90; C07D239/28; C07D239/36; C07D277/20; C07D277/28; C07D277/30; C07D277/42; C07D277/48; C07D277/56; C07D285/135; C07D295/14; C07D295/155; C07D295/18; C07D295/20; C07D295/215; C07D307/56; C07D307/68; C07D317/68; C07D333/20; C07D333/38; C07D333/68; C07D401/12; C07D405/06; C07D405/12; C07D409/04; C07D417/04; C07D417/12; (IPC1-7): C07C255/29; A61K31/277; A61K31/341; A61K31/343; A61K31/36; A61K31/381; A61K31/40; A61K31/404; A61K31/4045; A61K31/4164; A61K31/417; A61K31/426; A61K31/433; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4436; A61K31/445; A61K31/4453; A61K31/455; A61K31/47; A61K31/495; A61K31/496; A61K31/505; A61K31/535; A61K31/5375; A61K31/54; A61P3/10; A61P5/14; A61P9/00; A61P9/10; A61P11/00; A61P11/06; A61P17/02; A61P19/02; A61P21/04; A61P25/28; A61P27/02; A61P29/00; A61P37/02; A61P37/08; A61P43/00; C07C253/30; C07C269/06; C07C271/22; C07C273/18; C07C275/24; C07C303/40; C07C311/06; C07C315/04; C07C317/50; C07C319/20; C07C323/52; C07C323/60; C07C323/62; C07D207/14; C07D209/08; C07D209/14; C07D209/22; C07D209/42; C07D213/34; C07D213/40; C07D213/56; C07D213/71; C07D213/81; C07D213/82; C07D215/54; C07D233/64; C07D233/90; C07D239/36; C07D277/28; C07D277/42; C07D277/56; C07D285/135; C07D295/12; C07D295/18; C07D295/20; C07D307/56; C07D307/68; C07D317/68; C07D333/20; C07D333/38; C07D333/68; C07D401/12; C07D405/06; C07D405/12; C07D409/04
Foreign References:
WO1998001133A11998-01-15
Attorney, Agent or Firm:
Takashi Ishida (4 others)