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Title:
医薬物質としての新規ピロール誘導体
Document Type and Number:
Japanese Patent JP2004535404
Kind Code:
A
Abstract:
Novel pyrrazole derivative compounds and their use as pharmaceutical agents, in particular their use as TGF-beta signal transduction inhibitors. The disclosed invention relates to compounds of the structure (I) wherein (I) is a four, five, or six membered saturated ring and X is C, O or S

Inventors:
Jason Scott Sawyer
Douglas Wade Bait
Paola Cappetti
Todd vincent decoro
Alexander Glen Godfrey
Theodore Goodson Jr.
David Kent Heron
Lee Hong-You
Liao Junkai
William Thomas McMillen
Sean Christopher Miller
Nicholas Anthony Mort
Jonathan Michael Ingling
Edward Sea Earl Smith
Application Number:
JP2002591506A
Publication Date:
November 25, 2004
Filing Date:
May 13, 2002
Export Citation:
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Assignee:
ELI LILLY AND COMPANY
International Classes:
A61K31/4439; A61K31/444; A61K31/4709; A61K31/496; A61K31/5383; A61K31/55; A61K45/00; A61P3/10; A61P7/04; A61P9/10; A61P13/12; A61P17/02; A61P17/12; A61P19/02; A61P21/02; A61P25/28; A61P27/02; A61P29/00; A61P31/00; A61P31/18; A61P35/00; A61P37/02; A61P37/08; A61P43/00; C07D401/12; C07D471/04; C07D487/04; C07D498/04; (IPC1-7): C07D471/04; A61K31/4439; A61K31/444; A61K31/4709; A61K31/496; A61K31/5383; A61K31/55; A61K45/00; A61P3/10; A61P9/10; A61P13/12; A61P17/02; A61P17/12; A61P19/02; A61P21/02; A61P25/28; A61P27/02; A61P29/00; A61P31/18; A61P35/00; A61P37/02; A61P37/08; A61P43/00; C07D401/12; C07D487/04; C07D498/04
Foreign References:
WO2001016138A12001-03-08
Attorney, Agent or Firm:
Kyousei Tamura
Hiromitsu Takayama
Minato Saito