Title:
S1P1受容体アゴニストとしての新規ジカルボン酸誘導体
Document Type and Number:
Japanese Patent JP5346016
Kind Code:
B2
Abstract:
The present invention provides a novel class of 3-phenyl or 5-phenyl-1,2,4-oxadiazole based dicarboxylic acid derivatives useful as S1P1 receptor agonists, their process of preparation and their therapeutic use.
Inventors:
Marc Cape
Nicolas Levoin
Isabel Belbi-Bertrand
Philip Robert
Jean-Charles Schwartz
Jeanne-Marie Lecomte
Giraj Dirip by Aradier
Mutukumaran Natarajan Pilai
Bavesh Mohanbai Panchal
Jignes Cantilal Zivani
Biswagit Samantha
Ranjan Kumar Pal
Raja Mannar Sennaty
Nicolas Levoin
Isabel Belbi-Bertrand
Philip Robert
Jean-Charles Schwartz
Jeanne-Marie Lecomte
Giraj Dirip by Aradier
Mutukumaran Natarajan Pilai
Bavesh Mohanbai Panchal
Jignes Cantilal Zivani
Biswagit Samantha
Ranjan Kumar Pal
Raja Mannar Sennaty
Application Number:
JP2010511664A
Publication Date:
November 20, 2013
Filing Date:
June 16, 2008
Export Citation:
Assignee:
Biopologue
Sun Pharma Advanced Research Company Limited
Sun Pharma Advanced Research Company Limited
International Classes:
C07D271/06; A61K31/4245; A61K31/454; A61K31/4545; A61K31/5377; A61P1/04; A61P3/10; A61P9/00; A61P9/08; A61P9/10; A61P11/00; A61P11/02; A61P11/06; A61P11/16; A61P13/12; A61P17/00; A61P17/06; A61P19/02; A61P21/00; A61P25/00; A61P25/28; A61P29/00; A61P31/04; A61P31/12; A61P31/14; A61P31/16; A61P35/00; A61P35/02; A61P37/02; A61P37/06; A61P37/08; A61P43/00; C07D413/10; C07D413/14
Foreign References:
| WO2006043149A1 | ||||
| WO2004035538A1 |
Other References:
Journal of Medicinal Chemistry,2005年,Vol.48,No.20,P.6169-6173
J. Med. Chem.,2004年,Vol.47,No.27,P.6662-6665
J. Med. Chem.,2004年,Vol.47,No.27,P.6662-6665
Attorney, Agent or Firm:
Yasuhiko Murayama
Masatake Shiga
Takashi Watanabe
Shinya Mitsuhiro
Masatake Shiga
Takashi Watanabe
Shinya Mitsuhiro