Login| Sign Up| Help| Contact|

Patent Searching and Data


Title:
インドール誘導体を含む殺寄生虫性組成物、寄生虫駆除方法及びこれらの使用
Document Type and Number:
Japanese Patent JP2017518352
Kind Code:
A
Abstract:
本発明は少なくとも一種のインドール誘導体活性薬剤を含む、哺乳類の肝吸虫寄生虫と闘うための経口、局所又は注射可能な組成物に関する。また、本発明は必要とする哺乳類に本発明の組成物を投与することを含む哺乳類の肝吸虫寄生虫感染症及び外寄生を撲滅し、抑制するための改良された方法を提供する。

Inventors:
Meng Charles
Le Healed Farois Royce
Application Number:
JP2016574080A
Publication Date:
July 06, 2017
Filing Date:
June 19, 2015
Export Citation:
Click for automatic bibliography generation   Help
Assignee:
Merial Incorporated
International Classes:
C07D209/10; A61K31/277; A61K31/365; A61K31/404; A61K31/4439; A61K45/00; A61P33/14; C07D401/04; C07D401/12; H03K5/04; H03K7/00
Domestic Patent References:
JPH08119807A1996-05-14
JP2008037760A2008-02-21
JP2013511475A2013-04-04
JP2012507534A2012-03-29
JP2004505965A2004-02-26
JP2014500332A2014-01-09
JP2011521961A2011-07-28
JP2005518351A2005-06-23
Foreign References:
WO2002016348A12002-02-28
WO2008050207A12008-05-02
WO2013158894A12013-10-24
US20100033088A12010-02-11
DE19515371A11995-11-02
FR1446368A1966-07-22
CN102153544A2011-08-17
WO2012088431A12012-06-28
Other References:
JOHN F POLETTO: "SYNTHESIS AND ANTIINFLAMMATORY EVALUATION OF CERTAIN 5-ALKOXY-2,7-DIALKYLTRYPTAMINES", JOURNAL OF MEDICINAL CHEMISTRY, vol. VOL:16, NR:7, JPN5017005189, July 1973 (1973-07-01), pages 757 - 765, ISSN: 0003959605
CONDE J J: "TOWARDS THE SYNTHESIS OF OSTEOCLAST INHIBITOR SB-242784", TETRAHEDRON LET, vol. VOL:44, NR:15, JPN5017005190, 7 April 2003 (2003-04-07), GB, pages 3081 - 3084, ISSN: 0003959606
WANG: "FLUORINATED N-[2-(HALOALKYL)PHENYL]IMIDOYL CHLORIDE, A KEY INTERMEDIATE FOR THE SYNTHESIS 以下備考", JOURNAL OF FLUORINE CHEMISTRY, vol. VOL:128, NR:10, JPN5017005192, 1 October 2007 (2007-10-01), NL, pages 1143 - 1152, ISSN: 0003959607
HONG X: "PHOTODESULFONYLATION OF INDOLES INITIATED BY ELECTRON TRANSFER FROM TRIETHYLAMINE", TETRAHEDRON LETTERS, vol. VOL:47, NR:14, JPN5017005194, 3 April 2006 (2006-04-03), GB, pages 2409 - 2412, ISSN: 0003959608
CAN ZHU: "COUPLING AND CYCLIZATION OF O -IODOANILINES AND PROPARGYLIC BROMIDES VIA ALLENES: AN 以下備考", ORGANIC LETTERS, vol. VOL:15, NR:11, JPN5017005196, 7 June 2013 (2013-06-07), pages 2782 - 2785, ISSN: 0003959609
LARISA V POLITANSKAYA: "SYNTHESIS OF INDOLES WITH A POLYFLUORINATED BENZENE RING", TETRAHEDRON, vol. VOL:69, NR:39, JPN5017005198, 17 July 2013 (2013-07-17), pages 8477 - 8486, ISSN: 0003959610
TETRAHEDRON LETT., vol. 45, JPN6019001353, 2004, pages 1857 - 1859, ISSN: 0003959611
ELECTROCHIMICA ACTA., vol. 29, JPN6019001355, 1984, pages 1075 - 1082, ISSN: 0003959612
HETEROCYCLES, vol. 86, JPN6019001356, 2012, pages 979 - 983, ISSN: 0003959613
QUIM. NOVA, vol. 35, JPN6019001358, 2012, pages 1157 - 1163, ISSN: 0003959614
Attorney, Agent or Firm:
Takaki Nishijima
Disciple Maru Ken
Shinichiro Tanaka
Atsushi Hakoda
Kenji Asai
Kazuo Yamazaki
Satsuki Ichikawa
Hironobu Hattori
Kobayashi Machiko