Title:
Method for preparing 4-amino-1-((1S, 4R, 5S) -2-fluoro-4,5-dihydroxy-3-hydroxymethyl-cyclopent-2-enyl) -1H-pyrimidine-2-one
Document Type and Number:
Japanese Patent JP6334676
Kind Code:
B2
Abstract:
Processes for the preparation of 4-amino-1-((1S,4R,5S)-2-fluoro-4,5-dihydroxy-3-hydroxymethyl-cyclopent-2-enyl)-1H-pyrimidin-2-one (13, RX-3117) and its intermediates are described.
Inventors:
Hai Phong Inn
Theog Jun Kim
Eriezer Farb
Ray Andre Pearcy
Jonathan Cummins
Petra Dietrich
Jean-Francois Carnot
E one
Bikram Chandrakant Purochit
Theog Jun Kim
Eriezer Farb
Ray Andre Pearcy
Jonathan Cummins
Petra Dietrich
Jean-Francois Carnot
E one
Bikram Chandrakant Purochit
Application Number:
JP2016503433A
Publication Date:
May 30, 2018
Filing Date:
March 17, 2014
Export Citation:
Assignee:
Lexan Pharmaceuticals, Inc.
International Classes:
C07D317/44; C07D239/47; C07D317/20; C07D317/26; C07D405/04; C07H9/04
Domestic Patent References:
JP2007531736A |
Attorney, Agent or Firm:
Patent Business Corporation Tani/Abe Patent Office
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