The use for treating and preventing heterocyclic carbonyl aminothiazole, the object for makeup containing it or the tablet for dermatology, and the pigmentation of the skin which is not desirable

Japanese Patent JP6045593

B2

The invention relates to heterocyclocarbonylaminothiazoles of general formula (I), wherein R 1 = -morpholino, -piperidin-1-yl, -piperazin-1-yl, -((4-alkyl)-piperazin-1-yl), -pyrrolidinyl, -(1H-pyrrol-1-yl), -azetidin-1-yl, -azepan-1-yl, -2,3,4,5-tetrahydro-1-H-azepin-1-yl, -2,3-dihydro-1H-azepin-1-yl, -1H-azepin-1-yl, -tetrahydro-2H-pyran-4-yl, -4H-pyran-4-yl, -2H-pyran-4-yl, -oxepanyl, -dioxanyl, -tetrahydrofuranyl, -pyrrazolyl. The invention further relates to cosmetic or dermatological preparations having an effective content of one or more heteroalkylamidothiazoles and to the use thereof for the cosmetic or dermatological treatment and/or prophylaxis of undesired skin pigmentation.

Kolbe, Rutger
Catherner, Katrin

JP2014531200A

December 14, 2016

September 18, 2012

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Beiersdorf AG

C07D277/48; A61K8/49; A61K31/427; A61K31/454; A61K31/496; A61K31/5377; A61P17/00; A61Q19/02; C07D417/12

JP2007531740A
JP2007504255A
JP2004521871A
JP54154764A
JP2009503107A
JP2009537473A
JP2008508352A
JP7502014A

WO2005007151A1
WO2003015778A1
US20060003968
WO2011117034A1

Biochemical Journal,2011年,438(1),53-62
Tetrahedron Letters,2011年,52(26),3298-3302
International Journal of Pharmacy and Pharmaceutical Sciences,2011年,3(Suppl. 3),120-125
Journal of Medicinal Chemistry,2009年,52(6),1757-1767
Journal of Chemical Research, Synopses,2002年,(12),598-600

Einzel Felix-Reinhard
Junichi Maekawa
Hiroyasu Ninomiya
Ueshima

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