Title:
4-METHYL-1H-DIARYL PYRAZOLE DERIVATIVES AND THEIR USES AS MEDICAMENT
Document Type and Number:
WIPO Patent Application WO/2007/121687
Kind Code:
A1
Abstract:
The present application discloses 4-methyl-1H-diaryl pyrazole derivatives of
formula (I), their preparation methods, pharmaceutical compositions containing the
same which are used as cannabinoid receptors type I(CB1) inhibitors in brain especially
useful of treatment of obesity,ameliorating memory or stopping smoking.
Inventors:
LI, Song (N0.27, Taiping RoadHaidian District, Beijing 0, 100850, CN)
李松 (中国北京市海淀区太平路27号, Beijing 0, 100850, CN)
LIU, Mengjia (N0.27, Taiping RoadHaidian District, Beijing 0, 100850, CN)
刘梦佳 (中国北京市海淀区太平路27号, Beijing 0, 100850, CN)
李松 (中国北京市海淀区太平路27号, Beijing 0, 100850, CN)
LIU, Mengjia (N0.27, Taiping RoadHaidian District, Beijing 0, 100850, CN)
刘梦佳 (中国北京市海淀区太平路27号, Beijing 0, 100850, CN)
Application Number:
CN2007/001404
Publication Date:
November 01, 2007
Filing Date:
April 26, 2007
Export Citation:
Assignee:
INSTITUTE OF PHARMACOLOGY AND TOXICOLOGY ACADEMY OF MILITARY MEDICAL SCIENCES P.L.A. CHINA (N0.27, Taiping RoadHaidian District, Beijing 0, 100850, CN)
中国人民解放军军事医学科学院毒物药物研究所 (中国北京市海淀区太平路27号, Beijing 0, 100850, CN)
LI, Song (N0.27, Taiping RoadHaidian District, Beijing 0, 100850, CN)
李松 (中国北京市海淀区太平路27号, Beijing 0, 100850, CN)
LIU, Mengjia (N0.27, Taiping RoadHaidian District, Beijing 0, 100850, CN)
中国人民解放军军事医学科学院毒物药物研究所 (中国北京市海淀区太平路27号, Beijing 0, 100850, CN)
LI, Song (N0.27, Taiping RoadHaidian District, Beijing 0, 100850, CN)
李松 (中国北京市海淀区太平路27号, Beijing 0, 100850, CN)
LIU, Mengjia (N0.27, Taiping RoadHaidian District, Beijing 0, 100850, CN)
International Classes:
C07D231/14; A61K31/415; A61K31/4152; A61P3/04; A61P25/28; A61P25/34; C07D401/12; C07D403/12; C07D405/12; C07D409/12
Attorney, Agent or Firm:
CCPIT PATENT AND TRADEMARK LAW OFFICE (8/F Vantone New World Plaza, 2 Fuchengmenwai Street, Beijing 7, 100037, CN)
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