Title:
5,8-DIHYDRO-1,7-NAPHTHYRIDINE DERIVATIVES AS GLP-1 AGONISTS FOR THE TREATMENT OF DIABETES
Document Type and Number:
WIPO Patent Application WO/2023/179542
Kind Code:
A1
Abstract:
The present disclosure relates generally to GLP-1 agonists and pharmaceutical compositions comprising the same, as well as methods for treating a GLP-1 associated disease, disorder, or condition.
Inventors:
LEI HUI (CN)
LIN XICHEN (CN)
MENG QINGHUA (CN)
ZHANG HAIZHEN (CN)
LIN XICHEN (CN)
MENG QINGHUA (CN)
ZHANG HAIZHEN (CN)
Application Number:
PCT/CN2023/082518
Publication Date:
September 28, 2023
Filing Date:
March 20, 2023
Export Citation:
Assignee:
GASHERBRUM BIO INC (US)
LEI HUI (CN)
LEI HUI (CN)
International Classes:
A61K31/4375; C07D471/04; A61P3/10
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"Pharmaceutical Preformulation and Formulation", 2009, THE PHARMACEUTICAL PRESS AND THE AMERICAN PHARMACEUTICAL ASSOCIATION
"Handbook of Pharmaceutical Additives", 2007, GOWER PUBLISHING COMPANY
SKELLY ET AL., J HEPATOL, vol. 1-2, 2001, pages 195 - 9
CHITTURI ET AL., HEPATOLOGY, vol. 35, no. 2, 2002, pages 373 - 9
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BERHMAN REKLIEGMAN RARVIN AMNELSON WE: "Nelson Textbook of Pediatrics", 1996, W.B. SAUNDERS COMPANY
RUDOLPH AM ET AL.: "Rudolph's Pediatrics", 2002, MCGRAW-HILL
AVERY MDFIRST LR: "Pediatric Medicine", 1994, WILLIAMS & WILKINS
T. W. GREENEG. M. WUTS: "Protecting Groups in Organic Synthesis", 1999, WILEY
"Fieser and Fieser's Reagents for Organic Synthesis", vol. 1-40, 1991, JOHN WILEY, AND SONS
"Larock's Comprehensive Organic Transformations", vol. 1-5, 1989, ELSEVIER SCIENCE PUBLISHERS
"March's Advanced Organic Chemistry", 2001, JOHN WILEY, AND SONS
Attorney, Agent or Firm:
WU , FENG & ZHANG (CN)
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