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Title:
ALKYLIDENE DERIVATIVES AS KRAS INHIBITORS
Document Type and Number:
WIPO Patent Application WO/2023/284730
Kind Code:
A1
Abstract:
The present disclosure provides certain alkylidenyl derivatives that inhibit certain K-Ras proteins and are therefore useful for the treatment of cancers mediated by such proteins. Also provided are pharmaceutical compositions containing such compounds and processes for preparing such compounds. 114342739v.1

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Inventors:
FU JIPING (US)
LOU YAN (US)
SUN YONGFENG (CN)
Application Number:
PCT/CN2022/105169
Publication Date:
January 19, 2023
Filing Date:
July 12, 2022
Export Citation:
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Assignee:
NIKANG THERAPEUTICS INC (US)
SHANGHAI BLUERAY BIOPHARMA CO LTD (CN)
International Classes:
C07D519/00; A61K31/519; A61P35/00
Domestic Patent References:
WO2021041671A12021-03-04
WO2020146613A12020-07-16
WO2021106231A12021-06-03
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Attorney, Agent or Firm:
CHINA PATENT AGENT (H.K.) LTD. (CN)
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