Title:
AMINO ACID CONJUGATES PROVIDING FOR SUSTAINED SYSTEMIC CONCENTRATIONS OF GABA ANALOGUES
Document Type and Number:
WIPO Patent Application WO2002100344
Kind Code:
A3
Abstract:
This invention is directed to compounds that provide for sustained systemic concentrations of GABA analogs following administration to animals. This invention is also directed to pharmaceutical compositions including and methods using such compounds.
More Like This:
Inventors:
GALLOP MARK A (US)
CUNDY KENNETH C (US)
SCHEUERMAN RANDALL A (US)
BARRETT RONALD W (US)
ZERANGUE NOA (US)
CUNDY KENNETH C (US)
SCHEUERMAN RANDALL A (US)
BARRETT RONALD W (US)
ZERANGUE NOA (US)
Application Number:
PCT/US2002/018493
Publication Date:
February 12, 2004
Filing Date:
June 11, 2002
Export Citation:
Assignee:
XENOPORT INC (US)
GALLOP MARK A (US)
CUNDY KENNETH C (US)
SCHEUERMAN RANDALL A (US)
BARRETT RONALD W (US)
ZERANGUE NOA (US)
GALLOP MARK A (US)
CUNDY KENNETH C (US)
SCHEUERMAN RANDALL A (US)
BARRETT RONALD W (US)
ZERANGUE NOA (US)
International Classes:
C07D295/18; A61K31/197; A61K31/198; A61K31/275; A61K31/381; A61K31/40; A61K31/426; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4453; A61K31/4458; A61K31/47; A61K47/48; A61P1/00; A61P25/00; A61P25/04; A61P25/08; A61P25/18; A61P25/20; A61P25/22; A61P25/24; A61P25/28; A61P25/32; A61P29/00; A61P43/00; C07C237/12; C07C237/20; C07C237/24; C07C255/58; C07C317/50; C07C323/59; C07C323/60; C07D207/16; C07D211/60; C07D213/53; C07D213/56; C07D215/12; C07D229/02; C07D233/54; C07D277/20; C07D277/30; C07D333/24; C07D333/60; C07K5/02; G01N33/566; A61K38/00; (IPC1-7): C07C261/00
Foreign References:
| US6342529B1 | 2002-01-29 | |||
| US6140366A | 2000-10-31 | |||
| US6255345B1 | 2001-07-03 | |||
| US6291526B1 | 2001-09-18 |
Other References:
See also references of EP 1412324A4
Download PDF: