ANTIFUNGAL 1, 2, 4-TRIAZOLYL DERIVATIVES

Description

The present invention relates to novel triazole compounds of the formulae I and Il as defined below which carry a sulfur substituent, to agricultural compositions containing them, to their use as fungicides and to intermediate compounds used in the method of producing them.

The control of plant diseases caused by phythopathogenic fungi is extremely important for achieving high crop efficiency. Plant disease damage to ornamental, vegetable, field, cereal, and fruit crops can cause significant reduction in productivity and thereby result in increased costs to the consumer.

DE 19528046, DE 19529089, DE 19528300, DE 19617461 , DE 19617282, DE

19620407, DE 19620590, WO96/16048 and WO 97/43269 describe sulfurized triazolyl derivatives. The compounds are used for combating harmful fungi.

There is a continuous need for new compounds which are more effective, less costly, less toxic, environmentally safer and/or have different modes of action.

Accordingly, it is an object of the present invention to provide compounds having a better fungicidal activity and/or a better crop plant compatibility.

Surprisingly, these objects are achieved by triazole compounds of the general formulae I and II, defined below, and by the agriculturally acceptable salts of the compounds I and II.

Accordingly, the present invention relates to triazole compounds of the formulae I and Il and to agriculturally useful salts thereof

5a

R

(I) (H)

wherein R ¹ is group of formula V or

(V) (Vl) wherein

# is the attachment point to the remainder of the molecule;

A is a linear d-Cs-alkylene bridge which may be substituted by 1 , 2, 3 or 4 sub- stituents R ⁶ ;

R ² is aryl which may carry 1 , 2, 3, 4 or 5 substituents R ⁷ , or is a 5- or 6-membered heteroaromatic ring containing 1 , 2 or 3 heteroatoms selected from N, O and S as ring members, where the heteroaromatic ring may carry 1 , 2, 3 or 4 substituents R ⁸ ;

R ³ is selected from Ci-Cio-alkyl which may carry 1 or 2 substituents R ⁹ , C1-C10- haloalkyl which may carry 1 or 2 substituents R ⁹ , Cs-Cs-cycloalkyl, C3-C8- cycloalkyl-Ci-C4-alkyl, where the cycloalkyl moiety in the 2 last-mentioned radicals may carry 1 , 2, 3 or 4 substituents R ¹⁰ , aryl and aryl-Ci-C4-alkyl, where the aryl moiety in the 2 last-mentioned radicals may carry 1 , 2, 3, 4 or 5 substituents R ¹¹ ;

R ⁴ is hydrogen, OH or CN;

R ⁵ is selected from hydrogen, Ci-Cio-alkyl, Ci-Cio-haloalkyl, C2-Cio-alkenyl, C2-C10- haloalkenyl, C2-Cio-alkynyl, C2-Cio-haloalkynyl, C3-Cio-cycloalkyl, C3-C10- halocycloalkyl, phenyl, phenyl-Ci-C4-alkyl, where the phenyl moiety in the 2 last- mentioned radicals may carry 1 , 2, 3, 4 or 5 substituents R ¹² , and a 5- or 6- membered saturated, partially unsaturated or aromatic heterocyclic ring containing 1 , 2 or 3 heteroatoms selected from N, O and S as ring members, where the heterocyclic ring may carry 1 , 2 or 3 substituents R ¹² ; or, in case m is 0, may also be selected from -C(=O)R ¹³ , -C(=S)R ¹³ , -S(O) ₂ R ¹³ , -CN, -P(=Q)R ¹⁴ R ¹⁵ , M and a group of the formula III wherein

R ¹ is as defined for formulae I and II; and # is the attachment point to the remainder of the molecule;

R ^5a is selected from hydrogen, Ci-Cio-alkyl, Ci-Cio-haloalkyl, C2-Cio-alkenyl, C2-C10- haloalkenyl, C2-Cio-alkynyl, C2-Cio-haloalkynyl, C3-Cio-cycloalkyl, C3-C10- halocycloalkyl, phenyl, phenyl-Ci-C4-alkyl, where the phenyl moiety in the 2 last- mentioned radicals may carry 1 , 2, 3, 4 or 5 substituents R ¹² , a 5- or 6-membered saturated, partially unsaturated or aromatic heterocyclic ring containing 1 , 2 or 3 heteroatoms selected from N, O and S as ring members, where the heterocyclic ring may carry 1 , 2 or 3 substituents R ¹² , -C(=O)R ¹³ , -C(=S)R ¹³ , -S(O) ₂ R ¹³ , -CN, -P(=Q)R ¹⁴ R ¹⁵ and M;

each R ⁶ is independently selected from halogen, OH, SH, NR ¹⁶ R ¹⁷ , Ci-C ₄ -alkyl, Ci-C ₄ - haloalkyl, C2-C ₄ -alkenyl, C2-C ₄ -haloalkenyl, C2-C ₄ -alkynyl, C2-C ₄ -haloalkynyl, Ci- C ₄ -alkoxy, Ci-C ₄ -haloalkoxy, Ci-C ₄ -alkylthio and Ci-C ₄ -haloalkylthio, where the aliphatic moieties in the above radicals may carry 1 , 2 or 3 substituents R ¹⁸ ; or

two radicals R ⁶ bound on two adjacent carbon atoms, together with the carbon atoms to which they are bound, form a 3-, 4-, 5-, 6- or 7-membered saturated, partly unsaturated or maximum unsaturated carbocyclic ring or a 3-, 4-, 5-, 6- or 7-membered saturated, partly unsaturated or maximum unsaturated heterocyclic ring containing 1 , 2, or 3 heteroatoms selected from O, S and N as ring members, where the carbocyclic or heterocyclic ring may carry 1 , 2 or 3 substituents R ¹² ;

each R ⁷ is independently selected from halogen, nitro, CN, Ci-C ₄ -alkyl, Ci-C ₄ -haloalkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -haloalkoxy and NR ¹⁶ R ¹⁷ ;

each R ⁸ is independently selected from halogen, nitro, CN, Ci-C ₄ -alkyl, Ci-C ₄ -haloalkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -haloalkoxy and NR ¹⁶ R ¹⁷ ;

each R ⁹ is independently selected from nitro, CN, OH, SH, Si(R ²⁰ ) ₃ , NR ¹⁶ R ¹⁷ , CrC ₄ - alkoxy, Ci-C ₄ -haloalkoxy, Cs-Cβ-cycloalkyl, Cs-Cβ-halocycloalkyl and C3-C6- cycloaloxy; each R ¹⁰ is independently selected from halogen, nitro, CN, Ci-C4-alkyl, CrC ₄ - haloalkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -haloalkoxy and NR ¹⁶ R ¹⁷ ;

each R ¹¹ is independently selected from halogen, nitro, CN, Ci-C ₄ -alkyl, C1-C4- haloalkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -haloalkoxy and NR ¹⁶ R ¹⁷ ;

each R ¹² is independently selected from halogen, nitro, CN, Ci-C ₄ -alkyl, C1-C4- haloalkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -haloalkoxy and NR ¹⁶ R ¹⁷ ;

R ¹³ is selected from hydrogen, Ci-Cio-alkyl, Ci-Cio-haloalkyl, Ci-Cio-alkoxy, C1-C10- haloalkoxy, Ci-Cio-aminoalkyl, C3-Cio-cycloalkyl, C3-Cio-halocycloalkyl, phenyl, phenyl-Ci-C ₄ -alkyl, where the phenyl moiety in the 2 last-mentioned radicals may carry 1 , 2, 3, 4 or 5 substituents R ¹² , a 5- or 6-membered saturated, partially unsaturated or aromatic heterocyclic ring containing 1 , 2 or 3 heteroatoms selected from N, O and S as ring members, where the heterocyclic ring may carry 1 , 2 or 3 substituents R ¹² , and NR ¹⁶ R ¹⁷ ;

R ¹⁴ and R ¹⁵ , independently of each other, are selected from Ci-Cio-alkyl, Ci-Cio- haloalkyl, C2-Cio-alkenyl, C2-Cio-haloalkenyl, C2-Cio-alkynyl, C2-Cio-haloalkynyl, C3-Cio-cycloalkyl, C3-Cio-halocycloalkyl, Ci-Cio-alkoxy, Ci-Cio-haloalkoxy, C1-C4- alkoxy-Ci-Cio-alkyl, Ci-C4-alkoxy-Ci-Cio-alkoxy, Ci-Cio-alkylthio, C1-C10- haloalkylthio, C2-Cio-alkenyloxy, C2-Cio-alkenylthio, C2-Cio-alkynyloxy, C2-C10- alkynylthio, C3-Cio-cycloalkoxy, C3-Cio-cycloalkylthio, phenyl, phenyl-Ci-C ₄ -alkyl, phenylthio, phenyl-Ci-C ₄ -alkoxy, and NR ¹⁶ R ¹⁷ ;

each R ¹⁶ is independently selected from hydrogen and Ci-Cs-alkyl;

each R ¹⁷ is independently selected from hydrogen, Ci-Cs-alkyl, phenyl, and phenyl-Ci-

CU-alkyl;

or R ¹⁶ and R ¹⁷ together form a linear C ₄ - or Cs-alkylene bridge or a group -CH2CH2OCH2CH2- or -CH ₂ CH ₂ NR ¹⁹ CH ₂ CH ₂ -;

each R ¹⁸ is independently selected from nitro, CN, OH, SH, COR ¹³ , NR ¹⁶ R ¹⁷ , C ₃ -C ₆ - cycloalkyl, Cs-Cβ-halocycloalkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -haloalkoxy, C3-C6- cycloaloxy, phenyl and phenoxy;

each R ¹⁹ is independently selected from hydrogen and Ci-C ₄ -alkyl; each R ²⁰ is independently selected from d-Cε-alkyl, C-i-Cβ-haloalkyl, phenyl, phenyl- Ci-C4-alkyl, Ci-C4-alkoxy and Ci-C4-haloalkoxy;

Q is O or S;

M is a metal cation equivalent or an ammonium cation of formula (NR ^a R ^b R ^c R ^d ) ⁺ , wherein R ^a , R ^b , R ^c and R ^d , independently of each other, are selected from hydrogen, Ci-Cio-alkyl, phenyl and benzyl, where the phenyl moiety in the 2 last- mentioned radicals may carry 1 , 2 or 3 substituents independently selected from halogen, CN, nitro, Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy, Ci-C4-haloalkoxy and NR ¹⁶ R ¹⁷ ; and

m is 0, 1 , 2 or 3;

preferably with the proviso that R ² is not 2-fluorophenyl if R ³ is 4-fluorophenyl and R ⁴ is OH; with the proviso that R ³ is not 2-fluorophenyl if R ² is 4-fluorophenyl and R ⁴ is OH; with the proviso that R ³ is not n-butyl if R ² is 4-fluorophenyl, 2-chlorophenyl, 4- chlorophenyl, 2,4-dichlorophenyl, 4-bromophenyl, 4-tert-butylphenyl or 4-biphenyl and R ⁴ is CN; with the proviso that R ³ is not tert-butyl if R ² is 2-chlorophenyl, 4-chlorophenyl, 2,4- dichlorophenyl, 2,4,6-trichlorophenyl, 4-trifluoromethylphenyl or 2- difluoromethoxyphenyl and R ⁴ is CN; with the proviso that R ² is not 4-chlorophenyl if R ³ is 2-fluoromethylprop-2-yl, 1 ,3- difluoro-2-methylprop-2-yl, 4-chlorophenyl, 4-chlorophenyl-methyl, 4-chlorophenyl-1- ethyl, 4-chlorophenyl-2-ethyl or 4-fluorophenyl-2-ethyl and R ⁴ is CN; with the proviso that R ² is not 2,4-dichlorophenyl if R ³ is methyl, ethyl, propyl, isopropyl, n-butyl, sec-butyl, isobutyl, tert-butyl, 2,2,2-trifluoroethyl, pentafluoroethyl, trifluoro- methoxymethyl, 1 ,1-difluoroethoxymethyl, 1 ,1 ,2,2-tetrafluoroethoxymethyl, cyclopropyl, 1-chlorocyclopropyl, 1-fluorocyclopropyl, 1-cyclopropylethyl, cyclopentyl, cyclohexyl, cyclohexylmethyl, 4-fluorophenyl, 4-chlorophenyl, 4-fluorophenylmethyl or 4- chlorophenylmethyl and R ⁴ is H; with the proviso that R ³ is not n-propyl if R ² is 4-fluorophenyl, 2-chlorophenyl, 4- chlorophenyl, 2,4,6-trichlorophenyl, 4-methylphenyl, 4-trifluoromethylphenyl or 2- trifluoromethoxyphenyl and R ⁴ is H; with the proviso that R ³ is not 1 ,1 ,2,2-tetrafluoroethoxymethyl if R ² is 4-fluorophenyl, 2- chlorophenyl or 4-chlorophenyl and R ⁴ is H; with the proviso that R ² is not 2,4-dichlorophenyl if R ³ is n-butyl, R ⁴ is OH and R ⁵ is H, methyl or CN, preferably with the proviso that R ² is not 2,4-dichlorophenyl if R ³ is n- Butyl and R ⁴ is OH; with the proviso that in case R ¹ is a group Vl, R ² is not phenyl, 4-fluorophenyl, 2,4- difluorophenyl, 4-chlorophenyl, 2,4-dichlorophenyl, 2,4,6-trichlorophenyl, 4- trifluoromethylphenyl, 2-difluoromethoxyphenyl or 4-trifluoromethoxyphenyl.

The present invention also provides the use of triazole compounds of the formulae I and Il and/or their agriculturally useful salts for controlling harmful fungi.

The invention further provides fungicidal compositions comprising these triazole compounds of the formulae I and/or Il (and/or also of the formula IV; see below) and/or their agriculturally acceptable salts and suitable carriers. Suitable agriculturally acceptable carriers are described below.

The compounds I and Il can exist as one or more stereoisomers. The various stereoisomers include enantiomers, diastereomers, atropisomers and geometric isomers. One skilled in the art will appreciate that one stereoisomer may be more active and/or may exhibit beneficial effects when enriched relative to the other stereoisomer(s) or when separated from the other stereoisomer(s). Additionally, the skilled artisan knows how to separate, enrich, and/or to selectively prepare said stereoisomers. The compounds of the invention may be present as a mixture of stereoisomers, e.g. a racemate, individual stereoisomers, or as an optically active form.

Compounds I and Il can be understood as positional/double bond isomers of each other, at least in case the radicals R ⁵ /R ^5a are identical. In case R ⁵ (and of course also R ^5a ) is hydrogen, the respective compounds I and Il are tautomers.

Suitable agriculturally useful salts are especially the salts of those cations or the acid addition salts of those acids whose cations and anions, respectively, have no adverse effect on the fungicidal action of the compounds I and II. Thus, suitable cations are in particular the ions of the alkali metals, preferably sodium and potassium, of the alkaline earth metals, preferably calcium, magnesium and barium, and of the transition metals, preferably manganese, copper, zinc and iron, and also the ammonium ion which, if desired, may carry one to four Ci-C4-alkyl substituents and/or one phenyl or benzyl substituent, preferably diisopropylammonium, tetramethylammonium, tetrabutylammo- nium, trimethylbenzylammonium, furthermore phosphonium ions, sulfonium ions, preferably tri(Ci-C4-alkyl)sulfonium and sulfoxonium ions, preferably tri(Ci-C4-alkyl)sulf- oxonium. Anions of useful acid addition salts are primarily chloride, bromide, fluoride, hydrogen- sulfate, sulfate, dihydrogenphosphate, hydrogenphosphate, phosphate, nitrate, bicarbonate, carbonate, hexafluorosilicate, hexafluorophosphate, benzoate, and also the anions of Ci-C4-alkanoic acids, preferably formate, acetate, propionate and butyrate. They can be formed by reacting I or Il with an acid of the corresponding anion, preferably hydrochloric acid, hydrobromic acid, sulfuric acid, phosphoric acid or nitric acid.

In the definitions of the variables given in the formulae above, collective terms are used which are generally representative for the substituents in question. The term C _n -Cm indicates the number of carbon atoms possible in each case in the substituent or sub- stitutent moiety in question:

Halogen: fluorine, chlorine, bromine and iodine;

Alkyl and the alkyl moieties in alkoxy, alkoxyalkyl, alkoxyalkoxy, alkylcarbonyl, alkyl- thiocarbonyl, aminoalkyl, alkylamino, dialkylamino, alkylaminocarbonyl, dialkylamino- carbonyl, alkylthio, alkylsulfonyl and the like: saturated straight-chain or branched hydrocarbon radicals having 1 to 2 (Ci-C ₂ -alkyl), 2 or 3 (C ₂ -C ₃ -alkyl), 1 to 4 (Ci-C ₄ -alkyl), 1 to 6 (d-Ce-alkyl), 1 to 8 (Ci-C ₈ -alkyl) or 1 to 10 (Ci-Cio-alkyl) carbon atoms. C ₂ -C ₃ - Alkyl is ethyl, n-propyl or isopropyl. Ci-C ₂ -Alkyl is methyl or ethyl. CrC ₄ -AIkVl is methyl, ethyl, propyl, isopropyl, butyl, 1-methylpropyl (sec-butyl), 2-methylpropyl (isobutyl) or 1 ,1-dimethylethyl (tert-butyl). Ci-Cβ-Alkyl is additionally also, for example, pentyl, 1-methylbutyl, 2-methylbutyl, 3-methylbutyl, 2,2-dimethylpropyl, 1-ethylpropyl, 1 ,1-dimethylpropyl, 1 ,2-dimethylpropyl, hexyl, 1-methylpentyl, 2-methylpentyl,

3-methylpentyl, 4-methylpentyl, 1 ,1-dimethylbutyl, 1 ,2-dimethylbutyl, 1 ,3-dimethylbutyl, 2,2-dimethylbutyl, 2,3-dimethylbutyl, 3,3-dimethylbutyl, 1-ethylbutyl, 2-ethylbutyl, 1 ,1 ,2-trimethylpropyl, 1 ,2,2-trimethylpropyl, 1-ethyl-1-methylpropyl, or 1-ethyl-2- methylpropyl. d-Cs-Alkyl is additionally also, for example, heptyl, octyl, 2-ethylhexyl and positional isomers thereof. Ci-Cio-Alkyl is additionally also, for example, nonyl, decyl, 2-propyl heptyl, 3-propylheptyl and positional isomers thereof.

Haloalkyl: straight-chain or branched alkyl groups having 1 to 2 (Ci-C ₂ -haloalkyl), 1 to 3 (d-Cs-haloalkyl), 1 to 4 (Ci-C ₄ -haloalkyl), 1 to 6 (Ci-C ₆ -haloalkyl), 1 to 8 (CrC ₈ - haloalkyl), 1 to 10 (Ci-Cio-haloalkyl) or 2 to 10 (C ₂ -Cio-haloalkyl) carbon atoms (as mentioned above), where some or all of the hydrogen atoms in these groups may be replaced by halogen atoms as mentioned above: in particular Ci-C ₂ -haloalkyl, such as chloromethyl, bromomethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoro- methyl, trifluoromethyl, chlorofluoromethyl, dichlorofluoromethyl, chlorodifluoromethyl, 1-chloroethyl, 1-bromoethyl, 1-fluoroethyl, 2-fluoroethyl, 2,2-difluoroethyl, 2,2,2- trifluoroethyl, 2-chloro-2-fluoroethyl, 2-chloro-2,2-difluoroethyl, 2,2-dichloro-2- fluoroethyl, 2,2,2-trichloroethyl, or pentafluoroethyl. Ci-C3-Haloalkyl is additionally, for example, 1 ,1 ,1-trifluoroprop-2-yl, 3,3,3-trifluoropropyl or heptafluoropropyl. CrC ₄ - Haloalkyl is additionally, for example, 1-chlorobuty, 2-chlorobutyl, 3-chlorobutyl or 4- chlorobutyl.

Ci-Cio-Hydroxyalkyl: straight-chain or branched alkyl groups having 1 to 2 (Ci-C ₂ - hydroxyalkyl), 1 to 4 (Ci-C ₄ -hydroxyalkyl), 2 to 4 (C ₂ -C ₄ -hydroxyalkyl), 1 to 6 (Ci-C ₆ - hydroxyalkyl), 2 to 6 (C ₂ -C ₆ -hydroxyalkyl), 1 to 8 (Ci-C ₈ -hydroxyalkyl), 2 to 8 (C ₂ -C ₈ - hydroxyalkyl), 1 to 10 (Ci-Cio-hydroxyalkyl) or 2 to 10 (C ₂ -Cio-hydroxyalkyl) carbon atoms (as mentioned above), where at least one of the hydrogen atoms is replaced by a hydroxyl group, such as in 2-hydroxyethyl or 3-hydroxypropyl.

Alkenyl and the alkenyl moieties in alkenyloxy, alkenylthio, alkenylcarbonyl and the like: monounsaturated straight-chain or branched hydrocarbon radicals having 2 to 4 (C ₂ - C ₄ -alkenyl), 2 to 6 (C ₂ -C ₆ -alkenyl), 2 to 8 (C ₂ -C ₈ -alkenyl), 3 to 8 (C ₃ -C ₈ -alkenyl), 2 to 10 (C ₂ -Cio-alkenyl) or 3 to 10 (C3-Cio-alkenyl) carbon atoms and a double bond in any position, for example C ₂ -C ₄ -alkenyl, such as ethenyl, 1-propenyl, 2-propenyl, 1- methylethenyl, 1-butenyl, 2-butenyl, 3-butenyl, 1-methyl-1-propenyl, 2-methyl-1- propenyl, 1-methyl-2-propenyl or 2-methyl-2-propenyl, or, for example, C ₂ -C6-alkenyl, such as ethenyl, 1-propenyl, 2-propenyl, 1 -methylethenyl, 1-butenyl, 2-butenyl, 3- butenyl, 1-methyl-1-propenyl, 2-methyl-1-propenyl, 1-methyl-2-propenyl, 2-methyl-2- propenyl, 1-pentenyl, 2-pentenyl, 3-pentenyl, 4-pentenyl, 1-methyl-1-butenyl, 2-methyl- 1-butenyl, 3-methyl-1-butenyl, 1-methyl-2-butenyl, 2-methyl-2-butenyl, 3-methyl-2- butenyl, 1-methyl-3-butenyl, 2-methyl-3-butenyl, 3-methyl-3-butenyl, 1 ,1-dimethyl-2- propenyl, 1 ,2-dimethyl-1-propenyl, 1 ,2-dimethyl-2-propenyl, 1-ethyl-1-propenyl, 1-ethyl- 2-propenyl, 1-hexenyl, 2-hexenyl, 3-hexenyl, 4-hexenyl, 5-hexenyl, 1-methyl-1- pentenyl, 2-methyl-1-pentenyl, 3-methyl-1-pentenyl, 4-methyl-1-pentenyl, 1-methyl-2- pentenyl, 2-methyl-2-pentenyl, 3-methyl-2-pentenyl, 4-methyl-2-pentenyl, 1-methyl-3- pentenyl, 2-methyl-3-pentenyl, 3-methyl-3-pentenyl, 4-methyl-3-pentenyl, 1-methyl-4- pentenyl, 2-methyl-4-pentenyl, 3-methyl-4-pentenyl, 4-methyl-4-pentenyl, 1 ,1-dimethyl- 2-butenyl, 1 ,1-dimethyl-3-butenyl, 1 ,2-dimethyl-1-butenyl, 1 ,2-dimethyl-2-butenyl, 1 ,2- dimethyl-3-butenyl, 1 ,3-dimethyl-1-butenyl, 1 ,3-dimethyl-2-butenyl, 1 ,3-dimethyl-3- butenyl, 2,2-dimethyl-3-butenyl, 2,3-dimethyl-1-butenyl, 2,3-dimethyl-2-butenyl, 2,3- dimethyl-3-butenyl, 3, 3-dimethyl-1 -butenyl, 3,3-dimethyl-2-butenyl, 1-ethyl-1 -butenyl, 1- ethyl-2-butenyl, 1-ethyl-3-butenyl, 2-ethyl-1 -butenyl, 2-ethyl-2-butenyl, 2-ethyl-3- butenyl, 1 ,1 ,2-trimethyl-2-propenyl, 1-ethyl-1-methyl-2-propenyl, 1-ethyl-2-methyl-1- propenyl, 1 -ethyl-2-methyl-2-propenyl and the like;

Haloalkenyl and the haloalkenyl moieties in haloalkenyloxy, haloalkenylcarbonyl and the like: unsaturated straight-chain or branched hydrocarbon radicals having 2 to 4 (C ₂ - C ₄ -haloalkenyl), 2 to 6 (C ₂ -C ₆ -haloalkenyl), 2 to 8 (C ₂ -C ₈ -haloalkenyl) or 2 to 10 (C ₂ - Cio-haloalkenyl) carbon atoms and a double bond in any position (as mentioned above), where some or all of the hydrogen atoms in these groups may be replaced by halogen atoms as mentioned above, in particular fluorine, chlorine and bromine, for example chlorovinyl, chloroallyl and the like;

Alkynyl and the alkynyl moieties in alkynyloxy, alkynylthio, alkynylcarbonyl and the like: straight-chain or branched hydrocarbon groups having 2 to 4 (C ₂ -C4-alkynyl), 2 to 6 (C ₂ -C ₆ -alkynyl), 2 to 8 (C ₂ -C ₈ -alkynyl), 3 to 8 (C ₃ -C ₈ -alkynyl), 2 to 10 (C ₂ -Cio-alkynyl) or 3 to 10 (C3-Cio-alkynyl) carbon atoms and one or two triple bonds in any position, for example C ₂ -C4-alkynyl, such as ethynyl, 1-propynyl, 2-propynyl, 1-butynyl, 2-butynyl, 3- butynyl, or 1-methyl-2-propynyl, or, for example, C ₂ -C6-alkynyl, such as ethynyl, 1- propynyl, 2-propynyl, 1-butynyl, 2-butynyl, 3-butynyl, 1-methyl-2-propynyl, 1-pentynyl, 2-pentynyl, 3-pentynyl, 4-pentynyl, 1-methyl-2-butynyl, 1-methyl-3-butynyl, 2-methyl-3- butynyl, 3-methyl-1-butynyl, 1 ,1-dimethyl-2-propynyl, 1-ethyl-2-propynyl, 1-hexynyl, 2- hexynyl, 3-hexynyl, 4-hexynyl, 5-hexynyl, 1-methyl-2-pentynyl, 1-methyl-3-pentynyl, 1- methyl-4-pentynyl, 2-methyl-3-pentynyl, 2-methyl-4-pentynyl, 3-methyl-1-pentynyl, 3- methyl-4-pentynyl, 4-methyl-1-pentynyl, 4-methyl-2-pentynyl, 1 ,1-dimethyl-2-butynyl, 1 ,1-dimethyl-3-butynyl, 1 ,2-dimethyl-3-butynyl, 2,2-dimethyl-3-butynyl, 3,3-dimethyl-1- butynyl, 1-ethyl-2-butynyl, 1-ethyl-3-butynyl, 2-ethyl-3-butynyl, 1-ethyl-1-methyl-2- propynyl and the like;

Haloalkynyl and the haloalkynyl moieties in haloalkynyloxy, haloalkynylcarbonyl and the like: unsaturated straight-chain or branched hydrocarbon radicals having 2 to 4 (C ₂ - C ₄ -haloalkynyl), 2 to 6 (C ₂ -C ₆ -haloalkynyl), 2 to 8 (C ₂ -C ₈ -haloalkynyl) or 2 to 10 (C ₂ -Ci ₀ - haloalkynyl) carbon atoms and one or two triple bonds in any position (as mentioned above), where some or all of the hydrogen atoms in these groups may be replaced by halogen atoms as mentioned above, in particular fluorine, chlorine and bromine;

Cycloalkyl and the cycloalkyl moieties in cycloalkoxy, cycloalkylcarbonyl and the like; monocyclic saturated hydrocarbon groups having 3 to 6 (Cs-Cβ-cycloalkyl), 3 to 8 (C3- C ₈ -cycloalkyl) or 3 to 10 (C3-Cio-cycloalkyl) carbon ring members, such as cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, cycloheptyl, cyclooctyl, cyclononyl and cyclodecyl; Halocycloalkyl and the halocycloalkyl moieties in halocycloalkoxy, halocycloalkylcar- bonyl and the like: monocyclic saturated hydrocarbon groups having 3 to 6 (C3-C6- halocycloalkyl), 3 to 8 (C ₃ -C8-halocycloalkyl) or 3 to 10 (C3-Cio-halocycloalkyl) carbon ring members (as mentioned above) in which some or all of the hydrogen atoms may be replaced by halogen atoms as mentioned above, in particular fluorine, chlorine and bromine;

Cycloalkenyl and the cycloalkenyl moieties in cycloalkenyloxy, cycloalkenylcarbonyl and the like; monocyclic monounsaturated hydrocarbon groups having 3 to 6 (C3-C6- cycloalkenyl), 3 to 8 (C ₃ -C8-cycloalkenyl) or 3 to 10 (C3-Cio-cycloalkenyl) carbon ring members, such as cyclopropenyl, cyclobutenyl, cyclopentenyl, cyclohexenyl, cyclohep- tenyl, cyclooctenyl, cyclononenyl and cyclodecenyl;

Halocycloalkenyl and the halocycloalkenyl moieties in halocycloalkenyloxy, halo- cycloalkenylcarbonyl and the like: monocyclic monounsaturated hydrocarbon groups having 3 to 6 (C ₃ -C ₆ -halocycloalkenyl), 3 to 8 (C ₃ -C ₈ -halocycloalkenyl) or 3 to 10 (C ₃ - Cio-halocycloalkenyl) carbon ring members (as mentioned above) in which some or all of the hydrogen atoms may be replaced by halogen atoms as mentioned above, in particular fluorine, chlorine and bromine;

C ₃ -C6-cycloalkyl-Ci-C2-alkyl: a Ci-C2-alkyl residue, as decribed above, wherein one of the hydrogen atoms is replaced by a C ₃ -C6-cycloalkyl group. Examples are cyclopro- pylmethyl, cyclobutylmethyl, cyclopentylmethyl, cyclohexylmethyl, cyclopropyl-1 -ethyl, cyclobutyl-1 -ethyl, cyclopentyl-1 -ethyl, cyclohexyl-1 -ethyl, cyclopropyl-2-ethyl, cyclobu- tyl-2-ethyl, cyclopentyl-2-ethyl, cyclohexyl-2-ethyl and the like. C ₃ -Cio-cycloalkyl-Ci-C4- alkyl is a Ci-C4-alkyl residue, as decribed above, wherein one of the hydrogen atoms is replaced by a C ₃ -Cio-cycloalkyl group. Examples are, apart those mentioned above for C ₃ -C6-cycloalkyl-Ci-C4-alkyl, cycloheptylmethyl, cyclooctylmethyl, cyclononylmethyl, cyclodecylmethyl, cycloheptyl-1 -ethyl, cyclooctyl-1 -ethyl, cyclononyl-1 -ethyl, cyclode- cyl-1 -ethyl, cycloheptyl-2 -ethyl, cyclooctyl-2 -ethyl, cyclononyl-2 -ethyl, cyclodecylmethyl, cyclopropyl-1 -propyl, cyclopropyl-2-propyl, cyclopropyl-3-propyl, cyclobutyl-1 - propyl, cyclobutyl-2-propyl, cyclobutyl-3-propyl, cyclopentyl-1 -propyl, cyclopentyl-2- propyl, cyclopentyl-3-propyl, cyclohexyl-1 -propyl, cyclohexyl-2-propyl, cyclohexyl-3- propyl, cycloheptyl-1 -propyl, cycloheptyl-2-propyl, cycloheptyl-3-propyl, cyclooctyl-1 - propyl, cyclooctyl-2-propyl, cyclooctyl-3-propyl, cyclononyl-1 -propyl, cyclononyl-2- propyl, cyclononyl-3-propyl, cyclodecyl-1 -propyl, cyclodecyl-2-propyl, cyclodecyl-3- propy, cyclopropyl-1 -butyl, cyclopropyl-2-butyl, cyclopropyl-3-butyl, cyclopropyl-4-butyl, cyclobutyl-1 -butyl, cyclobutyl-2-butyl, cyclobutyl-3-butyl, cyclobutyl-4-butyl, cyclopentyl- 1 -butyl, cyclopentyl-2-butyl, cyclopentyl-3-butyl, cyclopentyl-4-butyl, cyclohexyl-1 -butyl, cyclohexyl-2-butyl, cyclohexyl-3-butyl, cyclohexyl-4-butyl, cycloheptyl-1 -butyl, cyclohep- tyl-2-butyl, cycloheptyl-3-butyl, cycloheptyl-4-butyl, cyclooctyl-1 -butyl, cyclooctyl-2- butyl, cyclooctyl-3-butyl, cyclooctyl-4-butyl, cyclononyl-1 -butyl, cyclononyl-2-butyl, cyc- lononyl-3-butyl, cyclononyl-4-butyl, cyclodecyl-1 -butyl, cyclodecyl-2-butyl, cyclodecyl-3- butyl, cyclodecyl-4-butyl, and the like.

C3-C6-halocycloalkyl-Ci-C2-alkyl: a Ci-C2-alkyl residue, as decribed above, wherein one of the hydrogen atoms is replaced by a Cs-Cβ-halocycloalkyl group. Examples are 1- chlorocyclopropylmethyl, i-chlorocyclobutylmethyl, i-chlorocyclopentylmethyl, 1- chlorocyclohexylmethyl, 1-chlorocyclopropyl-i -ethyl, 1-chlorocyclobutyl-1 -ethyl, 1- chlorocyclopentyl-1 -ethyl, 1-chlorocyclohexyl-i -ethyl, 1-chlorocyclopropyl-2-ethyl, 1- chlorocyclobutyl-2 -ethyl, 1-chlorocyclopentyl-2-ethyl, 1-chlorocyclohexyl-2-ethyl, 2- chlorocyclopropylmethyl, 2-chlorocyclobutylmethyl, 2-chlorocyclopentylmethyl, 2- chlorocyclohexylmethyl, 2-chlorocyclopropyl-1 -ethyl, 2-chlorocyclobutyl-1 -ethyl, 2- chlorocyclopentyl-1 -ethyl, 2-chlorocyclohexyl-1 -ethyl, 2-chlorocyclopropyl-2-ethyl, 2- chlorocyclobutyl-2 -ethyl, 2-chlorocyclopentyl-2-ethyl, 2-chlorocyclohexyl-2-ethyl, 1- fluorocyclopropylmethyl, 1-fluorocyclobutylmethyl, 1-fluorocyclopentylmethyl, 1- fluorocyclohexylmethyl, 1-fluorocyclopropyl-1 -ethyl, 1-fluorocyclobutyl-1 -ethyl, 1- fluorocyclopentyl-1 -ethyl, 1-fluorocyclohexyl-i -ethyl, 1-fluorocyclopropyl-2-ethyl, 1- fluorocyclobutyl-2 -ethyl, 1-fluorocyclopentyl-2-ethyl, i-fluorocyclohexyl-2-ethyl, 2- fluorocyclopropylmethyl, 2-fluorocyclobutylmethyl, 2-fluorocyclopentylmethyl, 2- fluorocyclohexylmethyl, 2-fluorocyclopropyl-1 -ethyl, 2-fluorocyclobutyl-1 -ethyl, 2- fluorocyclopentyl-1 -ethyl, 2-fluorocyclohexyl-1 -ethyl, 2-fluorocyclopropyl-2-ethyl, 2- fluorocyclobutyl-2-ethyl, 2-fluorocyclopentyl-2-ethyl, 2-fluorocyclohexyl-2-ethyl, and the like. C3-Cio-halocycloalkyl-Ci-C4-alkyl is a Ci-C4-alkyl residue, as decribed above, wherein one of the hydrogen atoms is replaced by a C3-Cio-halocycloalkyl group.

Alkoxy: an alkyl group attached via oxygen. Ci-C2-Alkoxy is methoxy or ethoxy. C1-C3- Alkoxy is additionally, for example, n-propoxy or 1-methylethoxy (isopropoxy). C1-C4- Alkoxy is additionally, for example, butoxy, 1-methylpropoxy (sec-butoxy), 2- methylpropoxy (isobutoxy) or 1 ,1-dimethylethoxy (tert-butoxy). d-Cβ-Alkoxy is additionally, for example, pentoxy, 1-methylbutoxy, 2-methylbutoxy, 3-methylbutoxy, 1 ,1- dimethylpropoxy, 1 ,2-dimethylpropoxy, 2,2-dimethylpropoxy, 1-ethylpropoxy, hexoxy, 1-methylpentoxy, 2-methylpentoxy, 3-methylpentoxy, 4-methylpentoxy, 1 ,1- dimethylbutoxy, 1 ,2-dimethylbutoxy, 1 ,3-dimethylbutoxy, 2,2-dimethylbutoxy, 2,3- dimethylbutoxy, 3,3-dimethylbutoxy, 1-ethylbutoxy, 2-ethylbutoxy, 1 ,1 ,2- trimethylpropoxy, 1 ,2,2-trimethylpropoxy, 1-ethyl-1-methylpropoxy or 1 -ethyl-2- methylpropoxy. Ci-Cs-Alkoxy is additionally, for example, heptyloxy, octyloxy, 2- ethylhexyloxy and positional isomers thereof. Ci-Cio-Alkoxy is additionally, for example, nonyloxy, decyloxy and positional isomers thereof. C2-Cio-Alkoxy is like Ci-Cio-alkoxy with the exception of methoxy.

Haloalkoxy: an alkoxy radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, preferably by fluorine. Ci-C2-Haloalkoxy is, for example, OCH ₂ F, OCHF ₂ , OCF ₃ , OCH ₂ CI, OCHCI ₂ , OCCI ₃ , chlorofluoromethoxy, dichlorofluoromethoxy, chlorodifluoromethoxy, 2-fluoroethoxy, 2-chloroethoxy, 2-bromoethoxy, 2-iodoethoxy, 2,2-difluoroethoxy, 2,2,2-trifluoroethoxy, 2-chloro-2- fluoroethoxy, 2-chloro-2,2-difluoroethoxy, 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloroethoxy or OC ₂ Fs. Ci-C4-Haloalkoxy is additionally, for example, 2-fluoropropoxy, 3-fluoropropoxy, 2,2-difluoropropoxy, 2,3-difluoropropoxy, 2-chloropropoxy, 3-chloropropoxy, 2,3-dichloropropoxy, 2-bromopropoxy, 3-bromopropoxy, 3,3,3-trifluoropropoxy, 3,3,3-trichloropropoxy, OCH ₂ -C ₂ F ₅ , OCF ₂ - C ₂ F ₅ , 1-(CH ₂ F)-2-fluoroethoxy, 1-(CH ₂ CI)-2-chloroethoxy, 1-(CH ₂ Br)-2-bromoethoxy, 4-fluorobutoxy, 4-chlorobutoxy, 4-bromobutoxy or nonafluorobutoxy. Ci-Cβ-Haloalkoxy is additionally, for example, 5-fluoropentoxy, 5-chloropentoxy, 5-brompentoxy, 5-iodopentoxy, undecafluoropentoxy, 6-fluorohexoxy, 6-chlorohexoxy, 6-bromohexoxy, 6-iodohexoxy or dodecafluorohexoxy.

Alkenyloxy: alkenyl as mentioned above which is attached via an oxygen atom, for example C ₂ -Cio-alkenyloxy, such as 1-ethenyloxy, 1-propenyloxy, 2-propenyloxy, 1- methylethenyloxy, 1-butenyloxy, 2-butenyloxy, 3-butenyloxy, 1-methyl-1-propenyloxy, 2-methyl-1-propenyloxy, 1-methyl-2-propenyloxy, 2-methyl-2-propenyloxy, 1- pentenyloxy, 2-pentenyloxy, 3-pentenyloxy, 4-pentenyloxy, 1-methyl-1-butenyloxy, 2- methyl-1-butenyloxy, 3-methyl-1-butenyloxy, 1-methyl-2-butenyloxy, 2-methyl-2- butenyloxy, 3-methyl-2-butenyloxy, 1-methyl-3-butenyloxy, 2-methyl-3-butenyloxy, 3- methyl-3-butenyl, 1 ,1-dimethyl-2-propenyloxy, 1 ,2-dimethyl-1-propenyloxy, 1 ,2- dimethyl-2-propenyloxy, 1-ethyl-1-propenyloxy, 1-ethyl-2-propenyloxy, 1-hexenyloxy, 2-hexenyloxy, 3-hexenyloxy, 4-hexenyloxy, 5-hexenyloxy, 1-methyl-1-pentenyloxy, 2-methyl-1-pentenyloxy, 3-methyl-1-pentenyloxy, 4-methyl-1-pentenyloxy, 1-methyl-2- pentenyloxy, 2-methyl-2-pentenyloxy, 3-methyl-2-pentenyloxy, 4-methyl-2-pentenyloxy, 1-methyl-3-pentenyloxy, 2-methyl-3-pentenyloxy, 3-methyl-3-pentenyloxy, 4-methyl-3- pentenyloxy, 1-methyl-4-pentenyloxy, 2-methyl-4-pentenyloxy, 3-methyl-4-pentenyloxy, 4-methyl-4-pentenyloxy, 1 ,1-dimethyl-2-butenyloxy, 1 ,1-dimethyl-3-butenyloxy, 1 ,2-dimethyl-1-butenyloxy, 1 ,2-dimethyl-2-butenyloxy, 1 ,2-dimethyl-3-butenyloxy, 1 ,3-dimethyl-1-butenyloxy, 1 ,3-dimethyl-2-butenyloxy, 1 ,3-dimethyl-3-butenyloxy, 2,2-dimethyl-3-butenyloxy, 2,3-dimethyl-1 -butenyloxy, 2,3-dimethyl-2-butenyloxy, 2,3-dimethyl-3-butenyloxy, 3,3-dimethyl-1 -butenyloxy, 3,3-dimethyl-2-butenyloxy, 1 -ethyl-1 -butenyloxy, 1-ethyl-2-butenyloxy, 1-ethyl-3-butenyloxy, 2-ethyl-1 -butenyloxy, 2-ethyl-2-butenyloxy, 2-ethyl-3-butenyloxy, 1 ,1 ,2-trimethyl-2-propenyloxy, 1 -ethyl-1 - methyl-2-propenyloxy, 1-ethyl-2-methyl-1-propenyloxy and 1-ethyl-2-methyl-2- propenyloxy and the like;

Haloalkenyloxy: an alkenyloxy radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, preferably by fluorine.

Alkynyloxy: alkynyl as mentioned above which is attached via an oxygen atom, for example C2-Cio-alkynyloxy, such as 2-propynyloxy, 2-butynyloxy, 3-butynyloxy, 1-methyl- 2-propynyloxy, 2-pentynyloxy, 3-pentynyloxy, 4-pentynyloxy, 1-methyl-2-butynyloxy, 1- methyl-3-butynyloxy, 2-methyl-3-butynyloxy, 1 -ethyl-2-propynyloxy, 2-hexynyloxy, 3- hexynyloxy, 4-hexynyloxy, 5-hexynyloxy, 1-methyl-2-pentynyloxy, 1-methyl-3- pentynyloxy and the like;

Haloalkynyloxy: an alkynyloxy radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, preferably by fluorine.

Cycloalkoxy: cycloalkyl as mentioned above which is attached via an oxygen atom, for example C3-Cio-cycloalkoxy or Cs-Cs-cycloalkoxy, such as cyclopropoxy, cyclopentoxy, cyclohexoxy, cycloheptoxy, cyclooctoxy, cyclononyloxy, cyclodecyloxy and the like;

Halocycloalkoxy: a cycloalkoxy radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, preferably by fluorine.

Cycloalkenyloxy: cycloalkenyl as mentioned above which is attached via an oxygen atom, for example C3-Cio-cycloalkenyloxy, Cs-Cs-cycloalkenyloxy or, preferably, Cs-Cβ- cycloalkenyloxy, such as cyclopent-1-enoxy, cyclopent-2-enoxy, cyclohex-1-enoxy and cyclohex-2-enoxy;

Alkoxyalkyl: alkyl as defined above having 1 to 10, 1 to 8, 1 to 6 or 1 to 4, in particular 1 to 3, carbon atoms, in which one hydrogen atom is replaced by an alkoxy group having 1 to 8, 1 to 6, 1 to 4 or 1 to 3 carbon atoms, for example methoxymethyl, 2- methoxyethyl, ethoxymethyl, 3-methoxypropyl, 3-ethoxypropyl and the like.

Alkoxyalkoxy: alkoxy as defined above having 1 to 10, 1 to 8, 1 to 6 or 1 to 4, in particular 1 to 3, carbon atoms, in which one hydrogen atom is replaced by an alkoxy group having 1 to 8, 1 to 6 or in particular 1 to 4 carbon atoms, for example 2-methoxyethoxy, 2-ethoxyethoxy, 3-methoxypropoxy, 3-ethoxypropoxy and the like. Alkylcarbonyl: group of the formula R-CO- in which R is an alkyl group as defined above, for example Ci-Cio-alkyl, Ci-Cs-alkyl, Ci-Cβ-alkyl, Ci-C4-alkyl, Ci-C2-alkyl or C3- C4-alkyl. Examples are acetyl, propionyl and the like. Examples for C3-C4-alkylcarbonyl are propylcarbonyl, isopropylcarbonyl, n-butylcarbonyl, sec-butylcarbonyl, isobutylcar- bonyl and tert-butylcarbonyl.

Haloalkylcarbonyl: group of the formula R-CO- in which R is a haloalkyl group as defined above, for example Ci-Cio-haloalkyl, Ci-Cs-haloalkyl, Ci-Cβ-haloalkyl, C1-C4- haloalkyl, Ci-C2-haloalkyl or C3-C4-haloalkyl. Examples are difluoromethylcarbonyl, trifluoromethylcarbonyl, 2,2-difluoroethylcarbony, 2,2,3-trifluoroethylcarbonyl and the like.

Alkoxycarbonyl: group of the formula R-CO- in which R is an alkoxy group as defined above, for example Ci-Cio-alkoxy, Ci-Cs-alkoxy, Ci-Cβ-alkoxy, Ci-C4-alkoxy or C1-C2- alkoxy. Examples for Ci-C4-alkoxycarbonyl are methoxycarbonyl, ethoxycarbonyl, pro- poxycarbonyl, isopropoxycarbonyl, n-butoxycarbonyl, sec-butoxycarbonyl, isobutoxy- carbonyl and tert-butoxycarbonyl.

Haloalkoxycarbonyl: group of the formula R-CO- in which R is a haloalkoxy group as defined above, for example Ci-Cio-haloalkoxy, Ci-Cs-haloalkoxy, Ci-Cβ-haloalkoxy, Ci- C4-haloalkoxy or Ci-C2-haloalkoxy. Examples for Ci-C4-haloalkoxycarbonyl are di- fluoromethoxycarbonyl, trifluoromethoxycarbonyl, 2,2-difluoroethoxycarbony, 2,2,3- trifluoroethoxycarbonyl and the like.

Alkylaminocarbonyl: group of the formula R-NH-CO- in which R is an alkyl group as defined above, for example Ci-Cio-alkyl, Ci-Cs-alkyl, Ci-Cβ-alkyl, Ci-C4-alkyl, C1-C2- alkyl or C3-C4-alkyl. Examples for Ci-C4-alkylaminocarbonyl are methylaminocarbonyl, ethylaminocarbonyl, propylaminocarbonyl, isopropylaminocarbonyl, butylaminocar- bonyl, sec-butylaminocarbonyl, isobutylaminocarbonyl and tert-butylaminocarbonyl.

Dialkylaminocarbonyl: group of the formula RR'N-CO- in which R and R', independently of each other, are an alkyl group as defined above, for example Ci-Cio-alkyl, Ci-Cs- alkyl, d-Ce-alkyl, Ci-d-alkyl, Ci-C ₂ -alkyl or drd-alkyl. Examples for di-(Ci-C ₄ -alkyl)- aminocarbonyl are dimethylaminocarbonyl, diethylaminocarbonyl, dipropylaminocar- bonyl, diisopropylaminocarbonyl and dibutylaminocarbonyl.

Aminoalkyl: group of the formula R-NH2 in which R is an alkyl group as defined above, for example Ci-Cio-alkyl, Ci-Cs-alkyl, Ci-Ce-alkyl, Ci-C ₄ -alkyl, Ci-C ₂ -alkyl or C ₃ -C ₄ - alkyl. Examples are aminomethyl, 1- and 2-aminoethyl, 1-, 2- and 3-aminopropyl, 1- and 2-amino1-methylethyl, 1-, 2-, 3- and 4-aminobutyl and the like.

Alkylsulfonyl: group of the formula R-S(O)2- in which R is an alkyl group as defined above, for example Ci-Cio-alkyl, Ci-Cs-alkyl, d-Cε-alkyl, Ci-C4-alkyl or Ci-C2-alkyl. Examples for Ci-C4-alkylsulfonyl are methylsulfonyl, ethylsulfonyl, propylsulfonyl, iso- propylsulfonyl, n-butylsulfonyl, sec-butylsulfonyl, isobutylsulfonyl and tert-butylsulfonyl.

Alkylthio: alkyl as defined above which is attached via a sulfur atom.

Haloalkylthio: haloalkyl as defined above which is attached via a sulfur atom.

Alkenylthio: alkenyl as defined above which is attached via a sulfur atom.

Haloalkenylthio: haloalkenyl as defined above which is attached via a sulfur atom.

Alkynylthio: alkynyl as defined above which is attached via a sulfur atom.

Haloalkynylthio: haloalkynyl as defined above which is attached via a sulfur atom.

Cycloalkylthio: cycloalkyl as defined above which is attached via a sulfur atom.

Aryl is a carbocyclic aromatic monocyclic or polycyclic ring containing 6 to 16 carbon atoms as ring members. Examples are phenyl, naphthyl, anthracenyl, phenanthrenyl, fluorenyl and azulenyl. Preferably, aryl is phenyl or naphthyl, and especially phenyl.

Aryl-Ci-C4-alkyl: Ci-C4-alkyl (as defined above), where a hydrogen atom is replaced by an aryl group as defined above, such as benzyl, phenethyl, naphthylmethyl, 2- naphthylethyl and the like.

Phenyl-Ci-C4-alkyl: Ci-C4-alkyl (as defined above), where a hydrogen atom is replaced by a phenyl group, such as benzyl, phenethyl and the like.

Phenyl-Ci-C4-alkoxy: Ci-C4-alkoxy (as defined above), where one hydrogen atom is replaced by a phenyl group, such as benzyloxy, phenethyloxy and the like.

3-, 4-, 5-, 6- or 7-membered saturated, partially unsaturated or maximum unsaturated carbocyclic radical: cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, cycloheptyl, cyclo- propenyl, cyclobutenyl, cyclopentenyl, cyclohexenyl, cycloheptenyl, cyclobutadienyl, cyclopentadienyl, cyclohexadienyl, cycloheptadienyl or cycloheptatrienyl. Formally, phenyl is also included in this definition, but as it is also encompassed in the term aryl, it is not listed here.

3-, 4-, 5-, 6- or 7-membered saturated, partially unsaturated or maximum unsaturated heterocycle which contains 1 , 2 or 3 heteroatoms or heteroatom containing groups selected from oxygen, nitrogen (as N or NR) and sulfur (as S, SO or SO2) and optionally 1 or 2 groups selected from C(=O) and C(=S) as ring members:

- three- or four-membered saturated or partially unsaturated heterocycle (hereinbe- low also referred to as heterocyclyl) which contains 1 , 2 or 3 heteroatoms selected from the group consisting of oxygen, nitrogen (as N or NR) and sulfur (as S, SO or SO2) and optionally 1 or 2 groups selected from C(=O) and C(=S) as ring members: for example monocyclic saturated or partially unsaturated hetero- cycles which, in addition to carbon ring members, contain one to three nitrogen atoms and/or one oxygen or sulfur atom or one or two oxygen and/or sulfur atoms and optionally 1 or 2 groups selected from C(=O) and C(=S), for example 2- oxiranyl, 2-thiiranyl, 1- or 2-aziridinyl, 1-, 2- or 3-azetidinyl,

- five- or six-membered saturated or partially unsaturated heterocycle (hereinbelow also referred to as heterocyclyl) which contains 1 , 2 or 3 heteroatoms selected from the group consisting of oxygen, nitrogen (as N or NR) and sulfur (as S, SO or SO2) and optionally 1 or 2 groups selected from C(=O) and C(=S) as ring members: for example monocyclic saturated or partially unsaturated heterocycles which, in addition to carbon ring members, contain one to three nitrogen atoms and/or one oxygen or sulfur atom or one or two oxygen and/or sulfur atoms and optionally 1 or 2 groups selected from C(=O) and C(=S), for example 2-tetrahydrofuranyl, 3-tetrahydrofuranyl, 3-tetrahydrofuran-2-onyl, 4-tetrahydrofuran-2-onyl, 5-tetrahydrofuran-2-onyl, 2-tetrahydrofuran-3-onyl, 4-tetrahydrofuran-3-onyl, 5-tetrahydrofuran-3-onyl, 2-tetrahydrothienyl,

3-tetrahydrothienyl, 3-tetrahydrothien-2-onyl, 4-tetrahydrothien-2-onyl, 5-tetrahydrothien-2-onyl, 2-tetrahydrothien-3-onyl, 4-tetrahydrothien-3-onyl, 5-tetrahydrothien-3-onyl, 2-pyrrolidinyl, 3-pyrrolidinyl, 1 -pyrrolidin-2-onyl, 3-pyrrolidin-2-onyl, 4-pyrrolidin-2-onyl, 5-pyrrolidin-2-onyl, 1 -pyrrolidin-3-onyl, 2-pyrrolidin-3-onyl, 4-pyrrolidin-3-onyl, 5-pyrrolidin-3-onyl, 1-pyrrolidin-2,5-dionyl,

3-pyrrolidin-2,5-dionyl, 3-isoxazolidinyl, 4-isoxazolidinyl, 5-isoxazolidinyl, 3-isothiazolidinyl, 4-isothiazolidinyl, 5-isothiazolidinyl, 3-pyrazolidinyl, 4-pyrazolidinyl, 5-pyrazolidinyl, 2-oxazolidinyl, 4-oxazolidinyl, 5-oxazolidinyl, 2-thiazolidinyl, 4-thiazolidinyl, 5-thiazolidinyl, 2-imidazolidinyl, 4-imidazolidinyl, 1 ,2,4-oxadiazolidin-3-yl, 1 ,2,4-oxadiazolidin-5-yl, 1 ,2,4-thiadiazolidin-3-yl,

1 ,2,4-thiadiazolidin-5-yl, 1 ,2,4-triazolidin-3-yl, 1 ,3,4-oxadiazolidin-2-yl, 1 ,3,4-thiadiazolidin-2-yl, 1 ,3,4-triazolidin-2-yl, 2,3-dihydrofur-2-yl, 2,3-dihydrofur- 3-yl, 2,4-dihydrofur-2-yl, 2,4-dihydrofur-3-yl, 2,3-dihydrothien-2-yl, 2,3-dihydrothien-3-yl, 2,4-dihydrothien-2-yl, 2,4-dihydrothien-3-yl, 2-pyrrolin-2-yl, 2-pyrrolin-3-yl, 3-pyrrolin-2-yl, 3-pyrrolin-3-yl, 2-isoxazolin-3-yl, 3-isoxazolin-3-yl, 4-isoxazolin-3-yl, 2-isoxazolin-4-yl, 3-isoxazolin-4-yl, 4-isoxazolin-4-yl,

2-isoxazolin-5-yl, 3-isoxazolin-5-yl, 4-isoxazolin-5-yl, 2-isothiazolin-3-yl, 3-isothiazolin-3-yl, 4-isothiazolin-3-yl, 2-isothiazolin-4-yl, 3-isothiazolin-4-yl, 4-isothiazolin-4-yl, 2-isothiazolin-5-yl, 3-isothiazolin-5-yl, 4-isothiazolin-5-yl, 2,3-dihydropyrazol-1 -yl, 2,3-dihydropyrazol-2-yl, 2,3-dihydropyrazol-3-yl, 2,3-dihydropyrazol-4-yl, 2,3-dihydropyrazol-5-yl, 3,4-dihydropyrazol-i-yl,

3,4-dihydropyrazol-3-yl, 3,4-dihydropyrazol-4-yl, 3,4-dihydropyrazol-5-yl, 4,5-dihydropyrazol-1 -yl, 4,5-dihydropyrazol-3-yl, 4,5-dihydropyrazol-4-yl, 4,5-dihydropyrazol-5-yl, 2,3-dihydrooxazol-2-yl, 2,3-dihydrooxazol-3-yl, 2,3-dihydrooxazol-4-yl, 2,3-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4-yl, 3,4-dihydrooxazol-5-yl,

3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4-yl, 2-piperidinyl, 3-piperidinyl, 4-piperidinyl, 1 ,3-dioxan-5-yl, 2-tetrahydropyranyl, 4-tetrahydropyranyl, 2-tetrahydrothienyl, 3-hexahydropyridazinyl, 4-hexahydropyridazinyl, 2-hexahydropyrimidinyl, 4-hexahydropyrimidinyl, 5-hexahydropyrimidinyl, 2-piperazinyl, 1 ,3,5-hexahydrotriazin-2-yl and

1 ,2,4-hexahydrotriazin-3-yl and also the corresponding -ylidene radicals;

a seven-membered saturated or partially unsaturated heterocycle which contains 1 , 2 or 3 heteroatoms selected from the group consisting of oxygen, nitrogen and sulfur as ring members: for example mono- and bicyclic heterocycles having 7 ring members which, in addition to carbon ring members, contain one to three nitrogen atoms and/or one oxygen or sulfur atom or one or two oxygen and/or sulfur atoms, for example tetra- and hexahydroazepinyl, such as 2,3,4,5-tetrahydro[1 H]azepin-1-, -2-, -3-, -4-, -5-, -6- or -7-yl, 3,4,5,6-tetrahydro[2H]azepin-2-, -3-, -A-, -5-, -6- or -7-yl,

2,3,4,7-tetrahydro[1 H]azepin-1-, -2-, -3-, -4-, -5-, -6- or -7-yl, 2,3,6,7-tetrahydro[1 H]azepin-1-, -2-, -3-, -4-, -5-, -6- or -7-yl, hexahydroazepin-1-, -2-, -3- or -4-yl, tetra- and hexahydrooxepinyl, such as 2,3,4,5-tetrahydro[1 H]oxepin-2-, -3-, -A-, -5-, -6- or -7-yl, 2,3,4,7-tetrahydro[1 H]oxepin-2-, -3-, -A-, -5-, -6- or -7-yl,

2,3,6,7-tetrahydro[1 H]oxepin-2-, -3-, -A-, -5-, -6- or -7-yl, hexahydroazepin-1-, -2-, -3- or -4-yl, tetra- and hexahydro-1 ,3-diazepinyl, tetra- and hexahydro-1 ,4-diazepinyl, tetra- and hexahydro-1 ,3-oxazepinyl, tetra- and hexahydro-1 ,4-oxazepinyl, tetra- and hexahydro-1 ,3-dioxepinyl, tetra- and hexahydro-1 ,4-dioxepinyl and the corresponding -ylidene radicals. a five- or six-membered aromatic (= maximum unsaturated) heterocycle (= het- eroaromatic radical) which contains 1 , 2 or 3 heteroatoms selected from the group consisting of oxygen, nitrogen and sulfur, for example 5-membered het- eroaryl which is attached via carbon and contains one to three nitrogen atoms or one or two nitrogen atoms and one sulfur or oxygen atom as ring members, such as 2-furyl, 3-furyl, 2-thienyl, 3-thienyl, 2-pyrrolyl, 3-pyrrolyl, 3-isoxazolyl, 4- isoxazolyl, 5-isoxazolyl, 3-isothiazolyl, 4-isothiazolyl, 5-isothiazolyl, 3-pyrazolyl, 4- pyrazolyl, 5-pyrazolyl, 2-oxazolyl, 4-oxazolyl, 5-oxazolyl, 2-thiazolyl, 4-thiazolyl, 5- thiazolyl, 2-imidazolyl, 4-imidazolyl, 1 ,2,4-oxadiazol-3-yl, 1 ,2,4-oxadiazol-5-yl, 1 ,2,4-thiadiazol-3-yl, 1 ,2,4-thiadiazol-5-yl, 1 ,2,4-triazol-3-yl, 1 ,3,4-oxadiazol-2-yl,

1 ,3,4-thiadiazol-2-yl and 1 ,3,4-triazol-2-yl; 5-membered heteroaryl which is attached via nitrogen and contains one to three nitrogen atoms as ring members, such as pyrrol-1-yl, pyrazol-1-yl, imidazol-1-yl, 1 ,2,3-triazol-1-yl and 1 ,2,4-triazol- 1-yl; 6-membered heteroaryl, which contains one, two or three nitrogen atoms as ring members, such as pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, 3-pyridazinyl, 4- pyridazinyl, 2-pyrimidinyl, 4-pyrimidinyl, 5-pyrimidinyl, 2-pyrazinyl, 1 ,3,5-triazin-2- yl and 1 ,2,4-triazin-3-yl;

Linear C2-alkylene: divalent unbranched chains having 2 carbon atoms, namely CH ₂ CH ₂ .

Linear C ₂ - or C3-alkylene: divalent unbranched chains having 2 or 3 carbon atoms, namely CH ₂ CH ₂ and CH ₂ CH ₂ CH ₂ .

Linear d-Cs-alkylene: divalent unbranched chains having 1 to 5 carbon atoms, namely CH ₂ , CH ₂ CH ₂ , CH ₂ CH ₂ CH ₂ , CH ₂ CH ₂ CH ₂ CH ₂ and CH ₂ CH ₂ CH ₂ CH ₂ CH ₂ .

C ₂ -C5-Alkylene: divalent branched or preferably unbranched chains having 2 to 5 carbon atoms, for example CH ₂ CH ₂ , -CH(CH ₃ )-, CH ₂ CH ₂ CH ₂ , CH(CH ₃ )CH ₂ , CH ₂ CH(CH ₃ ), CH ₂ CH ₂ CH ₂ CH ₂ , CH ₂ CH ₂ CH ₂ CH ₂ CH ₂ .

C4-C5-Alkylene: divalent branched or preferably unbranched chains having 4 to 5 carbon atoms, for example CH ₂ CH ₂ CH ₂ CH ₂ or CH ₂ CH ₂ CH ₂ CH ₂ CH ₂ .

The group -SM is more correctly spoken a group -S-M ⁺ , where M ⁺ is a metal cation equivalent or an ammonium cation as defined above. A metal cation equivalent is more correctly spoken 1/a M ^a+ , where a is the valence of the metal and is in general 1 , 2 or 3.

The statements made below with respect to suitable and preferred features of the com- pounds according to the invention, especially with respect to their substituents R ¹ , R ² , R ³ , R ⁴ , R ⁵ , R ^5a , R ⁶ , R ⁷ , R ⁸ , R ⁹ , R ¹⁰ , R ¹¹ , R ¹² , R ¹³ , R ¹⁴ , R ¹⁵ , R ¹⁶ , R ¹⁷ , R ¹⁸ , R ¹⁹ , R ²⁰ , R ^a , R ^b , R ^c , R ^d , Q, M and the index m, and to their use, are valid both per se and, in particular, in every possible combination with one another.

Unless specified otherwise in specific embodiments of the invention, R ⁷ , R ⁸ , R ¹⁰ , R ¹¹ and R ¹² are independently of each other and independently of each occurrence preferably selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy and C1-C4- haloalkoxy and more preferably from F, Cl, Br, methyl, difluoromethyl, trifluoromethyl, methoxy, difluoromethoxy and trifluoromethoxy.

Unless specified otherwise in specific embodiments of the invention, preferably, R ¹⁶ is hydrogen and R ¹⁷ is selected from hydrogen, Ci-C4-alkyl and phenyl, preferably from hydrogen and Ci-C4-alkyl, or the two of R ¹⁶ and R ¹⁷ are Ci-C4-alkyl.

Unless specified otherwise in specific embodiments of the invention, preferably, R ¹⁹ is hydrogen or methyl and in particular methyl.

Unless specified otherwise in specific embodiments of the invention, preferably, R ²⁰ is Ci-C4-alkyl and in particular methyl.

R ¹³ in the groups -C(=O)R ¹³ and -S(O) ₂ R ¹³ is preferably selected from Ci-C ₄ -alkyl, Ci- C2-haloalkyl, Ci-C4-alkoxy, Ci-C2-haloalkoxy, phenyl, phenoxy and NR ¹⁶ R ¹⁷ , more preferably from Ci-C ₄ -alkyl, Ci-C ₂ -haloalkyl, Ci-C ₄ -alkoxy, Ci-C ₂ -haloalkoxy and NR ¹⁶ R ¹⁷ and even more preferably from Ci-C4-alkyl, Ci-C4-alkoxy and NR ¹⁶ R ¹⁷ . In the group -C(=O)R ¹³ , R ¹³ is specifically Ci-C4-alkyl, such as methyl, ethyl, propyl, isopropyl, n- butyl, sec-butyl, isobutyl or tert-butyl, preferably methyl, or is Ci-C4-alkoxy, such as methoxy, ethoxy, propoxy, isopropoxy, n-butoxy, sec-butoxy, isobutoxy or tert-butoxy, preferably methoxy, and is more specifically methyl, and in the group -S(O) ₂ R ¹³ , R ¹³ is specifically methyl. Preferably, R ¹⁶ is hydrogen and R ¹⁷ is selected from hydrogen, Ci- C4-alkyl and phenyl, preferably from hydrogen and Ci-C4-alkyl, or the two of R ¹⁶ and R ¹⁷ are Ci-C ₄ -alkyl.

R ⁵ is preferably selected from hydrogen, Ci-C ₄ -alkyl, -C(=O)R ¹³ , -S(O) ₂ R ¹³ , -CN, M and a group of the formula III, where R ¹³ has one of the above general meanings or, in par- ticular, one of the above preferred meanings and M has one of the above general meanings or, in particular, one of the below-given preferred meanings.

R ⁵ is more preferably selected from hydrogen, Ci-C4-alkyl, C3-C4-alkylcarbonyl, C1-C4- alkoxycarbonyl, -C(=O)N(H)Ci-C ₄ -alkyl, -C(=O)N(Ci-C ₄ -alkyl) ₂ , Ci-C ₄ -alkylsulfonyl, CN and a group of the formula III. In particular, R ⁵ is selected from hydrogen, CN, methyl- carbonyl, methoxycarbonyl and methyl. Specifically, R ⁵ is hydrogen.

M is preferably selected from an alkali metal cation, an earth alkaline metal cation equivalent, a cation equivalent of Cu, Zn, Fe or Ni or an ammonium cation of formula (NR ^a R ^b R ^c R ^d ) ⁺ , wherein one of R ^a , R ^b , R ^c and R ^d is hydrogen and three of R ^a , R ^b , R ^c and R ^d , independently of each other, are selected from Ci-Cio-alkyl. More preferably, M is selected from Li ⁺ , Na ⁺ , K ⁺ , YiMg ²⁺ , a cation equivalent of Cu, Zn, Fe or Ni and an ammonium cation of formula (NR ^a R ^b R ^c R ^d ) ⁺ , wherein one of R ^a , R ^b , R ^c and R ^d is hydrogen and three of R ^a , R ^b , R ^c and R ^d , independently of each other, are selected from C1-C10- alkyl. Even more preferably, M is selected from Na ⁺ , K ⁺ , /4Mg ²⁺ , /4Cu ²⁺ , /4Zn ²⁺ , /4Fe ²⁺ , /4Ni ²⁺ , triethylammonium and trimethylammonium.

In the group of formula III, the variables preferably have the same meanings as in the remainder of the molecule I. Thus, the remarks made above as to preferred meanings of the radicals apply to this moiety, too.

R ^5a is preferably selected from hydrogen, Ci-Cio-alkyl, Ci-C4-haloalkyl, phenyl, phenyl- Ci-C4-alkyl, -C(=O)R ¹³ and -S(O)2R ¹³ , where R ¹³ has one of the above given general or, in particular, one of the above-given preferred meanings. More preferably, R ^5a is selected from hydrogen, Ci-C4-alkyl, Ci-C4-haloalkyl, phenyl, benzyl, -C(=O)R ¹³ and -S(O)2R ¹³ , where R ¹³ has one of the above given general or, in particular, one of the above-given preferred meanings, and more preferably from hydrogen, Ci-C4-alkyl, Ci- C4-haloalkyl, -C(=O)R ¹³ and -S(O)2R ¹³ , where R ¹³ has one of the above given general or, in particular, one of the above-given preferred meanings. In particular, R ^5a is hydrogen, Ci-C4-alkyl, preferably methyl, or -C(=O)R ¹³ , more particularly hydrogen, C1-C4- alkyl, preferably methyl, methylcarbonyl or methoxycarbonyl, even more particularly hydrogen or Ci-C4-alkyl, preferably methyl, and is specifically hydrogen.

If m is 1 , the oxygen atom is preferably bound via a double bond to the sulfur atom, the radical -S(O) _m -R ⁵ thus resulting in a group -S(=O)-R ⁵ . If m is 2, the two oxygen atoms are preferably both bound via a double bond to the sulfur atom, the radical -S(O) _m -R ⁵ thus resulting in a group -S(=O)2-R ⁵ . If m is 3, the radical -S(O) _m -R ⁵ is a group -S(=O)2- O-R ⁵ .

m is preferably 0 or 2 and more preferably 0.

In a particularly preferred embodiment, in compounds I, m is 0 and R ⁵ is H (or, alternatively, in compounds II, R ^5a is H). In a preferred embodiment of the invention (embodiment A), R ¹ is a group of formula V, where

R ² is phenyl which may carry 1 , 2, 3, 4 or 5 substituents R ⁷ ; R ³ is phenyl which may carry 1 , 2, 3, 4 or 5 substituents R ¹¹ ; R ⁴ is OH; and

R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings; except for compounds wherein R ² is 2-fluorophenyl, R ³ is 4-fluorophenyl and R ⁴ is OH; and except for compounds wherein R ² is 4-fluorophenyl, R ³ is 2-fluorophenyl and R ⁴ is OH.

More preferably (embodiment A.1 ), R ¹ is a group of formula V, where R ² is phenyl which may carry 1 , 2 or 3 substituents R ⁷ ; R ³ is phenyl which may carry 1 , 2 or 3 substituents R ¹¹ ; R ⁴ is OH; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH3, CHF2, CF3,

OCH ₃ , OCHF ₂ and OCF ₃ ; each R ¹¹ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH ₃ , CHF2, CF ₃ ,

OCH ₃ , OCHF ₂ and OCF ₃ ; and

R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings; except for compounds wherein R ² is 2-fluorophenyl, R ³ is 4-fluorophenyl and R ⁴ is OH; and except for compounds wherein R ² is 4-fluorophenyl, R ³ is 2-fluorophenyl and R ⁴ is OH.

Even more preferably (embodiment A.1.1 ), R ¹ is a group of formula V, where R ² is phenyl which may carry 1 or 2 substituents R ⁷ ; R ³ is phenyl which may carry 1 or 2 substituents R ¹¹ ; R ⁴ is OH; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH ₃ , CHF ₂ , CF ₃ , OCH ₃ , OCHF ₂ and OCF ₃ ; each R ¹¹ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH ₃ , CHF ₂ , CF ₃ ,

OCH ₃ , OCHF ₂ and OCF ₃ ; and R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings; except for compounds wherein R ² is 2-fluorophenyl, R ³ is 4-fluorophenyl and R ⁴ is OH; and except for compounds wherein R ² is 4-fluorophenyl, R ³ is 2-fluorophenyl and R ⁴ is OH.

If R ² is phenyl which carries 1 substituent R ⁷ , this is preferably bound in 2- or 4- position, more preferably in 2-position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

If R ³ is phenyl which carries 1 substituent R ¹¹ , this is preferably bound in 2- opposition, more preferably in 2-position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

If R ² is phenyl which carries 2 substituents R ⁷ , these are preferably bound in 2,4- position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

If R ³ is phenyl which carries 2 substituents R ¹¹ , these are preferably bound in 2,4- position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

Examples for preferred compounds I and Il of embodiment A are compounds of formulae I.A1 , IA.2 and II.A1 , where the variables R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ are hydrogen or have one of the general or, in particular, one of the preferred meanings given above for R ⁷ and where the variables R ³ , R ⁵ and R ^5a have one of the general or, in particular, one of the preferred meanings given above in context with embodiment A. Examples of preferred compounds are the individual compounds compiled in the tables 1 to 43380 below. Moreover, the meanings mentioned below for the individual variables in the ta- bles are per se, independently of the combination in which they are mentioned, a particularly preferred embodiment of the substituents in question.

Table 1

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is phenyl

Table 2

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluorophenyl

Table 3

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluorophenyl Table 4

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 4- fluorophenyl

Table 5 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chlorophenyl

Table 6

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chlorophenyl

Table 7

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 4- chlorophenyl

Table 8

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromophenyl

Table 9

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromophenyl

Table 10

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 4- bromophenyl Table 11

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methylphenyl

Table 12 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methylphenyl

Table 13

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 4- methylphenyl

Table 14

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- (difluoromethyl)-phenyl

Table 15

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3-

(difluoromethyl)-phenyl Table 16

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 4-

(difluoromethyl)-phenyl Table 17

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2-

(trifluoromethyl)-phenyl Table 18

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3-

(trifluoromethyl)-phenyl

Table 19 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 4-

(trifluoromethyl)-phenyl

Table 20

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxyphenyl

Table 21

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methoxyphenyl

Table 22

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 4- methoxyphenyl Table 23

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2-

(difluoromethoxy)-phenyl

Table 24 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3-

(difluoromethoxy)-phenyl

Table 25

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 4-

(difluoromethoxy)-phenyl

Table 26

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2-

(trifluoromethoxy)-phenyl

Table 27

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3-

(trifluoromethoxy)-phenyl

Table 28

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 4- (trifluoromethoxy)-phenyl

Table 29

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,3- difluorophenyl Table 30

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4- difluorophenyl

Table 31 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,5- difluorophenyl

Table 32

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- difluorophenyl

Table 33

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,4- difluorophenyl

Table 34

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,5- difluorophenyl Table 35

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,3- dichlorophenyl Table 36

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4- dichlorophenyl Table 37

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,5- dichlorophenyl

Table 38 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- dichlorophenyl

Table 39

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,4- dichlorophenyl

Table 40

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,5- dichlorophenyl

Table 41

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,3- dibromophenyl Table 42

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4- dibromophenyl

Table 43 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,5- dibromophenyl

Table 44

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- dibromophenyl

Table 45

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,4- dibromophenyl

Table 46

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,5- dibromophenyl

Table 47

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,3- dimethylphenyl

Table 48

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4- dimethylphenyl Table 49

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,5- dimethylphenyl

Table 50 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- dimethylphenyl

Table 51

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,4- dimethylphenyl

Table 52

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,5- dimethylphenyl

Table 53

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,3- di-(difluoromethyl)-phenyl Table 54

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4- di-(difluoromethyl)-phenyl Table 55

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,5- di-(difluoromethyl)-phenyl Table 56

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- di-(difluoromethyl)-phenyl

Table 57 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,4- di-(difluoromethyl)-phenyl

Table 58

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,5- di-(difluoromethyl)-phenyl

Table 59

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,3- di-(trifluoromethyl)-phenyl

Table 60

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4- di-(trifluoromethyl)-phenyl Table 61

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,5- di-(trifluoromethyl)-phenyl

Table 62 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- di-(trifluoromethyl)-phenyl

Table 63

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,4- di-(trifluoromethyl)-phenyl

Table 64

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,5- di-(trifluoromethyl)-phenyl

Table 65

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,3- dimethoxyphenyl

Table 66

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4- dimethoxyphenyl

Table 67

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,5- dimethoxyphenyl Table 68

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- dimethoxyphenyl

Table 69 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,4- dimethoxyphenyl

Table 70

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,5- dimethoxyphenyl

Table 71

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,3- di-(difluoromethoxy)-phenyl

Table 72

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4- di-(difluoromethoxy)-phenyl Table 73

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,5- di-(difluoromethoxy)-phenyl Table 74

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- di-(difluoromethoxy)-phenyl Table 75

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,4- di-(difluoromethoxy)-phenyl

Table 76 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,5- di-(difluoromethoxy)-phenyl

Table 77

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,3- di-(trifluoromethoxy)-phenyl

Table 78

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4- di-(trifluoromethoxy)-phenyl

Table 79

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,5- di-(trifluoromethoxy)-phenyl Table 80

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- di-(trifluoromethoxy)-phenyl

Table 81 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,4- di-(trifluoromethoxy)-phenyl

Table 82

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3,5- di-(trifluoromethoxy)-phenyl

Table 83

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-3-chlorophenyl

Table 84

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-4-chlorophenyl

Table 85

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-5-chlorophenyl

Table 86

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-6-chlorophenyl Table 87

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-4-chlorophenyl

Table 88 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-5-chlorophenyl

Table 89

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-3-fluorophenyl

Table 90

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-4-fluorophenyl

Table 91

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-5-fluorophenyl Table 92

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-4-fluorophenyl Table 93

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-3-bromophenyl Table 94

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-4-bromophenyl

Table 95 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-5-bromophenyl

Table 96

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-6-bromophenyl

Table 97

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-4-bromophenyl

Table 98

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-5-bromophenyl Table 99

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-3-fluorophenyl

Table 100 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-4-fluorophenyl

Table 101

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-5-fluorophenyl

Table 102

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-4-fluorophenyl

Table 103

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-3-methylphenyl

Table 104

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-4-methylphenyl

Table 105

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-5-methylphenyl Table 106

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-6-methylphenyl

Table 107 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-4-methylphenyl

Table 108

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-5-methylphenyl

Table 109

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-3-fluorophenyl

Table 110

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-4-fluorophenyl Table 11 1

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-5-fluorophenyl Table 112

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-4-fluorophenyl Table 113

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-3-difluoromethylphenyl

Table 114 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-4-difluoromethylphenyl

Table 115

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-5-difluoromethylphenyl

Table 116

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-6-difluoromethylphenyl

Table 117

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-4-difluoromethylphenyl Table 118

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-5-difluoromethylphenyl

Table 119 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-3-fluorophenyl

Table 120

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-4-fluorophenyl

Table 121

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-5-fluorophenyl

Table 122

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethyl-4-fluorophenyl

Table 123

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-3-trifluoromethylphenyl

Table 124

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-4-trifluoromethylphenyl Table 125

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-5-trifluoromethylphenyl

Table 126 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-6-trifluoromethylphenyl

Table 127

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-4-trifluoromethylphenyl

Table 128

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-5-trifluoromethylphenyl

Table 129

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-3-fluorophenyl Table 130

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-4-fluorophenyl Table 131

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-5-fluorophenyl Table 132

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethyl-4-fluorophenyl

Table 133 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-3-methoxyphenyl

Table 134

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-4-methoxyphenyl

Table 135

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-5-methoxyphenyl

Table 136

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-6-methoxyphenyl Table 137

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-4-methoxyphenyl

Table 138 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-5-methoxyphenyl

Table 139

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-3-fluorophenyl

Table 140

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-4-fluorophenyl

Table 141

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-5-fluorophenyl

Table 142

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methoxy-4-fluorophenyl

Table 143

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-3-difluoromethoxyphenyl Table 144

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-4-difluoromethoxyphenyl

Table 145 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-5-difluoromethoxyphenyl

Table 146

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-6-difluoromethoxyphenyl

Table 147

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-4-difluoromethoxyphenyl

Table 148

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-5-difluoromethoxyphenyl Table 149

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-3-fluorophenyl Table 150

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-4-fluorophenyl Table 151

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-5-fluorophenyl

Table 152 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethoxy-4-fluorophenyl

Table 153

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-3-trifluoromethoxyphenyl

Table 154

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-4-trifluoromethoxyphenyl

Table 155

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-5-trifluoromethoxyphenyl Table 156

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- fluoro-6-trifluoromethoxyphenyl

Table 157 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-4-trifluoromethoxyphenyl

Table 158

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- fluoro-5-trifluoromethoxyphenyl

Table 159

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-3-fluorophenyl

Table 160

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-4-fluorophenyl

Table 161

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-5-fluorophenyl

Table 162

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethoxy-4-fluorophenyl Table 163

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-3-bromophenyl

Table 164 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-4-bromophenyl

Table 165

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-5-bromophenyl

Table 166

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-6-bromophenyl

Table 167

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-4-bromophenyl Table 168

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-5-bromophenyl Table 169

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-3-chlorophenyl Table 170

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-4-chlorophenyl

Table 171 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-5-chlorophenyl

Table 172

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-4-chlorophenyl

Table 173

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-3-methylphenyl

Table 174

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-4-methylphenyl Table 175

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-5-methylphenyl

Table 176 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-6-methylphenyl

Table 177

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-4-methylphenyl

Table 178

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-5-methylphenyl

Table 179

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-3-chlorophenyl

Table 180

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-4-chlorophenyl

Table 181

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-5-chlorophenyl Table 182

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-4-chlorophenyl

Table 183 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-3-difluoromethylphenyl

Table 184

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-4-difluoromethylphenyl

Table 185

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-5-difluoromethylphenyl

Table 186

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-6-difluoromethylphenyl Table 187

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-4-difluoromethylphenyl Table 188

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-5-difluoromethylphenyl Table 189

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-3-chlorophenyl

Table 190 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-4-chlorophenyl

Table 191

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-5-chlorophenyl

Table 192

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethyl-4-chlorophenyl

Table 193

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-3-trifluoromethylphenyl Table 194

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-4-trifluoromethylphenyl

Table 195 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-5-trifluoromethylphenyl

Table 196

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-6-trifluoromethylphenyl

Table 197

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-4-trifluoromethylphenyl

Table 198

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-5-trifluoromethylphenyl

Table 199

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-3-chlorophenyl

Table 200

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-4-chlorophenyl Table 201

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-5-chlorophenyl

Table 202 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethyl-4-chlorophenyl

Table 203

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-3-methoxyphenyl

Table 204

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-4-methoxyphenyl

Table 205

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-5-methoxyphenyl Table 206

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-6-methoxyphenyl Table 207

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-4-methoxyphenyl Table 208

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-5-methoxyphenyl

Table 209 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-3-chlorophenyl

Table 210

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-4-chlorophenyl

Table 21 1

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-5-chlorophenyl

Table 212

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methoxy-4-chlorophenyl Table 213

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-3-difluoromethoxyphenyl

Table 214 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-4-difluoromethoxyphenyl

Table 215

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-5-difluoromethoxyphenyl

Table 216

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-6-difluoromethoxyphenyl

Table 217

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-4-difluoromethoxyphenyl

Table 218

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-5-difluoromethoxyphenyl

Table 219

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-3-chlorophenyl Table 220

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-4-chlorophenyl

Table 221 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-5-chlorophenyl

Table 222

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethoxy-4-chlorophenyl

Table 223

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-3-trifluoromethoxyphenyl

Table 224

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-4-trifluoromethoxyphenyl Table 225

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-5-trifluoromethoxyphenyl Table 226

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- chloro-6-trifluoromethoxyphenyl Table 227

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-4-trifluoromethoxyphenyl

Table 228 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- chloro-5-trifluoromethoxyphenyl

Table 229

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-3-chlorophenyl

Table 230

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-4-chlorophenyl

Table 231

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-5-chlorophenyl Table 232

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethoxy-4-chlorophenyl

Table 233 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-3-methylphenyl

Table 234

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-4-methylphenyl

Table 235

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-5-methylphenyl

Table 236

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-6-methylphenyl

Table 237

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-4-methylphenyl

Table 238

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-5-methylphenyl Table 239

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-3-bromophenyl

Table 240 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-4-bromophenyl

Table 241

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-5-bromophenyl

Table 242

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-4-bromophenyl

Table 243

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-3-difluoromethylphenyl Table 244

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-4-difluoromethylphenyl Table 245

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-5-difluoromethylphenyl Table 246

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-6-difluoromethylphenyl

Table 247 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-4-difluoromethylphenyl

Table 248

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-5-difluoromethylphenyl

Table 249

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-3-bromophenyl

Table 250

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-4-bromophenyl Table 251

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-5-bromophenyl

Table 252 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethyl-4-bromophenyl

Table 253

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-3-trifluoromethylphenyl

Table 254

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-4-trifluoromethylphenyl

Table 255

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-5-trifluoromethylphenyl

Table 256

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-6-trifluoromethylphenyl

Table 257

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-4-trifluoromethylphenyl Table 258

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-5-trifluoromethylphenyl

Table 259 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-3-bromophenyl

Table 260

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-4-bromophenyl

Table 261

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-5-bromophenyl

Table 262

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethyl-4-bromophenyl Table 263

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-3-methoxyphenyl Table 264

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-4-methoxyphenyl Table 265

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-5-methoxyphenyl

Table 266 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-6-methoxyphenyl

Table 267

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-4-methoxyphenyl

Table 268

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-5-methoxyphenyl

Table 269

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-3-bromophenyl Table 270

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-4-bromophenyl

Table 271 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-5-bromophenyl

Table 272

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methoxy-4-bromophenyl

Table 273

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-3-difluoromethoxyphenyl

Table 274

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-4-difluoromethoxyphenyl

Table 275

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-5-difluoromethoxyphenyl

Table 276

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-6-difluoromethoxyphenyl Table 277

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-4-difluoromethoxyphenyl

Table 278 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-5-difluoromethoxyphenyl

Table 279

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-3-bromophenyl

Table 280

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-4-bromophenyl

Table 281

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-5-bromophenyl Table 282

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethoxy-4-bromophenyl Table 283

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-3-trifluoromethoxyphenyl Table 284

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-4-trifluoromethoxyphenyl

Table 285 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-5-trifluoromethoxyphenyl

Table 286

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- bromo-6-trifluoromethoxyphenyl

Table 287

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-4-trifluoromethoxyphenyl

Table 288

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- bromo-5-trifluoromethoxyphenyl Table 289

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-3-bromophenyl

Table 290 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-4-bromophenyl

Table 291

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-5-bromophenyl

Table 292

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethoxy-4-bromophenyl

Table 293

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-3-difluoromethylphenyl

Table 294

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-4-difluoromethylphenyl

Table 295

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-5-difluoromethylphenyl Table 296

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-6-difluoromethylphenyl

Table 297 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-4-difluoromethylphenyl

Table 298

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-5-difluoromethylphenyl

Table 299

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-3-methylphenyl

Table 300

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-4-methylphenyl Table 301

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-5-methylphenyl Table 302

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethyl-4-methylphenyl Table 303

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-3-trifluoromethylphenyl

Table 304 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-4-trifluoromethylphenyl

Table 305

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-5-trifluoromethylphenyl

Table 306

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-6-trifluoromethylphenyl

Table 307

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-4-trifluoromethylphenyl Table 308

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-5-trifluoromethylphenyl

Table 309 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-3-methylphenyl

Table 310

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-4-methylphenyl

Table 31 1

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-5-methylphenyl

Table 312

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethyl-4-methylphenyl

Table 313

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-3-methoxyphenyl

Table 314

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-4-methoxyphenyl Table 315

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-5-methoxyphenyl

Table 316 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-6-methoxyphenyl

Table 317

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-4-methoxyphenyl

Table 318

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-5-methoxyphenyl

Table 319

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-3-methylphenyl Table 320

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-4-methylphenyl Table 321

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-5-methylphenyl Table 322

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methoxy-4-methylphenyl

Table 323 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-3-difluoromethoxyphenyl

Table 324

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-4-difluoromethoxyphenyl

Table 325

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-5-difluoromethoxyphenyl

Table 326

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-6-difluoromethoxyphenyl Table 327

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-4-difluoromethoxyphenyl

Table 328 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-5-difluoromethoxyphenyl

Table 329

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-3-methylphenyl

Table 330

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-4-methylphenyl

Table 331

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-5-methylphenyl

Table 332

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethoxy-4-methylphenyl

Table 333

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-3-trifluoromethoxyphenyl Table 334

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-4-trifluoromethoxyphenyl

Table 335 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-5-trifluoromethoxyphenyl

Table 336

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methyl-6-trifluoromethoxyphenyl

Table 337

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-4-trifluoromethoxyphenyl

Table 338

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methyl-5-trifluoromethoxyphenyl Table 339

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-3-methylphenyl Table 340

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-4-methylphenyl Table 341

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-5-methylphenyl

Table 342 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethoxy-4-methylphenyl

Table 343

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-3-trifluoromethylphenyl

Table 344

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-4-trifluoromethylphenyl

Table 345

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-5-trifluoromethylphenyl Table 346

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-6-trifluoromethylphenyl

Table 347 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethyl-4-trifluoromethylphenyl

Table 348

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethyl-5-trifluoromethylphenyl

Table 349

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-3-difluoromethylphenyl

Table 350

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-4-difluoromethylphenyl

Table 351

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-5-difluoromethylphenyl

Table 352

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethyl-4-difluoromethylphenyl Table 353

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-3-methoxyphenyl

Table 354 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-4-methoxyphenyl

Table 355

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-5-methoxyphenyl

Table 356

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-6-methoxyphenyl

Table 357

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethyl-4-methoxyphenyl Table 358

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethyl-5-methoxyphenyl Table 359

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-3-difluoromethylphenyl Table 360

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-4-difluoromethylphenyl

Table 361 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-5-difluoromethylphenyl

Table 362

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methoxy-4-difluoromethylphenyl

Table 363

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-3-difluoromethoxyphenyl

Table 364

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-4-difluoromethoxyphenyl Table 365

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-5-difluoromethoxyphenyl

Table 366 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-6-difluoromethoxyphenyl

Table 367

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethyl-4-difluoromethoxyphenyl

Table 368

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethyl-5-difluoromethoxyphenyl

Table 369

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-3-difluoromethylphenyl

Table 370

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-4-difluoromethylphenyl

Table 371

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-5-difluoromethylphenyl Table 372

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethoxy-4-difluoromethylphenyl

Table 373 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-3-trifluoromethoxyphenyl

Table 374

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-4-trifluoromethoxyphenyl

Table 375

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-5-trifluoromethoxyphenyl

Table 376

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethyl-6-trifluoromethoxyphenyl Table 377

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethyl-4-trifluoromethoxyphenyl Table 378

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethyl-5-trifluoromethoxyphenyl Table 379

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-3-difluoromethylphenyl

Table 380 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-4-difluoromethylphenyl

Table 381

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-5-difluoromethylphenyl

Table 382

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethoxy-4-difluoromethylphenyl

Table 383

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-3-methoxyphenyl Table 384

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-4-methoxyphenyl

Table 385 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-5-methoxyphenyl

Table 386

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-6-methoxyphenyl

Table 387

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethyl-4-methoxyphenyl

Table 388

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethyl-5-methoxyphenyl

Table 389

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-3-trifluoromethylphenyl

Table 390

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-4-trifluoromethylphenyl Table 391

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-5-trifluoromethylphenyl

Table 392 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methoxy-4-trifluoromethylphenyl

Table 393

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-3-difluoromethoxyphenyl

Table 394

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-4-difluoromethoxyphenyl

Table 395

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-5-difluoromethoxyphenyl Table 396

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-6-difluoromethoxyphenyl Table 397

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethyl-4-difluoromethoxyphenyl Table 398

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethyl-5-difluoromethoxyphenyl

Table 399 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-3-trifluoromethylphenyl

Table 400

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-4-trifluoromethylphenyl

Table 401

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-5-trifluoromethylphenyl

Table 402

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethoxy-4-trifluoromethylphenyl Table 403

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-3-trifluoromethoxyphenyl

Table 404 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-4-trifluoromethoxyphenyl

Table 405

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-5-trifluoromethoxyphenyl

Table 406

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethyl-6-trifluoromethoxyphenyl

Table 407

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethyl-4-trifluoromethoxyphenyl

Table 408

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethyl-5-trifluoromethoxyphenyl

Table 409

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-3-trifluoromethylphenyl Table 410

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-4-trifluoromethylphenyl

Table 41 1 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-5-trifluoromethylphenyl

Table 412

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethoxy-4-trifluoromethylphenyl

Table 413

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-3-difluoromethoxyphenyl

Table 414

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-4-difluoromethoxyphenyl Table 415

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-5-difluoromethoxyphenyl Table 416

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-6-difluoromethoxyphenyl Table 417

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methoxy-4-difluoromethoxyphenyl

Table 418 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methoxy-5-difluoromethoxyphenyl

Table 419

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-3-methoxyphenyl

Table 420

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-4-methoxyphenyl

Table 421

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-5-methoxyphenyl Table 422

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethoxy-4-methoxyphenyl

Table 423 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-3-trifluoromethoxyphenyl

Table 424

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-4-trifluoromethoxyphenyl

Table 425

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-5-trifluoromethoxyphenyl

Table 426

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- methoxy-6-trifluoromethoxyphenyl

Table 427

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methoxy-4-trifluoromethoxyphenyl

Table 428

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- methoxy-5-trifluoromethoxyphenyl Table 429

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-3-methoxyphenyl

Table 430 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-4-methoxyphenyl

Table 431

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-5-methoxyphenyl

Table 432

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethoxy-4-methoxyphenyl

Table 433

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-3-trifluoromethoxyphenyl Table 434

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-4-trifluoromethoxyphenyl Table 435

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-5-trifluoromethoxyphenyl Table 436

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- difluoromethoxy-6-trifluoromethoxyphenyl

Table 437 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethoxy-4-trifluoromethoxyphenyl

Table 438

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- difluoromethoxy-5-trifluoromethoxyphenyl

Table 439

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-3-difluoromethoxyphenyl

Table 440

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-4-difluoromethoxyphenyl Table 441

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2- trifluoromethoxy-5-difluoromethoxyphenyl

Table 442 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 3- trifluoromethoxy-4-difluoromethoxyphenyl

Table 443

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,4-trifluorophenyl

Table 444

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,5-trifluorophenyl

Table 445

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,6-trifluorophenyl

Table 446

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4,5-trifluorophenyl

Table 447

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,4,6-trifluorophenyl Table 448

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

3,4,5-trifluorophenyl

Table 449 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,4-trichlorophenyl

Table 450

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,5-trichlorophenyl

Table 451

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,3,6-trichlorophenyl

Table 452

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,4,5-trichlorophenyl Table 453

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,4,6-trichlorophenyl Table 454

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

3,4,5-trichlorophenyl Table 455

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,4-tribromophenyl

Table 456 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,5-tribromophenyl

Table 457

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,6-tribromophenyl

Table 458

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4,5-tribromophenyl

Table 459

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,4,6-tribromophenyl Table 460

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

3,4,5-tribromophenyl

Table 461 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,4-trimethylphenyl

Table 462

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,5-trimethylphenyl

Table 463

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,6-trimethylphenyl

Table 464

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,4,5-trimethylphenyl

Table 465

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4,6-trimethylphenyl

Table 466

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

3,4,5-trimethylphenyl Table 467

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,4-tri-(trifluoromethyl)-phenyl

Table 468 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,5-tri-(trifluoromethyl)-phenyl

Table 469

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,3,6-tri-(trifluoromethyl)-phenyl

Table 470

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,4,5-tri-(trifluoromethyl)-phenyl

Table 471

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

2,4,6-tri-(trifluoromethyl)-phenyl Table 472

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is

3,4,5-tri-(trifluoromethyl)-phenyl Table 473

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- difluoro-4-chlorophenyl Table 474

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- difluoro-4-methylphenyl

Table 475 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- difluoro-4-trifluoromethylphenyl

Table 476

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- difluoro-4-methoxyphenyl

Table 477

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- difluoro-4-trifluoromethoxyphenyl

Table 478

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- dichloro-4-fluorophenyl Table 479

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- dichloro-4-methylphenyl

Table 480 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- dichloro-4-trifluoromethylphenyl

Table 481

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- dichloro-4-methoxyphenyl

Table 482

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is H and R ³ is 2,6- dichloro-4-trifluoromethoxyphenyl

Tables 483 to 964

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is methyl

Tables 965 to 1446

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is ethyl

Tables 1447 to 1928

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is propyl Tables 1929 to 2410

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is isopropyl

Tables 2411 to 2892 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is n-butyl

Tables 2893 to 3374

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is sec-butyl

Tables 3375 to 3856

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is isobutyl

Tables 3857 to 4338

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is tert-butyl Tables 4339 to 4820

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is phenyl Tables 4821 to 5302

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is 4-methylphenyl Tables 5303 to 5784

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is benzyl

Tables 5785 to 6266 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is Li ⁺

Tables 6267 to 6748

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is Na ⁺

Tables 6749 to 7230

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is K ⁺

Tables 7231 to 7712

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is Y ₂ Mg ²⁺ Tables 7713 to 8194

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is Y ₂ Cu ²⁺

Tables 8195 to 8676 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is Y ₂ Zn ²⁺

Tables 8677 to 9158

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is Y ₂ Fe ²⁺

Tables 9159 to 9640

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is Y ₂ Ni ²⁺

Tables 9641 to 10122

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is NH(CHs) ₃ ⁺

Tables 10123 to 10604

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is NH(C ₂ Hs) ₃ ⁺

Tables 10605 to 11086

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is NH(CH ₂ CH ₂ CH ₂ ) ₃ ⁺ Tables 1 1087 to 11568

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is NH(CH(CH ₃ ) ₂ ) ₃ ⁺

Tables 11569 to 12050 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is NH(CH ₂ CH ₂ CH ₂ CH ₂ ) ₃ ⁺

Tables 12051 to 12532

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is methylcarbonyl

Tables 12533 to 13014

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is ethylcarbonyl

Tables 13015 to 13496

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is propylcarbonyl Tables 13497 to 13978

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is isopropylcarbonyl Tables 13979 to 14460

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is phenylcarbonyl Tables 14461 to 14942

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is methoxycarbonyl

Tables 14943 to 15424 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is ethoxycarbonyl

Tables 15425 to 15906

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is propoxycarbonyl

Tables 15907 to 16388

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is isopropoxycarbonyl

Tables 16389 to 16870

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is phenoxycarbonyl Tables 16871 to 17352

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is methylaminocarbonyl

Tables 17353 to 17834 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is ethylaminocarbonyl

Tables 17835 to 18316

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is propylaminocarbonyl

Tables 18317 to 18798

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is isopropylaminocarbonyl

Tables 18799 to 19280

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is phenylaminocarbonyl

Tables 19281 to 19762

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is methylsulfonyl

Tables 19763 to 20244

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is ethylsulfonyl Tables 20245 to 20726

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is propylsulfonyl

Tables 20727 to 21208 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is isopropylsulfonyl

Tables 21209 to 21690

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is phenylsulfonyl

Tables 21691 to 22172

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is methoxysulfonyl

Tables 22173 to 22654

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is ethoxysulfonyl Tables 22655 to 23136

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is propoxysulfonyl Tables 23137 to 23618

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is isopropoxysulfonyl Tables 23619 to 24100

Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is phenoxysulfonyl

Tables 24101 to 24582 Compounds of the formula I.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ⁵ is CN

Tables 24583 to 25064

Compounds of the formula I.A2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A and R ³ is as defined in any of tables 1 to 482

Tables 25065 to 25546

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is H

Tables 25547 to 26028

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is methyl Tables 26029 to 26510

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is ethyl

Tables 2651 1 to 26992 Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is propyl

Tables 26993 to 27474

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is isopropyl

Tables 27475 to 27956

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is n-butyl

Tables 27957 to 28438

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is sec-butyl

Tables 28439 to 28920

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is isobutyl

Tables 28921 to 29402

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is tert-butyl Tables 29403 to 29884

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is phenyl

Tables 29885 to 30366 Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is 4-methylphenyl

Tables 30367 to 30848

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is benzyl

Tables 30849 to 31330

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is methylcarbonyl

Tables 31331 to 31812

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is ethylcarbonyl Tables 31813 to 32294

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is propylcarbonyl Tables 32295 to 32776

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is isopropylcarbonyl Tables 32777 to 33258

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is phenylcarbonyl

Tables 33259 to 33740 Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is methoxycarbonyl

Tables 33741 to 34222

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is ethoxycarbonyl

Tables 34223 to 34704

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is propoxycarbonyl

Tables 34705 to 35186

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is isopropoxycarbonyl Tables 35187 to 35668

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is phenoxycarbonyl

Tables 35669 to 36150 Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is methylaminocarbonyl

Tables 36151 to 36632

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is ethylaminocarbonyl

Tables 36633 to 37114

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is propylaminocarbonyl

Tables 37115 to 37596

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is isopropylaminocarbonyl

Tables 37597 to 38078

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is phenylaminocarbonyl

Tables 38079 to 38560

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is methylsulfonyl Tables 38561 to 39042

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is ethylsulfonyl

Tables 39043 to 39524 Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is propylsulfonyl

Tables 39525 to 40006

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is isopropylsulfonyl

Tables 40007 to 40488

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is phenylsulfonyl

Tables 40489 to 40970

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is methoxysulfonyl Tables 40971 to 41452

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is ethoxysulfonyl Tables 41453 to 41934

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is propoxysulfonyl

Tables 41935 to 42416

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is isopropoxysulfonyl

Tables 42417 to 42898

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is phenoxysulfonyl

Tables 42899 to 43380

Compounds of the formula II.A1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ³ is as defined in any of tables 1 to 482 and R ^5a is CN

In the above tables 1 to 482, the given positions of the substituents on the phenyl ring (e.g. 2-fluoro) are to be understood as relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

Table A

In another preferred embodiment of the invention (embodiment B), R ¹ is a group of formula V, where

R ² is aryl which may carry 1 , 2, 3, 4 or 5 substituents R ⁷ , or is a 5- or 6-membered heteroaromatic ring containing 1 , 2 or 3 heteroatoms selected from N, O and S as ring members, where the heteroaromatic ring may carry 1 , 2, 3 or 4 substituents R ⁸ ; R ³ is selected from Ci-Cio-alkyl, Ci-Cio-haloalkyl, aryl and aryl-Ci-C4-alkyl, where the aryl moiety in the 2 last-mentioned radicals may carry 1 , 2, 3, 4 or 5 substitu- ents R ¹¹ ; R ⁴ is CN; and R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings; except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl, 4-chlorophenyl, 2,4-dichlorophenyl, 4-bromophenyl, 4-tert-butylphenyl or 4-biphenyl, R ³ is n-butyl and R ⁴ is CN; except for compounds wherein R ² is 2-chlorophenyl, 4-chlorophenyl, 2,4-dichlorophenyl, 2,4,6-trichlorophenyl, 4-trifluoromethylphenyl or 2-difluoromethoxyphenyl, R ³ is tert-butyl and R ⁴ is CN; and except for compounds wherein R ² is 4-chlorophenyl, R ³ is 2-fluoromethylprop-2-yl, 1 ,3- difluoro-2-methylprop-2-yl, 4-chlorophenyl, 4-chlorophenyl-methyl, 4-chlorophenyl-1- ethyl, 4-chlorophenyl-2-ethyl or 4-fluorophenyl-2-ethyl, and R ⁴ is CN.

In this embodiment B, aryl is preferably phenyl.

In a more preferred embodiment of the invention (embodiment B.1 ), R ¹ is a group of formula V, where

R ² is aryl, preferably phenyl, which may carry 1 , 2 or 3 substituents R ⁷ ;

R ³ is selected from Ci-Cβ-alkyl, Ci-C4-haloalkyl, phenyl and phenyl-Ci-C4-alkyl, where the phenyl moiety in the 2 last-mentioned radicals may carry 1 , 2 or 3 substituents R ¹¹ ; R ⁴ is CN; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH3, CHF2, CF3, OCH ₃ , OCHF ₂ and OCF ₃ ; and each R ¹¹ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C ₄ -haloalkoxy, and preferably from F, Cl, Br, CH ₃ , CHF ₂ , CF ₃ ,

OCH ₃ , OCHF ₂ and OCF ₃ ; except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl, 4-chlorophenyl, 2,4-dichlorophenyl, 4-bromophenyl, 4-tert-butylphenyl or 4-biphenyl, R ³ is n-butyl and R ⁴ is CN; except for compounds wherein R ² is 2-chlorophenyl, 4-chlorophenyl, 2,4-dichlorophenyl, 2,4,6-trichlorophenyl, 4-trifluoromethylphenyl or 2-difluoromethoxyphenyl, R ³ is tert-butyl and R ⁴ is CN; and except for compounds wherein R ² is 4-chlorophenyl, R ³ is 2-fluoromethylprop-2-yl, 1 ,3- difluoro-2-methylprop-2-yl, 4-chlorophenyl, 4-chlorophenyl-methyl, 4-chlorophenyl-1- ethyl, 4-chlorophenyl-2-ethyl or 4-fluorophenyl-2-ethyl, and R ⁴ is CN.

In an even more preferred embodiment of the invention (embodiment B.1.1 ), R ¹ is a group of formula V, where

R ² phenyl which may carry 1 , 2 or 3 substituents R ⁷ ; R ³ is selected from Ci-Cβ-alkyl and phenyl-Ci-C4-alkyl, where the phenyl moiety may carry 1 , 2 or 3 substituents R ¹¹ ; R ⁴ is CN; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH3, CHF2, CF3, OCH ₃ , OCHF ₂ and OCF ₃ ; and each R ¹¹ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH ₃ , CHF2, CF ₃ ,

OCH ₃ , OCHF ₂ and OCF ₃ ; except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl, 4-chlorophenyl, 2,4-dichlorophenyl, 4-bromophenyl, 4-tert-butylphenyl or 4-biphenyl, R ³ is n-butyl and R ⁴ is CN; except for compounds wherein R ² is 2-chlorophenyl, 4-chlorophenyl, 2,4-dichlorophenyl, 2,4,6-trichlorophenyl, 4-trifluoromethylphenyl or 2-difluoromethoxyphenyl, R ³ is tert-butyl and R ⁴ is CN; and except for compounds wherein R ² is 4-chlorophenyl, R ³ is 2-fluoromethylprop-2-yl, 1 ,3- difluoro-2-methylprop-2-yl, 4-chlorophenyl, 4-chlorophenyl-methyl, 4-chlorophenyl-1- ethyl, 4-chlorophenyl-2-ethyl or 4-fluorophenyl-2-ethyl, and R ⁴ is CN.

If R ² is phenyl which carries 1 substituent R ⁷ , this is preferably bound in 2- or 4- position, more preferably in 2-position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

If R ³ is phenyl which carries 1 substituent R ¹¹ , this is preferably bound in 2- opposition, more preferably in 2-position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule. If R ³ is phenyl-Ci-C4-alkyl, where the phenyl moiety carries 1 substituent R ¹¹ , this is preferably bound in 2- or 4-position, more preferably in 2-position, relative to the 1 -position of the attachment point of the phenyl ring to the Ci-C4-alkyl group. If R ² is phenyl which carries 2 substituents R ⁷ , these are preferably bound in 2,4- position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

If R ³ is phenyl which carries 2 substituents R ¹¹ , these are preferably bound in 2,4- position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule. If R ³ is phenyl-Ci-C4-alkyl, where the phenyl moiety carries 2 substituents R ¹¹ , these are preferably bound in 2,4-position, relative to the 1-position of the attachment point of the phenyl ring to the Ci-C4-alkyl group.

Particular compounds of this embodiment B are compounds I or II, wherein

- R ⁵ or R ^5a are H, m is 0, R ⁴ is CN, R ³ is n-butyl and R ² is 2,4-difluorophenyl;

- R ⁵ or R ^5a are H, m is 0, R ⁴ is CN, R ³ is n-butyl and R ² is 3,4-difluorophenyl; - R ⁵ or R ^5a are H, m is 0, R ⁴ is CN, R ³ is n-butyl and R ² is 2-chloro-4-fluorophenyl;

- R ⁵ or R ^5a are H, m is 0, R ⁴ is CN, R ³ is n-butyl and R ² is 4-chloro-2-fluorophenyl.

Examples for preferred compounds I and Il of embodiment B are compounds of formulae I.B1 to I.B8 and II.B1 to II. B4, where the variables R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ are hydrogen or have one of the general or, in particular, one of the preferred meanings given above for R ⁷ , where the variables R ⁵ and R ^5a have one of the general or, in particular, one of the preferred meanings given above, where the variable R ³¹ has one of the preferred meanings given above for R ³ in context with embodiment B, but except for the meaning aryl and aryl-i-C4-alkyl, and the variable R ³² is aryl as defined above for R ³ in context with embodiment B. Examples of preferred compounds are the individual compounds compiled in the tables 1 to 184092 below. Moreover, the meanings mentioned below for the individual variables in the tables are per se, independently of the combination in which they are mentioned, a particularly preferred embodiment of the substituents in question.

(I B1 ) (I B2) (I B3) (I B4)

R ^5a R ^5a R ^5a R ^5a

(Il B1 ) (Il B2) (Il B3) (M B ₄ )

Table 1

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is H Table 2

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is methyl

Table 3 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is ethyl

Table 4

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is propyl

Table 5

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is isopropyl

Table 6

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is n-butyl

Table 7

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is sec-butyl

Table 8

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is isobutyl

Table 9

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is tert-butyl Table 10

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is phenyl

Table 11 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is 4-methylphenyl

Table 12

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is benzyl

Table 13

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is Li ⁺

Table 14

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is Na ⁺ Table 15

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is K ⁺ Table 16

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is Y ₂ Mg ²⁺ Table 17

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is ¹ / ₂ Cu ²⁺

Table 18 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is ¹ / ₂ Zn ²⁺

Table 19

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is ¹ / ₂ Fe ²⁺

Table 20

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is ¹ / ₂ Ni ²⁺

Table 21

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is NH(CHs) ₃ ⁺ Table 22

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is NH(C ₂ Hs) ₃ ⁺

Table 23 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is NH(CH ₂ CH ₂ CH ₂ ) ₃ ⁺

Table 24

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is NH(CH(CH ₃ ) ₂ ) ₃ ⁺

Table 25 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is NH(CH ₂ CH ₂ CH ₂ CH ₂ )S ⁺

Table 26 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is methylcarbonyl

Table 27

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is ethylcarbonyl

Table 28

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is propylcarbonyl

Table 29

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is isopropylcarbonyl Table 30

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is methoxycarbonyl

Table 31 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is ethoxycarbonyl

Table 32

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is propoxycarbonyl

Table 33

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is isopropoxycarbonyl

Table 34

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is phenoxycarbonyl Table 35

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is methylaminocarbonyl Table 36

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is ethylaminocarbonyl

Table 37 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is propylaminocarbonyl

Table 38

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is isopropylaminocarbonyl

Table 39

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is phenylaminocarbonyl

Table 40

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is methylsulfonyl Table 41

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is ethylsulfonyl

Table 42 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is propylsulfonyl

Table 43

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is isopropylsulfonyl

Table 44 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is phenylsulfonyl

Table 45 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is methoxysulfonyl

Table 46

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is ethoxysulfonyl

Table 47

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is propoxysulfonyl

Table 48

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is isopropoxysulfonyl Table 49

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is phenoxysulfonyl

Table 50 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ⁵ is CN

Tables 51 to 100

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³¹ is ethyl

Tables 101 to 150

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³¹ is propyl

Tables 151 to 200

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³¹ is isopropyl Tables 201 to 250

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³¹ is n-butyl Tables 251 to 300

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³¹ is sec-butyl

Tables 301 to 350 Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³¹ is isobutyl

Tables 351 to 400

Compounds of the formula I.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³¹ is tert-butyl

Tables 401 to 450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is phenyl

Tables 451 to 500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluorophenyl Tables 501 to 550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluorophenyl

Tables 551 to 600 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 4-fluorophenyl

Tables 601 to 650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chlorophenyl

Tables 651 to 700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chlorophenyl

Tables 701 to 750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 4-chlorophenyl

Tables 751 to 800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromophenyl

Tables 801 to 850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromophenyl Tables 851 to 900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 4-bromophenyl

Tables 901 to 950 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methylphenyl

Tables 951 to 1000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methylphenyl

Tables 1001 to 1050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 4-methylphenyl

Tables 1051 to 1 100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-(difluoromethyl)-phenyl Tables 1 101 to 1150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-(difluoromethyl)-phenyl Tables 1 151 to 1200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 4-(difluoromethyl)-phenyl Tables 1201 to 1250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-(trifluoromethyl)-phenyl

Tables 1251 to 1300 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-(trifluoromethyl)-phenyl

Tables 1301 to 1350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 4-(trifluoromethyl)-phenyl

Tables 1351 to 1400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxyphenyl

Tables 1401 to 1450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methoxyphenyl Tables 1451 to 1500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 4-methoxyphenyl

Tables 1501 to 1550 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-(difluoromethoxy)-phenyl

Tables 1551 to 1600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-(difluoromethoxy)-phenyl

Tables 1601 to 1650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 4-(difluoromethoxy)-phenyl

Tables 1651 to 1700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-(trifluoromethoxy)-phenyl

Tables 1701 to 1750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-(trifluoromethoxy)-phenyl

Tables 1751 to 1800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 4-(trifluoromethoxy)-phenyl Tables 1801 to 1850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,3-difluorophenyl

Tables 1851 to 1900 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,4-difluorophenyl

Tables 1901 to 1950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,5-difluorophenyl

Tables 1951 to 2000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,6-difluorophenyl

Tables 2001 to 2050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,4-difluorophenyl Tables 2051 to 2100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,5-difluorophenyl Tables 2101 to 2150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,3-dichlorophenyl Tables 2151 to 2200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,4-dichlorophenyl

Tables 2201 to 2250 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,5-dichlorophenyl

Tables 2251 to 2300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,6-dichlorophenyl

Tables 2301 to 2350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,4-dichlorophenyl

Tables 2351 to 2400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,5-dichlorophenyl Tables 2401 to 2450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,3-dibromophenyl

Tables 2451 to 2500 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,4-dibromophenyl

Tables 2501 to 2550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,5-dibromophenyl

Tables 2551 to 2600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,6-dibromophenyl

Tables 2601 to 2650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,4-dibromophenyl

Tables 2651 to 2700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,5-dibromophenyl

Tables 2701 to 2750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,3-dimethylphenyl Tables 2751 to 2800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,4-dimethylphenyl

Tables 2801 to 2850 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,5-dimethylphenyl

Tables 2851 to 2900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,6-dimethylphenyl

Tables 2901 to 2950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,4-dimethylphenyl

Tables 2951 to 3000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,5-dimethylphenyl Tables 3001 to 3050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,3-di-(difluoromethyl)-phenyl Tables 3051 to 3100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,4-di-(difluoromethyl)-phenyl Tables 3101 to 3150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,5-di-(difluoromethyl)-phenyl

Tables 3151 to 3200 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,6-di-(difluoromethyl)-phenyl

Tables 3201 to 3250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,4-di-(difluoromethyl)-phenyl

Tables 3251 to 3300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,5-di-(difluoromethyl)-phenyl

Tables 3301 to 3350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,3-di-(trifluoromethyl)-phenyl Tables 3351 to 3400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,4-di-(trifluoromethyl)-phenyl

Tables 3401 to 3450 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,5-di-(trifluoromethyl)-phenyl

Tables 3451 to 3500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,6-di-(trifluoromethyl)-phenyl

Tables 3501 to 3550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,4-di-(trifluoromethyl)-phenyl

Tables 3551 to 3600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,5-di-(trifluoromethyl)-phenyl

Tables 3601 to 3650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,3-dimethoxyphenyl

Tables 3651 to 3700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,4-dimethoxyphenyl Tables 3701 to 3750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,5-dimethoxyphenyl

Tables 3751 to 3800 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,6-dimethoxyphenyl

Tables 3801 to 3850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,4-dimethoxyphenyl

Tables 3851 to 3900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,5-dimethoxyphenyl

Tables 3901 to 3950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,3-di-(difluoromethoxy)-phenyl Tables 3951 to 4000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,4-di-(difluoromethoxy)-phenyl Tables 4001 to 4050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,5-di-(difluoromethoxy)-phenyl Tables 4051 to 4100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,6-di-(difluoromethoxy)-phenyl Tables 4101 to 4150 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,4-di-(difluoromethoxy)-phenyl Tables 4151 to 4200 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,5-di-(difluoromethoxy)-phenyl Tables 4201 to 4250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,3-di-(trifluoromethoxy)-phenyl Tables 4251 to 4300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,4-di-(trifluoromethoxy)-phenyl Tables 4301 to 4350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,5-di-(trifluoromethoxy)-phenyl Tables 4351 to 4400 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2,6-di-(trifluoromethoxy)-phenyl Tables 4401 to 4450 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,4-di-(trifluoromethoxy)-phenyl Tables 4451 to 4500 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3,5-di-(trifluoromethoxy)-phenyl

Tables 4501 to 4550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-3-chlorophenyl

Tables 4551 to 4600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-4-chlorophenyl

Tables 4601 to 4650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-5-chlorophenyl Tables 4651 to 4700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-6-chlorophenyl

Tables 4701 to 4750 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-4-chlorophenyl

Tables 4751 to 4800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-5-chlorophenyl

Tables 4801 to 4850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-3-fluorophenyl

Tables 4851 to 4900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-4-fluorophenyl Tables 4901 to 4950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-5-fluorophenyl Tables 4951 to 5000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-4-fluorophenyl Tables 5001 to 5050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-3-bromophenyl

Tables 5051 to 5100 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-4-bromophenyl

Tables 5101 to 5150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-5-bromophenyl

Tables 5151 to 5200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-6-bromophenyl

Tables 5201 to 5250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-4-bromophenyl Tables 5251 to 5300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-5-bromophenyl

Tables 5301 to 5350 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-3-fluorophenyl

Tables 5351 to 5400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-4-fluorophenyl

Tables 5401 to 5450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-5-fluorophenyl

Tables 5451 to 5500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-4-fluorophenyl

Tables 5501 to 5550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-3-methylphenyl

Tables 5551 to 5600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-4-methylphenyl Tables 5601 to 5650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-5-methylphenyl

Tables 5651 to 5700 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-6-methylphenyl

Tables 5701 to 5750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-4-methylphenyl

Tables 5751 to 5800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-5-methylphenyl

Tables 5801 to 5850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-3-fluorophenyl Tables 5851 to 5900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-4-fluorophenyl Tables 5901 to 5950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-5-fluorophenyl Tables 5951 to 6000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-4-fluorophenyl

Tables 6001 to 6050 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-3-difluoromethylphenyl

Tables 6051 to 6100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-4-difluoromethylphenyl

Tables 6101 to 6150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-5-difluoromethylphenyl

Tables 6151 to 6200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-6-difluoromethylphenyl Tables 6201 to 6250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-4-difluoromethylphenyl

Tables 6251 to 6300 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-5-difluoromethylphenyl

Tables 6301 to 6350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-3-fluorophenyl

Tables 6351 to 6400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-4-fluorophenyl Tables 6401 to 6450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-5-fluorophenyl Tables 6451 to 6500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethyl-4-fluorophenyl Tables 6501 to 6550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-3-trifluoromethylphenyl Tables 6551 to 6600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-4-trifluoromethylphenyl Tables 6601 to 6650 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-5-trifluoromethylphenyl Tables 6651 to 6700 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-6-trifluoromethylphenyl Tables 6701 to 6750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-4-trifluoromethylphenyl Tables 6751 to 6800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-5-trifluoromethylphenyl Tables 6801 to 6850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-3-fluorophenyl Tables 6851 to 6900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-4-fluorophenyl Tables 6901 to 6950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-5-fluorophenyl

Tables 6951 to 7000 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethyl-4-fluorophenyl

Tables 7001 to 7050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-3-methoxyphenyl

Tables 7051 to 7100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-4-methoxyphenyl

Tables 7101 to 7150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-5-methoxyphenyl Tables 7151 to 7200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-6-methoxyphenyl

Tables 7201 to 7250 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-4-methoxyphenyl

Tables 7251 to 7300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-5-methoxyphenyl

Tables 7301 to 7350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-3-fluorophenyl

Tables 7351 to 7400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-4-fluorophenyl

Tables 7401 to 7450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-5-fluorophenyl

Tables 7451 to 7500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methoxy-4-fluorophenyl Tables 7501 to 7550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-3-difluoromethoxyphenyl

Tables 7551 to 7600 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-4-difluoromethoxyphenyl

Tables 7601 to 7650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-5-difluoromethoxyphenyl

Tables 7651 to 7700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-6-difluoromethoxyphenyl

Tables 7701 to 7750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-4-difluoromethoxyphenyl Tables 7751 to 7800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-5-difluoromethoxyphenyl Tables 7801 to 7850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-3-fluorophenyl Tables 7851 to 7900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-4-fluorophenyl Tables 7901 to 7950 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-5-fluorophenyl Tables 7951 to 8000 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethoxy-4-fluorophenyl Tables 8001 to 8050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-3-trifluoromethoxyphenyl Tables 8051 to 8100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-4-trifluoromethoxyphenyl Tables 8101 to 8150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-5-trifluoromethoxyphenyl Tables 8151 to 8200 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-fluoro-6-trifluoromethoxyphenyl Tables 8201 to 8250 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-4-trifluoromethoxyphenyl Tables 8251 to 8300 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-fluoro-5-trifluoromethoxyphenyl

Tables 8301 to 8350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-3-fluorophenyl

Tables 8351 to 8400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-4-fluorophenyl

Tables 8401 to 8450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-5-fluorophenyl Tables 8451 to 8500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethoxy-4-fluorophenyl

Tables 8501 to 8550 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-3-bromophenyl

Tables 8551 to 8600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-4-bromophenyl

Tables 8601 to 8650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-5-bromophenyl

Tables 8651 to 8700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-6-bromophenyl Tables 8701 to 8750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-4-bromophenyl Tables 8751 to 8800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-5-bromophenyl Tables 8801 to 8850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-3-chlorophenyl

Tables 8851 to 8900 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-4-chlorophenyl

Tables 8901 to 8950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-5-chlorophenyl

Tables 8951 to 9000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-4-chlorophenyl

Tables 9001 to 9050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-3-methylphenyl Tables 9051 to 9100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-4-methylphenyl

Tables 9101 to 9150 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-5-methylphenyl

Tables 9151 to 9200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-6-methylphenyl

Tables 9201 to 9250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-4-methylphenyl

Tables 9251 to 9300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-5-methylphenyl

Tables 9301 to 9350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-3-chlorophenyl

Tables 9351 to 9400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-4-chlorophenyl Tables 9401 to 9450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-5-chlorophenyl

Tables 9451 to 9500 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-4-chlorophenyl

Tables 9501 to 9550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-3-difluoromethylphenyl

Tables 9551 to 9600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-4-difluoromethylphenyl

Tables 9601 to 9650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-5-difluoromethylphenyl Tables 9651 to 9700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-6-difluoromethylphenyl Tables 9701 to 9750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-4-difluoromethylphenyl Tables 9751 to 9800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-5-difluoromethylphenyl Tables 9801 to 9850 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-3-chlorophenyl Tables 9851 to 9900 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-4-chlorophenyl Tables 9901 to 9950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-5-chlorophenyl Tables 9951 to 10000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethyl-4-chlorophenyl Tables 10001 to 10050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-3-trifluoromethylphenyl Tables 10051 to 10100 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-4-trifluoromethylphenyl Tables 10101 to 10150 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-5-trifluoromethylphenyl Tables 10151 to 10200 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-6-trifluoromethylphenyl

Tables 10201 to 10250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-4-trifluoromethylphenyl

Tables 10251 to 10300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-5-trifluoromethylphenyl

Tables 10301 to 10350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-3-chlorophenyl Tables 10351 to 10400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-4-chlorophenyl

Tables 10401 to 10450 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-5-chlorophenyl

Tables 10451 to 10500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethyl-4-chlorophenyl

Tables 10501 to 10550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-3-methoxyphenyl

Tables 10551 to 10600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-4-methoxyphenyl Tables 10601 to 10650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-5-methoxyphenyl Tables 10651 to 10700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-6-methoxyphenyl Tables 10701 to 10750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-4-methoxyphenyl

Tables 10751 to 10800 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-5-methoxyphenyl

Tables 10801 to 10850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-3-chlorophenyl

Tables 10851 to 10900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-4-chlorophenyl

Tables 10901 to 10950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-5-chlorophenyl Tables 10951 to 1 1000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methoxy-4-chlorophenyl

Tables 11001 to 11050 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-3-difluoromethoxyphenyl

Tables 11051 to 11 100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-4-difluoromethoxyphenyl

Tables 11 101 to 11 150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-5-difluoromethoxyphenyl Tables 1 1 151 to 11200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-6-difluoromethoxyphenyl Tables 11201 to 11250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-4-difluoromethoxyphenyl Tables 11251 to 11300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-5-difluoromethoxyphenyl Tables 1 1301 to 11350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-3-chlorophenyl Tables 11351 to 11400 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-4-chlorophenyl Tables 11401 to 11450 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-5-chlorophenyl Tables 11451 to 11500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethoxy-4-chlorophenyl Tables 11501 to 11550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-3-trifluoromethoxyphenyl Tables 1 1551 to 11600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-4-trifluoromethoxyphenyl Tables 1 1601 to 11650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-5-trifluoromethoxyphenyl Tables 1 1651 to 11700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-chloro-6-trifluoromethoxyphenyl Tables 11701 to 11750 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-4-trifluoromethoxyphenyl Tables 11751 to 11800 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-chloro-5-trifluoromethoxyphenyl Tables 11801 to 11850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-3-chlorophenyl Tables 11851 to 11900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-4-chlorophenyl Tables 1 1901 to 1 1950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-5-chlorophenyl Tables 11951 to 12000 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethoxy-4-chlorophenyl Tables 12001 to 12050 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-3-methylphenyl Tables 12051 to 12100 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-4-methylphenyl

Tables 12101 to 12150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-5-methylphenyl

Tables 12151 to 12200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-6-methylphenyl

Tables 12201 to 12250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-4-methylphenyl Tables 12251 to 12300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-5-methylphenyl

Tables 12301 to 12350 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-3-bromophenyl

Tables 12351 to 12400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-4-bromophenyl

Tables 12401 to 12450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-5-bromophenyl

Tables 12451 to 12500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-4-bromophenyl Tables 12501 to 12550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-3-difluoromethylphenyl Tables 12551 to 12600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-4-difluoromethylphenyl Tables 12601 to 12650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-5-difluoromethylphenyl Tables 12651 to 12700 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-6-difluoromethylphenyl Tables 12701 to 12750 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-4-difluoromethylphenyl Tables 12751 to 12800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-5-difluoromethylphenyl Tables 12801 to 12850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-3-bromophenyl Tables 12851 to 12900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-4-bromophenyl Tables 12901 to 12950 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-5-bromophenyl Tables 12951 to 13000 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethyl-4-bromophenyl Tables 13001 to 13050 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-3-trifluoromethylphenyl Tables 13051 to 13100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-4-trifluoromethylphenyl Tables 13101 to 13150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-5-trifluoromethylphenyl Tables 13151 to 13200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-6-trifluoromethylphenyl Tables 13201 to 13250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-4-trifluoromethylphenyl Tables 13251 to 13300 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-5-trifluoromethylphenyl Tables 13301 to 13350 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-3-bromophenyl Tables 13351 to 13400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-4-bromophenyl Tables 13401 to 13450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-5-bromophenyl Tables 13451 to 13500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethyl-4-bromophenyl Tables 13501 to 13550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-3-methoxyphenyl Tables 13551 to 13600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-4-methoxyphenyl

Tables 13601 to 13650 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-5-methoxyphenyl

Tables 13651 to 13700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-6-methoxyphenyl

Tables 13701 to 13750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-4-methoxyphenyl

Tables 13751 to 13800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-5-methoxyphenyl Tables 13801 to 13850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-3-bromophenyl

Tables 13851 to 13900 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-4-bromophenyl

Tables 13901 to 13950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-5-bromophenyl

Tables 13951 to 14000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methoxy-4-bromophenyl Tables 14001 to 14050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-3-difluoromethoxyphenyl Tables 14051 to 14100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-4-difluoromethoxyphenyl Tables 14101 to 14150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-5-difluoromethoxyphenyl Tables 14151 to 14200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-6-difluoromethoxyphenyl Tables 14201 to 14250 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-4-difluoromethoxyphenyl Tables 14251 to 14300 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-5-difluoromethoxyphenyl Tables 14301 to 14350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-3-bromophenyl Tables 14351 to 14400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-4-bromophenyl Tables 14401 to 14450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-5-bromophenyl Tables 14451 to 14500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethoxy-4-bromophenyl Tables 14501 to 14550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-3-trifluoromethoxyphenyl Tables 14551 to 14600 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-4-trifluoromethoxyphenyl Tables 14601 to 14650 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-5-trifluoromethoxyphenyl Tables 14651 to 14700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-bromo-6-trifluoromethoxyphenyl Tables 14701 to 14750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-4-trifluoromethoxyphenyl Tables 14751 to 14800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-bromo-5-trifluoromethoxyphenyl Tables 14801 to 14850 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-3-bromophenyl Tables 14851 to 14900 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-4-bromophenyl Tables 14901 to 14950 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-5-bromophenyl Tables 14951 to 15000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethoxy-4-bromophenyl Tables 15001 to 15050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-3-difluoromethylphenyl Tables 15051 to 15100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-4-difluoromethylphenyl Tables 15101 to 15150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-5-difluoromethylphenyl Tables 15151 to 15200 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-6-difluoromethylphenyl Tables 15201 to 15250 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-4-difluoromethylphenyl Tables 15251 to 15300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-5-difluoromethylphenyl Tables 15301 to 15350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-3-methylphenyl Tables 15351 to 15400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-4-methylphenyl Tables 15401 to 15450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-5-methylphenyl Tables 15451 to 15500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethyl-4-methylphenyl Tables 15501 to 15550 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-3-trifluoromethylphenyl Tables 15551 to 15600 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-4-trifluoromethylphenyl Tables 15601 to 15650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-5-trifluoromethylphenyl Tables 15651 to 15700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-6-trifluoromethylphenyl Tables 15701 to 15750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-4-trifluoromethylphenyl Tables 15751 to 15800 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-5-trifluoromethylphenyl Tables 15801 to 15850 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-3-methylphenyl Tables 15851 to 15900 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-4-methylphenyl

Tables 15901 to 15950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-5-methylphenyl

Tables 15951 to 16000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethyl-4-methylphenyl

Tables 16001 to 16050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-3-methoxyphenyl Tables 16051 to 16100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-4-methoxyphenyl

Tables 16101 to 16150 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-5-methoxyphenyl

Tables 16151 to 16200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-6-methoxyphenyl

Tables 16201 to 16250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-4-methoxyphenyl

Tables 16251 to 16300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-5-methoxyphenyl Tables 16301 to 16350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-3-methylphenyl Tables 16351 to 16400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-4-methylphenyl Tables 16401 to 16450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-5-methylphenyl

Tables 16451 to 16500 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methoxy-4-methylphenyl

Tables 16501 to 16550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-3-difluoromethoxyphenyl

Tables 16551 to 16600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-4-difluoromethoxyphenyl

Tables 16601 to 16650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-5-difluoromethoxyphenyl Tables 16651 to 16700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-6-difluoromethoxyphenyl

Tables 16701 to 16750 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-4-difluoromethoxyphenyl

Tables 16751 to 16800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-5-difluoromethoxyphenyl

Tables 16801 to 16850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-3-methylphenyl Tables 16851 to 16900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-4-methylphenyl Tables 16901 to 16950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-5-methylphenyl Tables 16951 to 17000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethoxy-4-methylphenyl Tables 17001 to 17050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-3-trifluoromethoxyphenyl Tables 17051 to 17100 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-4-trifluoromethoxyphenyl Tables 17101 to 17150 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-5-trifluoromethoxyphenyl Tables 17151 to 17200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methyl-6-trifluoromethoxyphenyl Tables 17201 to 17250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-4-trifluoromethoxyphenyl Tables 17251 to 17300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methyl-5-trifluoromethoxyphenyl Tables 17301 to 17350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-3-methylphenyl Tables 17351 to 17400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-4-methylphenyl Tables 17401 to 17450 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-5-methylphenyl Tables 17451 to 17500 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethoxy-4-methylphenyl Tables 17501 to 17550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-3-trifluoromethylphenyl Tables 17551 to 17600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-4-trifluoromethylphenyl Tables 17601 to 17650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-5-trifluoromethylphenyl Tables 17651 to 17700 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-6-trifluoromethylphenyl Tables 17701 to 17750 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethyl-4-trifluoromethylphenyl Tables 17751 to 17800 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethyl-5-trifluoromethylphenyl Tables 17801 to 17850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-3-difluoromethylphenyl Tables 17851 to 17900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-4-difluoromethylphenyl Tables 17901 to 17950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-5-difluoromethylphenyl Tables 17951 to 18000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethyl-4-difluoromethylphenyl Tables 18001 to 18050 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-3-methoxyphenyl Tables 18051 to 18100 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-4-methoxyphenyl Tables 18101 to 18150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-5-methoxyphenyl Tables 18151 to 18200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-6-methoxyphenyl Tables 18201 to 18250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethyl-4-methoxyphenyl Tables 18251 to 18300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethyl-5-methoxyphenyl Tables 18301 to 18350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-3-difluoromethylphenyl Tables 18351 to 18400 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-4-difluoromethylphenyl Tables 18401 to 18450 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-5-difluoromethylphenyl Tables 18451 to 18500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methoxy-4-difluoromethylphenyl Tables 18501 to 18550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-3-difluoromethoxyphenyl Tables 18551 to 18600

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-4-difluoromethoxyphenyl Tables 18601 to 18650 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-5-difluoromethoxyphenyl Tables 18651 to 18700 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-6-difluoromethoxyphenyl Tables 18701 to 18750 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethyl-4-difluoromethoxyphenyl Tables 18751 to 18800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethyl-5-difluoromethoxyphenyl Tables 18801 to 18850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-3-difluoromethylphenyl Tables 18851 to 18900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-4-difluoromethylphenyl Tables 18901 to 18950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-5-difluoromethylphenyl Tables 18951 to 19000 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethoxy-4-difluoromethylphenyl Tables 19001 to 19050 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-3-trifluoromethoxyphenyl Tables 19051 to 19100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-4-trifluoromethoxyphenyl Tables 19101 to 19150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-5-trifluoromethoxyphenyl Tables 19151 to 19200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethyl-6-trifluoromethoxyphenyl Tables 19201 to 19250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethyl-4-trifluoromethoxyphenyl Tables 19251 to 19300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethyl-5-trifluoromethoxyphenyl Tables 19301 to 19350 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-3-difluoromethylphenyl Tables 19351 to 19400 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-4-difluoromethylphenyl Tables 19401 to 19450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-5-difluoromethylphenyl Tables 19451 to 19500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethoxy-4-difluoromethylphenyl Tables 19501 to 19550

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-3-methoxyphenyl Tables 19551 to 19600 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-4-methoxyphenyl Tables 19601 to 19650 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-5-methoxyphenyl Tables 19651 to 19700 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-6-methoxyphenyl Tables 19701 to 19750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethyl-4-methoxyphenyl Tables 19751 to 19800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethyl-5-methoxyphenyl Tables 19801 to 19850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-3-trifluoromethylphenyl Tables 19851 to 19900

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-4-trifluoromethylphenyl Tables 19901 to 19950 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-5-trifluoromethylphenyl Tables 19951 to 20000 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methoxy-4-trifluoromethylphenyl Tables 20001 to 20050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-3-difluoromethoxyphenyl Tables 20051 to 20100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-4-difluoromethoxyphenyl Tables 20101 to 20150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-5-difluoromethoxyphenyl Tables 20151 to 20200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-6-difluoromethoxyphenyl Tables 20201 to 20250

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethyl-4-difluoromethoxyphenyl Tables 20251 to 20300 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethyl-5-difluoromethoxyphenyl Tables 20301 to 20350 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-3-trifluoromethylphenyl Tables 20351 to 20400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-4-trifluoromethylphenyl Tables 20401 to 20450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-5-trifluoromethylphenyl Tables 20451 to 20500

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethoxy-4-trifluoromethylphenyl Tables 20501 to 20550 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-3-trifluoromethoxyphenyl Tables 20551 to 20600 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-4-trifluoromethoxyphenyl Tables 20601 to 20650 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-5-trifluoromethoxyphenyl Tables 20651 to 20700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethyl-6-trifluoromethoxyphenyl Tables 20701 to 20750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethyl-4-trifluoromethoxyphenyl Tables 20751 to 20800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethyl-5-trifluoromethoxyphenyl Tables 20801 to 20850

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-3-trifluoromethylphenyl Tables 20851 to 20900 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-4-trifluoromethylphenyl Tables 20901 to 20950 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-5-trifluoromethylphenyl Tables 20951 to 21000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethoxy-4-trifluoromethylphenyl Tables 21001 to 21050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-3-difluoromethoxyphenyl Tables 21051 to 21 100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-4-difluoromethoxyphenyl Tables 21 101 to 21 150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-5-difluoromethoxyphenyl Tables 21 151 to 21200

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-6-difluoromethoxyphenyl Tables 21201 to 21250 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methoxy-4-difluoromethoxyphenyl Tables 21251 to 21300 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methoxy-5-difluoromethoxyphenyl Tables 21301 to 21350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-3-methoxyphenyl Tables 21351 to 21400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-4-methoxyphenyl Tables 21401 to 21450

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-5-methoxyphenyl Tables 21451 to 21500 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethoxy-4-methoxyphenyl Tables 21501 to 21550 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-3-trifluoromethoxyphenyl Tables 21551 to 21600 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-4-trifluoromethoxyphenyl Tables 21601 to 21650

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-5-trifluoromethoxyphenyl Tables 21651 to 21700

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-methoxy-6-trifluoromethoxyphenyl Tables 21701 to 21750

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methoxy-4-trifluoromethoxyphenyl Tables 21751 to 21800

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-methoxy-5-trifluoromethoxyphenyl Tables 21801 to 21850 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-3-methoxyphenyl Tables 21851 to 21900 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-4-methoxyphenyl Tables 21901 to 21950

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-5-methoxyphenyl Tables 21951 to 22000

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethoxy-4-methoxyphenyl Tables 22001 to 22050

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-3-trifluoromethoxyphenyl Tables 22051 to 22100

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-4-trifluoromethoxyphenyl Tables 22101 to 22150

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-5-trifluoromethoxyphenyl Tables 22151 to 22200 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-difluoromethoxy-6-trifluoromethoxyphenyl Tables 22201 to 22250 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethoxy-4-trifluoromethoxyphenyl Tables 22251 to 22300

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-difluoromethoxy-5-trifluoromethoxyphenyl Tables 22301 to 22350

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-3-difluoromethoxyphenyl Tables 22351 to 22400

Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-4-difluoromethoxyphenyl Tables 22401 to 22450 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 2-trifluoromethoxy-5-difluoromethoxyphenyl Tables 22451 to 22500 Compounds of the formula I.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A, R ⁵ is as defined in any of tables 1 to 50 and R ³² is 3-trifluoromethoxy-4-difluoromethoxyphenyl Tables 22501 to 44600 Compounds of the formula I.B3 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A and the combination of R ⁵ and R ³² is as defined in any of tables 401 to 22500

Tables 44601 to 66700 Compounds of the formula I.B4 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A and the combination of R ⁵ and R ³² is as defined in any of tables 401 to 22500

Tables 66701 to 67100

Compounds of the formula I.B5 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A and the combination of R ⁵ and R ³¹ is as defined in any of tables 1 to 400

Tables 67101 to 89200

Compounds of the formula I.B6 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A and the combination of R ⁵ and R ³² is as defined in any of tables 401 to 22500

Tables 89201 to 11 1300

Compounds of the formula I.B7 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A and the combination of R ⁵ and R ³² is as defined in any of tables 401 to 22500 Tables 1 1131 to 133400

Compounds of the formula I.B8 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A and the combination of R ⁵ and R ³² is as defined in any of tables 401 to 22500

Table 133401 Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is H

Table 133402

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is methyl

Table 133403

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is ethyl

Table 133404

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is propyl Table 133405

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is isopropyl Table 133406

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is n-butyl

Table 133407 Compounds of the formula II.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is sec-butyl

Table 133408

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is isobutyl

Table 133409

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is tert-butyl

Table 133410

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is phenyl Table 13341 1

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is 4-methylphenyl

Table 133412 Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is benzyl

Table 133413

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is methylcarbonyl

Table 133414 Compounds of the formula II.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is ethylcarbonyl

Table 133415 Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is propylcarbonyl

Table 133416

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is isopropylcarbonyl

Table 133417

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is phenylcarbonyl

Table 133418

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is methoxycarbonyl Table 133419

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is ethoxycarbonyl

Table 133420 Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is propoxycarbonyl

Table 133421

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is isopropoxycarbonyl

Table 133422

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is phenoxycarbonyl

Table 133423

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is methylaminocarbonyl Table 133424

Compounds of the formula II.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is ethylaminocarbonyl Table 133425

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is propylaminocarbonyl

Table 133426 Compounds of the formula II.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is isopropylaminocarbonyl

Table 133427

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is phenylaminocarbonyl

Table 133428

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is methylsulfonyl

Table 133429

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is ethylsulfonyl Table 133430

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is propylsulfonyl

Table 133431 Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is isopropylsulfonyl

Table 133432

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is phenylsulfonyl

Table 133433 Compounds of the formula II.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is methoxysulfonyl Table 133434 Compounds of the formula II.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is ethoxysulfonyl Table 133435 Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is propoxysulfonyl Table 133436

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is isopropoxysulfonyl Table 133437

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is phenoxysulfonyl Table 133438

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³¹ is methyl and R ^5a is CN Tables 133439 to 133476 Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is as defined in any of tables 133401 to 133438 and R ³¹ is ethyl Tables 133477 to 133514 Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is as defined in any of tables 133401 to 133438 and R ³¹ is propyl Tables 133515 to 133552

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is as de- fined in any of tables 133401 to 133438 and R ³¹ is isopropyl Tables 133553 to 133590

Compounds of the formula II. B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is as defined in any of tables 133401 to 133438 and R ³¹ is n-butyl Tables 133591 to 133628

Compounds ofthe formula II.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row ofTable A above, R ^5a is as defined in any oftables 133401 to 133438 and R ³¹ is sec-butyl Tables 133629 to 133666

Compounds ofthe formula II.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row ofTable A above, R ^5a is as defined in any of tables 133401 to 133438 and R ³¹ is isobutyl Tables 133667 to 133704 Compounds ofthe formula II.B1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row ofTable A above, R ^5a is as defined in any of tables 133401 to 133438 and R ³¹ is tert-butyl

Tables 133705 to 150500 Compounds ofthe formula II.B2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row ofTable A above, R ^5a is as defined in any of tables 133401 to 133438 and R ³² is as defined in any of tables 401, 451, 501,551,601,651,701,751,801,851,901,951, 1001, 1051, 1101, 1151, 1201, 1251, 1301, 1351, 1401, 1451, 1501, 1551, 1601, 1651, 1701, 1751, 1801, 1851, 1901, 1951, 2001 , 2051,2101, 2151, 2201 , 2251 , 2301, 2351 , 2401, 2451 , 2501 , 2551, 2601 , 2651, 2701 , 2751, 2801 , 2851, 2901 , 2951 , 3001, 3051 , 3101, 3151 , 3201 , 3251, 3301 , 3351, 3401 , 3451 , 3501, 3551 , 3601 , 3651 , 3701 , 3751, 3801 , 3851 , 3901, 3951 , 4001 , 4051 , 4101 , 4151 , 4201, 4251 , 4301 , 4351 , 4401 , 4451, 4501 , 4551 , 4601, 4651 , 4701 , 4751 , 4801 , 4851 , 4901, 4951 , 5001 , 5051 , 5101 , 5151, 5201 , 5251 , 5301, 5351 , 5401 , 5451 , 5501, 5551, 5601, 5651, 5701, 5751, 5801, 5851, 5901, 5951, 6001, 6051, 6101, 6151, 6201 , 6251 , 6301, 6351 , 6401 , 6451 , 6501 , 6551, 6601 , 6651 , 6701, 6751 , 6801 , 6851 , 6901, 6951, 7001, 7051, 7101, 7151, 7201, 7251, 7301, 7351, 7401, 7451, 7501, 7551, 7601, 7651, 7701, 7751, 7801, 7851, 7901, 7951, 8001, 8051, 8101, 8151, 8201, 8251, 8301 , 8351 , 8401, 8451 , 8501 , 8551 , 8601 , 8651, 8701 , 8751 , 8801, 8851 , 8901 , 8951 , 9001, 9051, 9101, 9151, 9201, 9251, 9301, 9351, 9401, 9451, 9501, 9551, 9601, 9651, 9701, 9751, 9801, 9851, 9901, 9951, 10001, 10051, 10101, 10151, 10201, 10251, 10301, 10351, 10401, 10451, 10501, 10551, 10601, 10651, 10701, 10751, 10801, 10851, 10901, 10951, 11001, 11051, 11101, 11151, 11201, 11251, 11301, 11351, 11401, 11451, 11501, 11551, 11601, 11651, 11701, 11751, 11801, 11851, 11901, 11951, 12001, 12051, 12101, 12151, 12201, 12251, 12301, 12351, 12401, 12451, 12501, 12551, 12601, 12651, 12701, 12751, 12801, 12851, 12901, 12951, 13001, 13051, 13101, 13151, 13201, 13251, 13301, 13351, 13401, 13451, 13501, 13551, 13601, 13651, 13701, 13751, 13801, 13851, 13901, 13951, 14001, 14051, 14101, 14151, 14201, 14251, 14301, 14351, 14401, 14451, 14501, 14551, 14601, 14651, 14701, 14751, 14801, 14851, 14901, 14951, 15001, 15051, 15101, 15151, 15201, 15251, 15301, 15351, 15401, 15451, 15501, 15551, 15601, 15651, 15701, 15751, 15801, 15851, 15901, 15951, 16001, 16051, 16101, 16151, 16201, 16251, 16301, 16351, 16401, 16451, 16501, 16551, 16601, 16651, 16701, 16751, 16801, 16851, 16901, 16951, 17001, 17051, 17101, 17151, 17201, 17251, 17301, 17351, 17401, 17451, 17501, 17551, 17601, 17651, 17701, 17751, 17801, 17851, 17901, 17951, 18001, 18051, 18101, 18151, 18201, 18251, 18301, 18351, 18401, 18451, 18501, 18551, 18601, 18651, 18701, 18751, 18801, 18851, 18901, 18951, 19001, 19051, 19101, 19151, 19201, 19251, 19301, 19351, 19401, 19451, 19501, 19551, 19601, 19651,19701,19751,19801,19851,19901,19951,20001,20051,20101, 20151, 20201 , 20251 , 20301 , 20351 , 20401 , 20451 , 20501 , 20551 , 20601 , 20651 , 20701 , 20751 , 20801 , 20851 , 20901 , 20951 , 21001 , 21051 , 21101 , 21151 , 21201 , 21251 , 21301,21351,21401,21451,21501,21551,21601,21651,21701,21751, 21801, 21851 , 21901 , 21951 , 22001 , 22051 , 22101 , 22151 , 22201 , 22251 , 22301 , 22351 , 22401 and 22451

Tables 150501 to 167296

Compounds ofthe formula II.B3 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row ofTable A above, R ^5a is as de- fined in any of tables 133401 to 133438 and R ³² is as defined in any oftables 401, 451, 501,551,601,651,701,751,801,851,901,951, 1001, 1051, 1101, 1151, 1201, 1251, 1301, 1351, 1401, 1451, 1501, 1551, 1601, 1651, 1701, 1751, 1801, 1851, 1901, 1951, 2001 , 2051 , 2101, 2151 , 2201 , 2251 , 2301 , 2351, 2401 , 2451 , 2501, 2551 , 2601 , 2651 , 2701 , 2751 , 2801, 2851 , 2901 , 2951 , 3001 , 3051, 3101 , 3151 , 3201, 3251 , 3301 , 3351 , 3401 , 3451, 3501 , 3551, 3601 , 3651 , 3701, 3751 , 3801, 3851 , 3901 , 3951, 4001 , 4051, 4101 , 4151 , 4201, 4251 , 4301 , 4351 , 4401 , 4451, 4501 , 4551 , 4601, 4651 , 4701 , 4751 , 4801 , 4851 , 4901, 4951 , 5001 , 5051 , 5101 , 5151, 5201 , 5251 , 5301, 5351 , 5401 , 5451 , 5501, 5551, 5601, 5651, 5701, 5751, 5801, 5851, 5901, 5951, 6001, 6051, 6101, 6151, 6201 , 6251 , 6301, 6351 , 6401 , 6451 , 6501 , 6551, 6601 , 6651 , 6701, 6751 , 6801 , 6851 , 6901, 6951, 7001, 7051, 7101, 7151, 7201, 7251, 7301, 7351, 7401, 7451, 7501, 7551, 7601, 7651, 7701, 7751, 7801, 7851, 7901, 7951, 8001, 8051, 8101, 8151, 8201, 8251, 8301 , 8351 , 8401, 8451 , 8501 , 8551 , 8601 , 8651, 8701 , 8751 , 8801, 8851 , 8901 , 8951 , 9001, 9051, 9101, 9151, 9201, 9251, 9301, 9351, 9401, 9451, 9501, 9551, 9601, 9651, 9701, 9751, 9801, 9851, 9901, 9951, 10001, 10051, 10101, 10151, 10201, 10251, 10301, 10351, 10401, 10451, 10501, 10551, 10601, 10651, 10701, 10751, 10801, 10851, 10901, 10951, 11001, 11051, 11101, 11151, 11201, 11251, 11301, 11351, 11401, 11451, 11501, 11551, 11601, 11651, 11701, 11751, 11801, 11851, 11901, 11951, 12001, 12051, 12101, 12151, 12201, 12251, 12301, 12351, 12401, 12451, 12501, 12551, 12601, 12651, 12701, 12751, 12801, 12851, 12901, 12951, 13001, 13051, 13101, 13151, 13201, 13251, 13301, 13351, 13401, 13451, 13501, 13551, 13601, 13651, 13701, 13751, 13801, 13851, 13901, 13951, 14001, 14051, 14101, 14151, 14201, 14251, 14301, 14351, 14401, 14451, 14501, 14551, 14601, 14651, 14701, 14751, 14801, 14851, 14901, 14951, 15001, 15051, 15101, 15151, 15201, 15251, 15301, 15351, 15401, 15451, 15501, 15551, 15601, 15651, 15701, 15751, 15801, 15851, 15901, 15951, 16001, 16051, 16101, 16151, 16201, 16251, 16301, 16351, 16401, 16451, 16501, 16551, 16601, 16651, 16701, 16751, 16801, 16851, 16901, 16951, 17001, 17051, 17101, 17151, 17201, 17251, 17301, 17351, 17401, 17451, 17501, 17551, 17601, 17651, 17701, 17751, 17801, 17851, 17901, 17951, 18001, 18051, 18101, 18151, 18201, 18251, 18301, 18351, 18401, 18451, 18501, 18551, 18601, 18651, 18701, 18751, 18801, 18851, 18901, 18951, 19001, 19051, 19101, 19151, 19201, 19251, 19301, 19351, 19401, 19451, 19501, 19551, 19601, 19651,19701,19751,19801,19851,19901,19951,20001,20051,20101, 20151, 20201 , 20251 , 20301 , 20351 , 20401 , 20451 , 20501 , 20551 , 20601 , 20651 , 20701 , 20751,20801,20851,20901,20951,21001,21051,21101,21151,21201, 21251, 21301,21351,21401,21451,21501,21551,21601,21651,21701,21751, 21801, 21851 , 21901 , 21951 , 22001 , 22051 , 22101 , 22151 , 22201 , 22251 , 22301 , 22351 , 22401 and 22451

Tables 167297 to 184092

Compounds of the formula II. B4 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is as defined in any of tables 133401 to 133438 and R ³² is as defined in any of tables 401, 451, 501, 551, 601, 651, 701, 751, 801, 851, 901, 951, 1001, 1051, 1101, 1151, 1201, 1251, 1301, 1351, 1401, 1451, 1501, 1551, 1601, 1651, 1701, 1751, 1801, 1851, 1901, 1951, 2001 , 2051 , 2101 , 2151 , 2201 , 2251 , 2301 , 2351 , 2401 , 2451 , 2501 , 2551 , 2601 , 2651 , 2701 , 2751 , 2801 , 2851 , 2901 , 2951 , 3001 , 3051 , 3101 , 3151 , 3201 , 3251 , 3301 , 3351 , 3401 , 3451 , 3501 , 3551 , 3601 , 3651 , 3701 , 3751 , 3801 , 3851 , 3901 , 3951 , 4001 , 4051 , 4101 , 4151 , 4201 , 4251 , 4301 , 4351 , 4401 , 4451 , 4501 , 4551 , 4601 , 4651 , 4701 , 4751 , 4801 , 4851 , 4901 , 4951 , 5001 , 5051 , 5101 , 5151 , 5201 , 5251 , 5301 , 5351 , 5401 , 5451 , 5501, 5551, 5601, 5651, 5701, 5751, 5801, 5851, 5901, 5951, 6001, 6051, 6101, 6151, 6201 , 6251 , 6301 , 6351 , 6401 , 6451 , 6501 , 6551 , 6601 , 6651 , 6701 , 6751 , 6801 , 6851 , 6901, 6951, 7001, 7051, 7101, 7151, 7201, 7251, 7301, 7351, 7401, 7451, 7501, 7551, 7601, 7651, 7701, 7751, 7801, 7851, 7901, 7951, 8001, 8051, 8101, 8151, 8201, 8251, 8301 , 8351 , 8401 , 8451 , 8501 , 8551 , 8601 , 8651 , 8701 , 8751 , 8801 , 8851 , 8901 , 8951 , 9001, 9051, 9101, 9151, 9201, 9251, 9301, 9351, 9401, 9451, 9501, 9551, 9601, 9651, 9701, 9751, 9801, 9851, 9901, 9951, 10001, 10051, 10101, 10151, 10201, 10251, 10301, 10351, 10401, 10451, 10501, 10551, 10601, 10651, 10701, 10751, 10801, 10851, 10901, 10951, 11001, 11051, 11101, 11151, 11201, 11251, 11301, 11351, 11401, 11451, 11501, 11551, 11601, 11651, 11701, 11751, 11801, 11851, 11901, 11951, 12001, 12051, 12101, 12151, 12201, 12251, 12301, 12351, 12401, 12451, 12501, 12551, 12601, 12651, 12701, 12751, 12801, 12851, 12901, 12951, 13001, 13051, 13101, 13151, 13201, 13251, 13301, 13351, 13401, 13451, 13501, 13551, 13601, 13651, 13701, 13751, 13801, 13851, 13901, 13951, 14001, 14051, 14101, 14151, 14201, 14251, 14301, 14351, 14401, 14451, 14501, 14551, 14601, 14651, 14701, 14751, 14801, 14851, 14901, 14951, 15001, 15051, 15101, 15151, 15201, 15251, 15301, 15351, 15401, 15451, 15501, 15551, 15601, 15651, 15701, 15751, 15801, 15851, 15901, 15951, 16001, 16051, 16101, 16151, 16201, 16251, 16301, 16351, 16401, 16451, 16501, 16551, 16601, 16651, 16701, 16751, 16801, 16851, 16901, 16951, 17001, 17051, 17101, 17151, 17201, 17251, 17301, 17351, 17401, 17451, 17501, 17551, 17601, 17651, 17701, 17751, 17801, 17851, 17901, 17951, 18001, 18051, 18101, 18151, 18201, 18251, 18301, 18351, 18401, 18451, 18501, 18551, 18601, 18651, 18701, 18751, 18801, 18851, 18901, 18951, 19001, 19051, 19101, 19151, 19201, 19251, 19301, 19351, 19401, 19451, 19501, 19551, 19601, 19651, 19701, 19751, 19801, 19851, 19901, 19951,20001,20051,20101,20151, 20201 , 20251 , 20301 , 20351 , 20401 , 20451 , 20501 , 20551 , 20601 , 20651 , 20701 , 20751 , 20801 , 20851 , 20901 , 20951 , 21001 , 21051 , 21101 , 21151 , 21201 , 21251 , 21301, 21351, 21401, 21451, 21501, 21551, 21601, 21651, 21701, 21751, 21801, 21851 , 21901 , 21951 , 22001 , 22051 , 22101 , 22151 , 22201 , 22251 , 22301 , 22351 , 22401 and 22451

In the above tables 401 to 22500, the given positions of the substituents on the phenyl ring are to be understood as relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

In another preferred embodiment of the invention (embodiment C), R ¹ is a group of formula V, where

R ² is aryl which may carry 1 , 2, 3, 4 or 5 substituents R ⁷ , or is a 5- or 6-membered heteroaromatic ring containing 1 , 2 or 3 heteroatoms selected from N, O and S as ring members, where the heteroaromatic ring may carry 1 , 2, 3 or 4 substituents R ⁸ ;

R ³ is selected from Ci-Cio-alkyl which may carry 1 or 2 substituents R ⁹ , C1-C10- haloalkyl which may carry 1 or 2 substituents R ⁹ , Cs-Cs-cycloalkyl, C3-C8- cycloalkyl-d^-alkyl, where the cycloalkyl moiety in the 2 last-mentioned radicals may carry 1, 2, 3 or 4 substituents R ¹⁰ , aryl and aryl-Ci-C4-alkyl, where the aryl moiety in the 2 last-mentioned radicals may carry 1 , 2, 3, 4 or 5 substituents

R ⁴ is hydrogen; and R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings; except for compounds wherein R ² is 2,4-dichlorophenyl, R ³ is methyl, ethyl, propyl, isopropyl, n-butyl, sec-butyl, isobutyl, tert-butyl, 2,2,2-trifluoroethyl, pentafluoroethyl, trifluoromethoxymethyl, 1 ,1-difluoroethoxymethyl, 1 ,1 ,2,2-tetrafluoroethoxymethyl, cyclopropyl, 1-chlorocyclopropyl, 1-fluorocyclopropyl, 1-cyclopropylethyl, cyclopentyl, cyclohexyl, cyclohexylmethyl, 4-fluorophenyl, 4-chlorophenyl, 4-fluorophenylmethyl or 4-chlorophenylmethyl and R ⁴ is H; . except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl, 4-chlorophenyl, 2,4,6-trichlorophenyl, 4-methylphenyl, 4-trifluoromethylphenyl or 2- trifluoromethoxyphenyl, R ³ is n-propyl and R ⁴ is H; and except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl or 4-chlorophenyl, R ³ is 1 ,1 ,2,2-tetrafluoroethoxymethyl and R ⁴ is H.

In the above definitions, aryl is preferably phenyl.

More preferabyl (embodiment C.1 ), R ¹ is a group of formula V, where

R ² is phenyl which may carry 1 , 2 or 3 substituents R ⁷ ;

R ³ is selected from Ci-Cio-alkyl which may carry 1 or 2 substituents R ⁹ , C1-C4- haloalkyl, C ₃ -C8-cycloalkyl and C3-C8-cycloalkyl-Ci-C4-alkyl, where the cycloalkyl moiety in the 2 last-mentioned radicals may carry 1 , 2, 3 or 4 substituents R ¹⁰ ; R ⁴ is hydrogen; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH3, CHF2, CF3, OCH ₃ , OCHF ₂ and OCF ₃ ; each R ⁹ is independently selected from Ci-C4-alkoxy and Ci-C4-fluoroalkoxy; each R ¹⁰ is independently selected from halogen, Ci-C4-alkyl and Ci-C4-haloalkyl; and R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings; except for compounds wherein R ² is 2,4-dichlorophenyl, R ³ is methyl, ethyl, propyl, isopropyl, n-butyl, sec-butyl, isobutyl, tert-butyl, 2,2,2-trifluoroethyl, pentafluoroethyl, trifluoromethoxymethyl, 1 ,1-difluoroethoxymethyl, 1 ,1 ,2,2-tetrafluoroethoxymethyl, cyclopropyl, 1-chlorocyclopropyl, 1-fluorocyclopropyl, 1-cyclopropylethyl, cyclopentyl, cyclohexyl, cyclohexylmethyl, 4-fluorophenyl, 4-chlorophenyl, 4-fluorophenylmethyl or 4-chlorophenylmethyl and R ⁴ is H; . except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl, 4-chlorophenyl, 2,4,6-trichlorophenyl, 4-methylphenyl, 4-trifluoromethylphenyl or 2- trifluoromethoxyphenyl, R ³ is n-propyl and R ⁴ is H; and except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl or 4-chlorophenyl, R ³ is 1 ,1 ,2,2-tetrafluoroethoxymethyl and R ⁴ is H.

Even more preferably (embodiment C.1.1), R ¹ is a group of formula V, where R ² is phenyl which may carry 1 , 2 or 3 substituents R ⁷ ;

R ³ is selected from Ci-Cβ-alkyl, d-Cε-alkyl which carries 1 substituent R ⁹ , cyclopro- pyl and cyclopropyl-Ci-C2-alkyl, where the cyclopropyl moiety in the 2 last- mentioned radicals may carry 1 or 2 substituents R ¹⁰ ; R ⁴ is hydrogen; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH3, CHF2, CF3, OCH ₃ , OCHF ₂ and OCF ₃ ; R ⁹ is Ci-C4-fluoroalkoxy; each R ¹⁰ is independently selected from halogen and Ci-C4-alkyl; and R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings; except for compounds wherein R ² is 2,4-dichlorophenyl, R ³ is methyl, ethyl, propyl, isopropyl, n-butyl, sec-butyl, isobutyl, tert-butyl, 2,2,2-trifluoroethyl, pentafluoroethyl, trifluoromethoxymethyl, 1 ,1-difluoroethoxymethyl, 1 ,1 ,2,2-tetrafluoroethoxymethyl, cyclopropyl, 1-chlorocyclopropyl, 1-fluorocyclopropyl, 1-cyclopropylethyl, cyclopentyl, cyclohexyl, cyclohexylmethyl, 4-fluorophenyl, 4-chlorophenyl, 4-fluorophenylmethyl or 4-chlorophenylmethyl and R ⁴ is H; . except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl, 4-chlorophenyl, 2,4,6-trichlorophenyl, 4-methylphenyl, 4-trifluoromethylphenyl or 2- trifluoromethoxyphenyl, R ³ is n-propyl and R ⁴ is H; and except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl or 4-chlorophenyl, R ³ is 1 ,1 ,2,2-tetrafluoroethoxymethyl and R ⁴ is H.

Particularly preferably (embodiment C.1.1.1 ), R ¹ is a group of formula V, where R ² is phenyl which may carry 1 , 2 or 3 substituents R ⁷ ;

R ³ is selected from Ci-C4-alkyl, Ci-C2-alkyl which carries 1 substituent R ⁹ , cyclopropyl and cyclopropyl-Ci-C2-alkyl, where the cyclopropyl moiety in the 2 last- mentioned radicals may carry 1 or 2 substituents R ¹⁰ ;

R ⁴ is hydrogen; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH ₃ , CHF2, CF ₃ , OCH ₃ , OCHF ₂ and OCF ₃ ;

R ⁹ is Ci-C2-fluoroalkoxy; each R ¹⁰ is independently selected from halogen and Ci-C4-alkyl; and R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings; except for compounds wherein R ² is 2,4-dichlorophenyl, R ³ is methyl, ethyl, propyl, isopropyl, n-butyl, sec-butyl, isobutyl, tert-butyl, 2,2,2-trifluoroethyl, pentafluoroethyl, trifluoromethoxymethyl, 1 ,1-difluoroethoxymethyl, 1 ,1 ,2,2-tetrafluoroethoxymethyl, cyclopropyl, 1-chlorocyclopropyl, 1-fluorocyclopropyl, 1-cyclopropylethyl, cyclopentyl, cyclohexyl, cyclohexylmethyl, 4-fluorophenyl, 4-chlorophenyl, 4-fluorophenylmethyl or 4-chlorophenylmethyl and R ⁴ is H; . except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl, 4-chlorophenyl, 2,4,6-trichlorophenyl, 4-methylphenyl, 4-trifluoromethylphenyl or 2- trifluoromethoxyphenyl, R ³ is n-propyl and R ⁴ is H; and except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl or 4-chlorophenyl, R ³ is 1 ,1 ,2,2-tetrafluoroethoxymethyl and R ⁴ is H.

Specifically (embodiment C.1.1.1.1 ), R ¹ is a group of formula V, where

R ² is phenyl which may carry 1 , 2 or 3 substituents R ⁷ ;

R ³ is selected from Ci-C4-alkyl, methyl which carries 1 substituent R ⁹ , cyclopropyl and cyclopropyl-Ci-C2-alkyl, where the cyclopropyl moiety in the 2 last-mentioned radicals may carry 1 or 2 substituents R ¹⁰ ; R ⁴ is hydrogen; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH3, CHF2, CF3, OCH ₃ , OCHF ₂ and OCF ₃ ;

R ⁹ is selected from OCF ₃ , OCF ₂ CH ₃ , OCF ₂ CHF ₂ and OCF ₂ CF ₃ ; each R ¹⁰ is independently selected from halogen and Ci-C4-alkyl; and

R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings; except for compounds wherein R ² is 2,4-dichlorophenyl, R ³ is methyl, ethyl, propyl, isopropyl, n-butyl, sec-butyl, isobutyl, tert-butyl, 2,2,2-trifluoroethyl, pentafluoroethyl, trifluoromethoxymethyl, 1 ,1-difluoroethoxymethyl, 1 ,1 ,2,2-tetrafluoroethoxymethyl, cyclopropyl, 1-chlorocyclopropyl, 1-fluorocyclopropyl, 1-cyclopropylethyl, cyclopentyl, cyclohexyl, cyclohexylmethyl, 4-fluorophenyl, 4-chlorophenyl, 4-fluorophenylmethyl or

4-chlorophenylmethyl and R ⁴ is H; . except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl, 4-chlorophenyl, 2,4,6-trichlorophenyl, 4-methylphenyl, 4-trifluoromethylphenyl or 2- trifluoromethoxyphenyl, R ³ is n-propyl and R ⁴ is H; and except for compounds wherein R ² is 4-fluorophenyl, 2-chlorophenyl or 4-chlorophenyl,

R ³ is 1 ,1 ,2,2-tetrafluoroethoxymethyl and R ⁴ is H. If R ² is phenyl which carries 1 substituent R ⁷ , this is preferably bound in 2- or 4- position, more preferably in 2-position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

If R ³ is phenyl which carries 1 substituent R ¹¹ , this is preferably bound in 2- or 4- position, more preferably in 2-position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule. If R ³ is phenyl-Ci-C4-alkyl, where the phenyl moiety carries 1 substituent R ¹¹ , this is preferably bound in 2- or 4-position, more preferably in 2-position, relative to the 1 -position of the attachment point of the phenyl ring to the Ci-C4-alkyl group.

If R ² is phenyl which carries 2 substituents R ⁷ , these are preferably bound in 2,4- position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

If R ³ is phenyl which carries 2 substituents R ¹¹ , these are preferably bound in 2,4- position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule. If R ³ is phenyl-Ci-C4-alkyl, where the phenyl moiety carries 2 substituents R ¹¹ , these are preferably bound in 2,4-position, relative to the 1-position of the attachment point of the phenyl ring to the Ci-C4-alkyl group.

Examples for preferred compounds I and Il of embodiment C are compounds of formulae I.C1 , I.C2 and II.C1 , where the variables R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ are hydrogen or have one of the general or, in particular, one of the preferred meanings given above for R ⁷ , where the variables R ⁵ and R ^5a have one of the general or, in particular, one of the preferred meanings given above, where the variable R ³ has one of the preferred meanings given above for R ³ in context with embodiment C. Examples of preferred compounds are the individual compounds compiled in the tables 1 to 1068 below. More- over, the meanings mentioned below for the individual variables in the tables are per se, independently of the combination in which they are mentioned, a particularly preferred embodiment of the substituents in question.

Table 1

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ⁵ is H and R ³ is methyl

Table 2

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ⁵ is H and R ³ is ethyl

Table 3

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ⁵ is H and R ³ is propyl Table 4

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ⁵ is H and R ³ is isopropyl

Table 5 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ⁵ is H and R ³ is n-butyl

Table 6

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ⁵ is H and R ³ is sec-butyl

Table 7

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ⁵ is H and R ³ is isobutyl Table 8

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ⁵ is H and R ³ is tert-butyl Table 9

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ⁵ is H and R ³ is cyclopropyl Table 10

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ⁵ is H and R ³ is i-chlorocyclopropyl Table 11

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ⁵ is H and R ³ is 1-cyclopropylethyl Table 12 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ⁵ is H and R ³ is CH ₂ -O-CF ₂ CHF ₂ Tables 13 to 24 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is methyl Tables 25 to 36

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 1 to 12 and R ⁵ is ethyl Tables 37 to 48

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is propyl Tables 49 to 60

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is isopropyl Tables 61 to 72

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is n-butyl Tables 73 to 84

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is sec-butyl Tables 85 to 96 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is isobutyl Tables 97 to 108 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is tert-butyl Tables 109 to 120

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 1 to 12 and R ⁵ is phenyl Tables 121 to 132

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is 4-methylphenyl Tables 133 to 144

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is benzyl Tables 145 to 156 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is Li ⁺ Tables 157 to 168 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is Na ⁺ Tables 169 to 180 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is K ⁺ Tables 181 to 192

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is YiMg ²⁺ Tables 193 to 204

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 1 to 12 and R ⁵ is Y ₂ Cu ²⁺ Tables 205 to 216

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is YzZn ²⁺ Tables 229 to 240

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is YiFe ²⁺ Tables 217 to 228 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is VzNi ²⁺ Tables 241 to 252 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is NH(CH ₃ )S ⁺ Tables 253 to 264

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 1 to 12 and R ⁵ is NH(C ₂ H ₅ )S ⁺ Tables 265 to 276

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is NH(CH ₂ CH ₂ CH ₂ )S ⁺ Tables 277 to 288

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is NH(CH(CH ₃ ) ₂ )s ⁺ Tables 289 to 300 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is NH(CH ₂ CH ₂ CH ₂ CH ₂ )S ⁺ Tables 301 to 312 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is methylcarbonyl Tables 313 to 324 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is ethylcarbonyl Tables 325 to 336

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 1 to 12 and R ⁵ is propylcarbonyl Tables 337 to 348

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is isopropylcarbonyl Tables 349 to 360

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is methoxycarbonyl Tables 361 to 372 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is ethoxycarbonyl Tables 373 to 384 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is propoxycarbonyl Tables 385 to 396

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 1 to 12 and R ⁵ is isopropoxycarbonyl Tables 397 to 408

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is phenoxycarbonyl Tables 409 to 420

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is methylaminocarbonyl Tables 421 to 432

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is ethylaminocarbonyl Tables 433 to 444 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is propylaminocarbonyl Tables 445 to 456 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is isopropylaminocarbonyl Tables 457 to 468

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 1 to 12 and R ⁵ is phenylaminocarbonyl Tables 469 to 480

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is methylsulfonyl Tables 481 to 492

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is ethylsulfonyl Tables 493 to 504 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is propylsulfonyl Tables 505 to 516 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is isopropylsulfonyl Tables 517 to 528 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is phenylsulfonyl Tables 529 to 540 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is methoxysulfonyl Tables 541 to 552 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is ethoxysulfonyl Tables 553 to 564

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 1 to 12 and R ⁵ is propoxysulfonyl Tables 565 to 576

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is isopropoxysulfonyl Tables 577 to 588

Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is phenoxysulfonyl Tables 589 to 600 Compounds of the formula I.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 1 to 12 and R ⁵ is CN Tables 601 to 612 Compounds of the formula I.C2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ³ is as defined in any of tables 1 to 12 Table 613

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is H and R ³ is methyl Table 614

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is H and R ³ is ethyl Table 615

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is H and

R ³ is propyl Table 616

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is H and

R ³ is isopropyl

Table 617 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is H and

R ³ is n-butyl

Table 618

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is H and

R ³ is sec-butyl

Table 619

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is H and R ³ is isobutyl

Table 620

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is H and

R ³ is tert-butyl Table 621

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is H and

R ³ is cyclopropyl

Table 622 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is H and

R ³ is i-chlorocyclopropyl

Table 623

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is H and

R ³ is 1-cyclopropylethyl

Table 624

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ^5a is H and R ³ is CH ₂ -O-CF ₂ CH F ₂ Tables 625 to 636

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is methyl Tables 637 to 648

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 613 to 624 and R ^5a is ethyl Tables 649 to 660

Compounds of the formula II.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is propyl Tables 661 to 672

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is isopropyl Tables 673 to 684 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is n-butyl Tables 685 to 696 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is sec-butyl Tables 697 to 708

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 613 to 624 and R ^5a is isobutyl Tables 709 to 720

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is tert-butyl Tables 721 to 732

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is phenyl Tables 733 to 744

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is 4-methylphenyl Tables 745 to 756

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is benzyl Tables 757 to 768 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is methylcarbonyl Tables 769 to 780 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is ethylcarbonyl Tables 781 to 792

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 613 to 624 and R ^5a is propylcarbonyl Tables 793 to 804

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is isopropylcarbonyl Tables 805 to 816

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is phenylcarbonyl Tables 817 to 828 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is methoxycarbonyl Tables 829 to 840 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is ethoxycarbonyl Tables 841 to 852 Compounds of the formula II. C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is propoxycarbonyl Tables 853 to 864 Compounds of the formula II.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is isopropoxycarbonyl Tables 865 to 876 Compounds of the formula II.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is phenoxycarbonyl Tables 877 to 888

Compounds of the formula II.C1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 613 to 624 and R ^5a is methylaminocarbonyl Tables 889 to 900

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is ethylaminocarbonyl Tables 901 to 912

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is propylaminocarbonyl Tables 913 to 924 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is isopropylaminocarbonyl Tables 925 to 936 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is phenylaminocarbonyl Tables 937 to 948

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 613 to 624 and R ^5a is methylsulfonyl Tables 949 to 960

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is ethylsulfonyl Tables 961 to 972

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is propylsulfonyl Tables 973 to 984

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is isopropylsulfonyl Tables 985 to 996 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is phenylsulfonyl Tables 997 to 1008 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is methoxysulfonyl Tables 1009 to 1020

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as de- fined in any of tables 613 to 624 and R ^5a is ethoxysulfonyl Tables 1021 to 1032

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is propoxysulfonyl Tables 1033 to 1044

Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is isopropoxysulfonyl Tables 1045 to 1056 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is phenoxysulfonyl Tables 1057 to 1068 Compounds of the formula 11.01 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above, R ³ is as defined in any of tables 613 to 624 and R ^5a is CN In another preferred embodiment of the invention (embodiment D), R ¹ is a group of formula V, where

R ² is phenyl which may carry 1 , 2, 3, 4 or 5 substituents R ⁷ ; R ³ is selected from Ci-Cio-alkyl which may carry 1 substituent R ⁹ ; R ⁴ is OH;

R ⁹ is Si(R ²⁰ ) ₃ ; and

R ⁵ /R ^5a , R ²⁰ and m have one of the above given general or, preferably, one of the above-given preferred meanings; except for compounds wherein R ² is 2,4-dichlorophenyl, R ³ is n-Butyl, R ⁴ is OH and R ⁵ is H, methyl or CN, preferably except for compounds wherein R ² is 2,4-dichlorophenyl, R ³ is n-Butyl and R ⁴ is OH.

In a more preferred embodiment of the invention (embodiment D.1 ), R ¹ is a group of formula V, where R ² is phenyl which may carry 1 , 2 or 3 substituents R ⁷ ; R ³ is d-Cβ-alkyl; R ⁴ is OH; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH3, CHF2, CF3, OCH ₃ , OCHF ₂ and OCF ₃ ; and

R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings; except for compounds wherein R ² is 2,4-dichlorophenyl, R ³ is n-Butyl, R ⁴ is OH and R ⁵ is H, methyl or CN, preferably except for compounds wherein R ² is 2,4-dichlorophenyl, R ³ is n-Butyl and R ⁴ is OH.

Even more preferably (embodiment D.1.1 ), R ¹ is a group of formula V, where

R ² is phenyl which may carry 1 , 2 or 3 substituents R ⁷ ;

R ³ is Ci-C4-alkyl, specifically n-butyl; R ⁴ is OH; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH ₃ , CHF2, CF ₃ , OCH ₃ , OCHF ₂ and OCF ₃ ; and

R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings; except for compounds wherein R ² is 2,4-dichlorophenyl, R ³ is n-Butyl, R ⁴ is OH and R ⁵ is H, methyl or CN, preferably except for compounds wherein R ² is 2,4-dichlorophenyl,

R ³ is n-Butyl and R ⁴ is OH. In an alternatively more preferred embodiment of the invention (embodiment D.2), R ¹ is a group of formula V, where

R ² is phenyl which may carry 1 , 2 or 3 substituents R ⁷ ; R ³ is Ci-C2-alkyl which carries 1 substituent R ⁹ ; R ⁴ is OH; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH3, CHF2, CF3,

OCH ₃ , OCHF ₂ and OCF ₃ ; R ⁹ is Si(R ²⁰ ) ₃ ; and R ⁵ /R ^5a , R ²⁰ and m have one of the above given general or, preferably, one of the above-given preferred meanings.

Even more preferably (embodiment D.2.1 ), R ¹ is a group of formula V, where

R ² is phenyl which may carry 1 , 2 or 3 substituents R ⁷ ; R ³ is CH ₂ -Si(R ²⁰ ) ₃ ;

R ⁴ is OH; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C4-haloalkoxy, and preferably from F, Cl, Br, CH ₃ , CHF ₂ , CF ₃ , OCH ₃ , OCHF ₂ and OCF ₃ ; R ²⁰ is Ci-C ₄ -alkyl, preferably methyl; and

R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings.

If R ² is phenyl which carries 1 substituent R ⁷ , this is preferably bound in 2- or 4- position, more preferably in 2-position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

If R ² is phenyl which carries 2 substituents R ⁷ , these are preferably bound in 2,4- position, relative to the 1 -position of the attachment point of the phenyl ring to the re- mainder of the molecule.

Examples for preferred compounds I and Il of embodiment D are compounds of formulae I.D1 to I.D4, II.D1 and II. D2, where the variables R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ are hy- drogen or have one of the general or, in particular, one of the preferred meanings given above for R ⁷ , and where the variables R ⁵ and R ^5a have one of the general or, in particular, one of the preferred meanings given above. Examples of preferred compounds are the individual compounds compiled in the tables 1 to 178 below. Moreover, the meanings mentioned below for the individual variables in the tables are per se, independ- ently of the combination in which they are mentioned, a particularly preferred embodiment of the substituents in question.

Table 1 Compounds of the formula I. D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is H

Table 2

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is methyl

Table 3

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is ethyl

Table 4 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is propyl

Table 5

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- p ropy I Table 6

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is n- butyl Table 7

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is sec- butyl Table 8

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- butyl Table 9 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is tert- butyl Table 10 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is phenyl Table 11

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is 4- methylphenyl Table 12

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is benzyl Table 13

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is Li ⁺ Table 14

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is Na ⁺

Table 15 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is K ⁺

Table 16

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is Y ₂ Mg ²⁺

Table 17

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

¹ /_Cu ²⁺ Table 18

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

¹ Z-Zn ²⁺

Table 19 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

Y ₂ Fe ²⁺

Table 20

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is !4Ni ²⁺

Table 21

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

NH(CHs) ₃ ⁺ Table 22

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

NH(C ₂ Hs) ₃ ⁺

Table 23 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

Table 24 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

Table 25 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

Table 26

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is me- thylcarbonyl

Table 27

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is ethyl- carbonyl

Table 28

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is pro- pylcarbonyl Table 29

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- propylcarbonyl

Table 30 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is methoxycarbonyl

Table 31

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is eth- oxycarbonyl

Table 32

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is pro- poxycarbonyl

Table 33

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- propoxycarbonyl Table 34

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is phenoxycarbonyl Table 35

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is me- thylaminocarbonyl

Table 36 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is ethylaminocarbonyl

Table 37

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is pro- pylaminocarbonyl

Table 38

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- propylaminocarbonyl

Table 39

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is phenylaminocarbonyl Table 40

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is me- thylsulfonyl

Table 41 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is ethyl- sulfonyl

Table 42

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is pro- pylsulfonyl

Table 43 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- propylsulfonyl

Table 44 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is phenylsulfonyl

Table 45

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is methoxysulfonyl

Table 46

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is eth- oxysulfonyl

Table 47

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is pro- poxysulfonyl Table 48

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- propoxysulfonyl

Table 49 Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is phenoxysulfonyl

Table 50

Compounds of the formula I.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is CN

Table 51

Compounds of the formula I.D2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above

Tables 52 to 101 Compounds of the formula I.D3 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is as defined in any of tables 1 to 50

Table 102 Compounds of the formula I.D4 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above

Table 103

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is H

Table 104

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is methyl Table 105

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is ethyl

Table 106

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is propyl

Table 107

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- propyl

Table 108

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is n- butyl Table 109

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is sec- butyl

Table 110 Compounds of the formula II. D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- butyl

Table 11 1

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is tert- butyl

Table 112

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is phenyl

Table 113

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is 4- methylphenyl

Table 114

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is ben- zyl

Table 115

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is me- thylcarbonyl Table 116

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is ethylcarbonyl

Table 117 Compounds of the formula II. D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is pro- pylcarbonyl

Table 118

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- propylcarbonyl

Table 119

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is phenylcarbonyl

Table 120

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is methoxycarbonyl Table 121

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is eth- oxycarbonyl

Table 122 Compounds of the formula II. D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is pro- poxycarbonyl

Table 123 Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- propoxycarbonyl

Table 124

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is phenoxycarbonyl

Table 125

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is me- thylaminocarbonyl

Table 126

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is ethylaminocarbonyl Table 127

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is pro- pylaminocarbonyl

Table 128 Compounds of the formula II. D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- propylaminocarbonyl

Table 129

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is phenylaminocarbonyl

Table 130

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is me- thylsulfonyl

Table 131

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is ethylsulfonyl Table 132

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is pro- pylsulfonyl Table 133

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- propylsulfonyl

Table 134 Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is phenylsulfonyl

Table 135

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is methoxysulfonyl

Table 136

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is eth- oxysulfonyl

Table 137

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is pro- poxysulfonyl Table 138

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- propoxysulfonyl

Table 139 Compounds of the formula II. D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is phenoxysulfonyl

Table 140

Compounds of the formula II.D1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is CN

Tables 141 to 178

Compounds of the formula II.D2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is as defined in any of tables 103 to 140 In another preferred embodiment of the invention (embodiment E), R ¹ is a group of formula Vl, where A is selected from -(CH ₂ J ₂ -, -CH ₂ -CH(CH ₃ )-, -CH ₂ -CH(C ₂ H ₅ )-,

-CH ₂ -CH(CH ₂ CH ₂ CH ₃ )-, -CH ₂ -CH(CH ₂ CH ₂ CH ₂ CH ₃ )-, -CH ₂ -CHF-, -CH(CHs)-CH(CH ₃ )-, -(CH ₂ )S-, -CH ₂ -CH ₂ -CH(CH ₃ )-, -CH ₂ -CH(CHs)-CH ₂ - and -CH ₂ -C(CHs) ₂ -CH ₂ -, and is preferably -CH ₂ -CH(CH ₂ CH ₂ CHs)-; R ² is phenyl which may carry 1 , 2, 4 or 5 substituents R ⁷ ; and R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings; except for compounds wherein R ² is phenyl, 4-fluorophenyl, 2,4-difluorophenyl, A- chlorophenyl, 2,4-dichlorophenyl, 2,4,6-trichlorophenyl, 4-trifluoromethylphenyl, 2- difluoromethoxyphenyl or 4-trifluoromethoxyphenyl.

More preferably, (embodiment E.1 ), R ¹ is a group of formula Vl, where

A is -CH ₂ -CH(CH ₂ CH ₂ CH ₃ )- ;

R ² is phenyl which may carry 1 , 2 or 3 substituents R ⁷ ; each R ⁷ is independently selected from halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C1-C4- alkoxy and Ci-C ₄ -haloalkoxy, preferably from F, Cl, Br, CH ₃ , CHF ₂ , CF ₃ , OCH ₃ ,

OCHF ₂ and OCF ₃ , and more preferably from F and Cl; and R ⁵ /R ^5a and m have one of the above given general or, preferably, one of the above- given preferred meanings, except for compounds wherein R ² is phenyl, 4-fluorophenyl, 2,4-difluorophenyl, 2,4- dichlorophenyl, 2,4,6-trichlorophenyl, 4-trifluoromethylphenyl, 2-difluoromethoxyphenyl or 4-trifluoromethoxyphenyl, preferably except for compounds wherein R ² is phenyl, 4-fluorophenyl, 2,4- difluorophenyl, 4-chlorophenyl, 2,4-dichlorophenyl, 2,4,6-trichlorophenyl, A- trifluoromethylphenyl, 2-difluoromethoxyphenyl or 4-trifluoromethoxyphenyl.

If R ² is phenyl which carries 1 substituent R ⁷ , this is preferably bound in 2- or A- position, more preferably in 2-position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

If R ² is phenyl which carries 2 substituents R ⁷ , these are preferably bound in 2,4- position, relative to the 1 -position of the attachment point of the phenyl ring to the remainder of the molecule.

Particular compounds of this embodiment E are compounds I and II, wherein - R ⁵ or R ^5a are H, m is 0, A is is -CH ₂ -CH(CH ₂ CH ₂ CH ₃ )- and R ² is 2,3-difluorophenyl (compound E1 );

- R ⁵ or R ^5a are H, m is 0, A is is -CH ₂ -CH(CH ₂ CH ₂ CH ₃ )- and R ² is 2-fluoro-4- chlorophenyl (compound E2); - R ⁵ or R ^5a are H, m is 0, A is is -CH ₂ -CH(CH ₂ CH ₂ CH ₃ )- and R ² is 2-chloro-4- fluorophenyl (compound E3);

- R ⁵ or R ^5a are H, m is 0, A is is -CH ₂ -CH(CH ₂ CH ₂ CH ₃ )- and R ² is 3,4-difluorophenyl (compound E4).

Particular compounds of this embodiment E are also compounds I and II, wherein

- R ⁵ or R ^5a are H, m is 0, A is is -CH ₂ -CH(CH ₂ CH ₂ CH ₃ )- and R ² is 4-chlorophenyl (compound E5);

- R ⁵ or R ^5a are H, m is 0, A is is -CH ₂ -CH(CH ₂ CH ₂ CH ₃ )- and R ² is 2,4-difluorophenyl (compound E6).

Examples for preferred compounds I and Il of embodiment E are compounds of formulae I.E1 , I.E2 and II. E1 , where the variables R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ are hydrogen or have one of the general or, in particular, one of the preferred meanings given above for R ⁷ , and where the variables R ⁵ and R ^5a have one of the general or, in particular, one of the preferred meanings given above. Examples of preferred compounds are the individual compounds compiled in the tables 1 to 89 below. Moreover, the meanings mentioned below for the individual variables in the tables are per se, independently of the combination in which they are mentioned, a particularly preferred embodiment of the substituents in question.

Table 1

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is H Table 2

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is methyl Table 3

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is ethyl

Table 4 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is propyl

Table 5

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- p ropy I

Table 6

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is n- butyl

Table 7

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is sec- butyl Table 8

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- butyl

Table 9 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is tert- butyl

Table 10

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is phenyl

Table 11

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is 4- methylphenyl

Table 12

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is ben- zyl Table 13

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is Li ⁺

Table 14 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is Na ⁺

Table 15

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is K ⁺ Table 16

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

¹ / ₂ Mg ²⁺

Table 17 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

¹ Z-Cu ²⁺

Table 18

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

¹ Z-Zn ²⁺

Table 19

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

Table 20

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is !4Ni ²⁺

Table 21 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

NH(CHs) ₃ ⁺

Table 22

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

NH(C ₂ Hs) ₃ ⁺

Table 23 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

Table 24 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

Table 25

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is

Table 26

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is me- thylcarbonyl

Table 27

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is ethyl- carbonyl Table 28

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is pro- pylcarbonyl

Table 29 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- propylcarbonyl

Table 30

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is methoxycarbonyl

Table 31

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is eth- oxycarbonyl

Table 32

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is pro- poxycarbonyl Table 33

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- propoxycarbonyl Table 34

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is phenoxycarbonyl

Table 35 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is me- thylaminocarbonyl

Table 36

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is ethylaminocarbonyl

Table 37

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is pro- pylaminocarbonyl

Table 38

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- propylaminocarbonyl Table 39

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is phenylaminocarbonyl

Table 40 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is me- thylsulfonyl

Table 41

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is ethyl- sulfonyl

Table 42 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is pro- pylsulfonyl

Table 43 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- propylsulfonyl

Table 44

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is phenylsulfonyl

Table 45

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is methoxysulfonyl

Table 46

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is eth- oxysulfonyl Table 47

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is pro- poxysulfonyl

Table 48 Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is iso- propoxysulfonyl

Table 49

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is phenoxysulfonyl

Table 50

Compounds of the formula I.E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ⁵ is CN Table 51

Compounds of the formula I.E2 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above Table 52

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is H

Table 53 Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is methyl

Table 54

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is ethyl

Table 55

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is propyl Table 56

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- p ropy I

Table 57 Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is n- butyl

Table 58

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is sec- butyl

Table 59

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- butyl

Table 60

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is tert- butyl Table 61

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is phenyl Table 62

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is 4- methylphenyl Table 63

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is benzyl

Table 64 Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is me- thylcarbonyl

Table 65

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is ethylcarbonyl

Table 66

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is pro- pylcarbonyl

Table 67

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- propylcarbonyl Table 68

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is phenylcarbonyl

Table 69 Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is methoxycarbonyl

Table 70

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is eth- oxycarbonyl

Table 71 Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is pro- poxycarbonyl

Table 72 Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- propoxycarbonyl

Table 73

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is phenoxycarbonyl

Table 74

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is me- thylaminocarbonyl

Table 75

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is ethylaminocarbonyl Table 76

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is pro- pylaminocarbonyl

Table 77 Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- propylaminocarbonyl

Table 78

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is phenylaminocarbonyl

Table 79

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is me- thylsulfonyl

Table 80

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is ethylsulfonyl Table 81

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is pro- pylsulfonyl Table 82

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- propylsulfonyl

Table 83 Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is phenylsulfonyl

Table 84

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is methoxysulfonyl

Table 85

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is eth- oxysulfonyl

Table 86

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is pro- poxysulfonyl Table 87

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is iso- propoxysulfonyl

Table 88 Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is phenoxysulfonyl

Table 89

Compounds of the formula II. E1 in which the combination of R ⁷¹ , R ⁷² , R ⁷³ , R ⁷⁴ and R ⁷⁵ for a compound corresponds in each case to one row of Table A above and R ^5a is CN

Among the above embodiments A, B, C, D and E, preference is given to embodiment

E. Compounds of formulae I and Il can be prepared by one or more of the following methods and variations as described in schemes 1 to 14 and in the syntheses descriptions below. The variables are as defined above for formulae I and II.

Compounds of formula I, wherein R ⁵ is H and m is 0 (or compounds II, wherein R ^5a is H), can be prepared by sulfurizing the corresponding triazole derivative IV as outlined in scheme 1. Sulfurization can be carried out in analogy to known processes, for example as described in WO 96/16048, WO 97/06152 or DE-A-19620407. For instance, the triazolyl ring can be first deprotonated with a strong base, e.g. an organolithium base, such as n-butyllithium, tert-butyllithium or sec-butyllithium, lithium diisopropyl amide, sodium hydride, sodium amide or potassium tert-butylate mixed with tetrame- thylethylene diamine (TMEDA), and then the resulting anion is reacted with elemental sulfur. Sulfur is generally used in powdered form. The reaction is generally carried out in an inert solvent, such as ethers, e.g. diethylether, methyl-tert-butylether, tetrahydro- furan or dioxane, dimethoxyethane, liquid ammonia, dimethylsulfoxide or dimethylfor- mamide. The reaction temperature is not very critical and can range, for example, from -70 to +50 ⁰ C, preferably from -70 to 0 ⁰ C. Alternatively, sulfurization can be carried out in the absence of a base by reacting IV with elemental sulfur in a high-boiling solvent, such as N-methylpyrrolidinone, dimethylsulfoxide or N,N-dimethylformamide, while heating, e.g. to 160 to 250 ⁰ C. After completion of the reaction, the resulting mixture is hydrolyzed, e.g. by the addition of water or an aqueous acid, such as a mineral acid (e.g. dilute sulfuric acid or hydrochloric acid), acetic acid or ammoniumchloride, to give compound I.

Scheme 1

IV I

(R ⁵ /R ^5a = H; m = 0)

The triazole compound IV, wherein R ¹ is a group V wherein R ⁴ is OH, can be prepared in analogy to known methods, such as described, for example, in EP-A-15756, EP-A- 537957 or DE-A-3042302, as outlined in scheme 2. For instance, the oxirane compound 1 and [1 ,2,4]-1 H-triazole can be reacted in the presence of a base, such as an alkali metal hydride (e.g. sodium hydride, potassium hydride), an alkali metal hydroxide (e.g. sodium hydroxide, potassium hydroxide), or an alkali metal carbonate (e.g. so- dium carbonate, potassium carbonate, caesium carbonate). The reaction is suitably carried out in a solvent. Suitable solvents are, for example, toluene, N- methypyrrolidinone, ethers (e.g. diethyl ether, tetrahydrofuran), alcohols (e.g. methanol, ethanol, isopropanol or tert-butanol), acetonitrile, or N,N-dimethylformamide.

Scheme 2

(R ⁴ = OH)

The oxirane 1 in turn can be prepared in analogy to known methods, such as described, for example, in EP-A-0267778, Org. Syn. 49, 78 (1968) or J. Am. Chem. Soc. 1975, 1353, as outlined in scheme 3 below. For instance, the ketone 2 may be reacted with a sulfonium ylide or an oxosulfonium ylide, such as dimethyloxosulfonium me- thylide or dimethylsulfonium methylide in a solvent. Alternatively, the oxirane 1 can be prepared in an epoxidation reaction in analogy to the method described in Tetrahedron Lett. 23, 5283 (1982) or in EP-A-0655443 by subjecting 2 to the reaction with a trimethylsulfonium salt, such as trimethylsulfonium bromide, trimethylsulfonium iodide or methyltrimethylsulfonium sulfate, in the presence of a metal oxide, such as alkaline metal oxides (e.g. sodium oxide, potassium oxide), alkaline earth metal oxides (e.g. magnesium oxide, calcium oxide, barium oxide) or zinc oxide, and optionally a base, such as alkali metal hydrides (e.g. sodium hydride, potassium hydride), alkali metal hydroxides (e.g. sodium hydroxide, potassium hydroxide), alkali metal carbonates (e.g. sodium carbonate, potassium carbonate, caesium carbonate) in a two-phase solid/liquid system comprising an organic solvent, such as toluene, N- methypyrrolidinone, ethers (e.g. diethyl ether, tetrahydrofuran), acetonitrile or N, N- dimethylformamide. Alternatively, the oxirane 1 can be prepared in analogy to the method described in Tetrahedron 1985, 1259 by epoxidation of 2 with a trimethylsulfonium salt, such as trimethylsulfonium bromide, trimethylsulfonium iodide or methyltrimethylsulfonium sulfate, or a trimethylsulfoxonium salt, such as trimethylsulfoxonium bromide, trimethylsulfoxonium iodide or methyltrimethylsulfoxonium sulfate and potassium sulfate/aluminium oxide.

Scheme 3

The ketone 2 can be obtained from the halide 4" by a Grignard reaction with the aldehyde 5\ or from the halide 4" by a Grignard reaction with the aldehyde 5", as outlined in scheme 4 below. Oxidation of the obtained alcohol 3 via known methods, such as oxidation with the Swern reagent, hypervalent iodine compounds (IBX, Martin's reagent), chromine compounds (e.g. pyridinium dichromate, pyridinium chlorochromate, dipyridinium chromine trioxide), sodium hypochlorite and the like, yields the ketone 2.

Scheme 4

(Hal = halogen)

Alternatively, the ketone 2 can be prepared by a Friedel-Crafts acylation of R ² -H with the acylchloride R ³ -C(=O)-CI in the presence of a Lewis acid, such as AICb or FeCb, under reaction conditions customary for this reaction type.

As an alternative to the process described in scheme 3, the oxirane 1 can be prepared in analogy to the method described in Org. Syn. 40, 66, 1966, J. Org. Chem. 28, 1 128, 1963 and Org. Syn. Coll. Vol. 4, 552, 1963 as outlined in scheme 5 below by first subjecting the ketone 2 to a Wittig reaction, thus yielding the corresponding olefinic compound 6, and then subjecting this to an epoxidation reaction. The Wittig reaction can be carried out under standard conditions, such as the use of methyltriphenylphosphonium bromide or iodide in the presence of an alkali metal base, such as n-butyllithium, sec- butyllithium or tert-butyllithium. Epoxidation can also be carried out with standard reagents, such as peracetic acid, perbenzoic acid meta-chloroperbenzoic acid, perphthalic acid and the like. Olefination (i.e. transformation of the C=O into a C=CHb group) of 2 can alternatively be achieved by the use of Tebbe's reagent ((C ₅ Hs) ₂ TiCH ₂ CIAI(CHs) ₂ ).

Scheme 5

olefination epoxidation

As an alternative to the process described in scheme 1 , compounds I, wherein R ⁵ is H and m is 0 (or compounds II, wherein R ^5a is H) and wherein R ¹ is a group V wherein R ⁴ is OH, can also be prepared in analogy to the method described in WO 99/18088 as outlined in scheme 6 below. Epoxide opening of 1 with hydrazine, optionally in the presence of an acid (e.g. hydrochloric acid, hydrobromic acid, acetic acid, sulfuric acid or p-toluenesulfonic acid) or a base (e.g. triethylamine, diisopropylethylamine, sodium carbonate or potassium carbonate) in a suitable solvent, such as an alcohol (e.g. methanol, ethanol, isopropanol, tert-butanol), N-methylpyrrolidinone, an ether (e.g. diethyl ether, tetrahydrofuran, dioxane, 1 ,2-dimethoxyethane), acetonitrile, N,N-dimethyl- formamide or dimethylsulfoxide, yields 7. This is then converted into the semicarbazide 8 by reaction with a thiocyanate, such as sodium thiocyanate, potassium thiocyanate or ammonium thiocyanate (i.e. M ⁺ = e.g. Na ⁺ , K ⁺ , NH ₄ ⁺ ), in a suitable solvent, such as an alcohol (e.g. methanol, ethanol, isopropanol, tert-butanol), N-methylpyrrolidinone, an ether (e.g. diethyl ether, tetrahydrofuran, dioxane, 1 ,2-dimethoxyethane), acetonitrile, N,N-dimethylformamide, dimethylsulfoxide, toluene or xylene. The semicarbazide is then converted into l/ll via reaction with a formic acid alkyl ester (e.g. formic acid methyl ester, formic acid ethyl ester) in a solvent. Suitable solvents are, for example, alcohols (e.g. methanol, ethanol, isopropanol, tert-butanol), N-methylpyrrolidinone, ethers (e.g. diethyl ether, tetrahydrofuran, dioxane, 1 ,2-dimethoxyethane), acetonitrile, N,N-dimethylformamide, dimethylsulfoxide, toluene or xylene. Alternatively, 7 can be reacted with hydrogen thiocyanate and formaldehyde in a solvent. Suitable solvents are, for example, alcohols (e.g. methanol, ethanol, isopropanol, tert-butanol), N-methyl- pyrrolidinone, ethers (e.g. diethyl ether, tetrahydrofuran, dioxane, 1 ,2-dimethoxyethane), acetonitrile, N,N-dimethylformamide, dimethylsulfoxide, toluene or xylene. The resulting triazolidinthione 9 is then oxidized using, for example, FeCb in an aqueous acid (e.g. hydrochloric acid) or oxygen in the presence of an alkali metal hydroxide (e.g. sodium hydroxide, potassium hydroxide) and elemental sulfur to l/ll. In a yet fur- ther alternative, 7 is reacted with a dialkyl ketone (e.g. acetone, diethylketone, methyl ethyl ketone) and a thiocyanate (e.g. sodium thiocyanate, potassium thiocyanate, ammonium thiocyanate) in a solvent to give the triazolidinthione 10. Suitable solvents are, for example, alcohols (e.g. methanol, ethanol, isopropanol, tert-butanol), N- methylpyrrolidinone, ethers (e.g. diethyl ether, tetrahydrofuran, dioxane, 1 ,2- dimethoxyethane), acetonitrile, N,N-dimethylformamide, dimethylsulfoxide, toluene or xylene. The triazolidinthione 10 is then converted into l/ll by reaction with formic acid in the presence of an acid (e.g. hydrochloric acid, hydrobromic acid, acetic acid, sulfuric acid, p-toluenesulfonic acid) or a metal oxide (e.g. amorphous Tiθ2).

Scheme 6

Oxidation

(R ⁵ / _R ^5a = H, m = O, R ¹ = group V, wherein R ⁴ = OH)

The halides 4 ¹ and 4", the aldehydes 5 ¹ and 5" and the compounds R ² -H and R ³ -C(=O)-CI used in the above reactions are either commercially available or can be produced by standard methods known to the skilled person.

The triazole compound IV, wherein R ¹ is a group V wherein R ⁴ is CN, can be prepared in analogy to known methods, such as described, for example, in EP-A-145294 or DE- A-3721786, as outlined in scheme 7. For instance, the bromide 11 and [1 ,2,4]-1 H- triazole can be reacted in the presence of a base, such as an alkali metal hydride (e.g. sodium hydride, potassium hydride), an alkali metal hydroxide (e.g. sodium hydroxide, potassium hydroxide), or an alkali metal carbonate (e.g. sodium carbonate, potassium carbonate, caesium carbonate). The reaction is suitably carried out in a solvent. Suitable solvents are, for example, toluene, the xylenes, dimethylsulfoxide, or N, N- dimethylformamide. The reaction temperature is not very critical and can range, for example, from 0 to 150 ⁰ C and is preferably in the range from 25 to 100 ⁰ C.

Scheme 7

(R ⁴ = CN)

The bromide 11 can in turn be prepared by bromomethylation of 12 with methylene- bromide in the presence of a base, such as an alkali metal hydride (e.g. sodium hydride, potassium hydride), an alkali metal hydroxide (e.g. sodium hydroxide, potassium hydroxide), or an alkali metal alcoholate (e.g. sodium methoxide, potassium methoxide or potassium tert-butanolate), as outlined in scheme 8. The reaction temperature is not very critical and can range, for example, from 0 to 150°C and is preferably in the range from 25 to 100 ⁰ C.

Scheme 8 base 1 ^{2 11}

Compounds 12, wherein R ³ is an aliphatic or cycloaliphatic group, can be prepared by phase transfer alkylation of the benzylcyanide 13 with the compound 14, wherein X is a good leaving group, such as Cl, Br, I, tosylae or triflate, in the presence of a base, such as an alkali metal hydroxide (e.g. sodium hydroxide, potassium hydroxide), or an alkali metal alcoholate (e.g. sodium methoxide, potassium methoxide or potassium tert- butanolate), and a suitable phase transfer catalyst, such as tetrabutylammnium bromide, as outlined in scheme 9.

Scheme 9

14 13 12

Compounds 13 and 14 used in the above reactions are either commercially available or can be produced by standard methods known to the skilled person.

The triazole compound IV, wherein R ¹ is a group V wherein R ⁴ is H, can be prepared in analogy to known methods, such as described, for example, in EP-A-145294 or DE-A- 2735827, as outlined in scheme 10. For instance, compound 15, wherein X is a good leaving group, such as Cl, Br, I, tosylate or triflate, and [1 ,2,4]-1 H-triazole can be re- acted in the presence of a base, such as an alkali metal hydride (e.g. sodium hydride, potassium hydride), an alkali metal hydroxide (e.g. sodium hydroxide, potassium hydroxide), or an alkali metal carbonate (e.g. sodium carbonate, potassium carbonate, caesium carbonate). The reaction is suitably carried out in a solvent. Suitable solvents are, for example, toluene, the xylenes, dimethylsulfoxide, or N,N-dimethylformamide. The reaction temperature is not very critical and can range, for example, from 0 to 150 ⁰ C and is preferably in the range from 25 to 100 ⁰ C.

Scheme 10

(R ⁴ = H)

The triazole compound IV, wherein R ¹ is a group Vl, can be prepared in analogy to known methods, such as described, for example, in DE-A-255156 or EP-A-0065485, as outlined in scheme 1 1. For instance, the compound 16, wherein X is a good leaving group, such as a halogen atom, in particular Cl, Br or I, phenylsulfonyloxy, p-tosyloxy, trifluoroacetyloxy or alkylsulfonyloxy, such as mesyloxy, can be reacted with the [1 ,2,4]- 1 H-triazole compound 17, wherein M is a hydrogen atom or a metal atom, in particular an alkali metal atom, such as Li, Na or K. In case M is H, the reaction is suitably carried out in the presence of a base, such as an alkali metal hydride (e.g. sodium hydride, potassium hydride), an alkali metal hydroxide (e.g. sodium hydroxide, potassium hy- droxide), an alkali metal carbonate (e.g. sodium carbonate, potassium carbonate, caesium carbonate) or a suitable amine (e.g. triethylamine, triethylenediamine, piperidine, pyridine, 4-dimethylaminopyτidine, 4-pyrrolidylpyridine). If X is Cl or Br, the reaction can be accelerated by the addition of an alkali metal iodide, such as NaI or Kl. The reaction is suitably carried out in a solvent. Suitable solvents are inert versus the reacants and products and are rather polar, for example, N,N-dimethylformamide, N,N-dimethylacet- amide, dimethylsulfoxide, acetonitrile, benzonitrile, ethers, such as diethyl ether, dipro- pyl ether, methyl-tert-butyl ether, tetrahydrofuran or dioxane, and the like, and can be used in combination with other inert, less polar solvents, such as benzene, toluene, the xylenes, chlorobenzene, nitrobenzene, hexane, heptane, petrolether and the like. The reaction temperature is not very critical and can range, for example from 0 to 220 ⁰ C and preferably from 80 to 170 ⁰ C. Suitably, the reaction is carried out at reflux temperature of the reaction mixture.

Scheme 1 1

(R ¹ = a group Vl)

Compound 16 in turn can be prepared in analogy to known methods, such as described, for example, in DE-A-255156 or EP-A-0065485 or in Synthesis, 1974, I, 23, as outlined in scheme 12 below. For instance, the ketone 18 may be reacted with a diol HO-A-OH for several hours preferably in the presence of an azeotrope-forming com- pound, such as benzene, toluene, xylene, chloroform or tetrachloromethane, which can also serve as reaction solvents. Alternatively, a mixture of a solvent which doesn't form an azeotrope with water and an azeotrope-forming solvent, such as ethanol, propanol, butanol or pentanol, is used. The ketalization reaction is accelerated by the presence of a strong acid, such p-toluenesulfonic acid. The reaction is generally carried out at re- flux. Subsequent halogenation of the resulting ketale 19 yields ketale 16, wherein X is a halogen atom, which, if desired, can be converted into a compound 16, wherein X is a leaving group X other than halogen.

Scheme 12

18 19 16

As an alternative to the process described in scheme 11 , compound IV can be prepared in analogy to the method described in EP-A-0065485 as outlined in scheme 13 below by a ketalization reaction of the ketone 20 with a diol HO-A-OH. The ketalization reaction can be carried out under reaction conditions described for scheme 12.

Scheme 13

(R ¹ = a group Vl)

The ketone 20 in turn can be prepared in analogy to the method described in EP-A- 0065485 as outlined in scheme 14 below by reacting the compound 21 , wherein X is a good leaving group, such as a halogen atom, in particular Cl, Br or I, phenylsulfonyloxy, p-tosyloxy, trifluoroacetyloxy or alkylsulfonyloxy, such as mesyloxy, with the triazole compound 17 under reaction conditions described for the reaction in scheme 1 1. Compound 21 , in turn, can be obtained from the halogenation of the ketone 18.

Scheme 14

Ketone 18 used in the above reactions is either commercially available or can be produced by standard methods known to the skilled person, for instance by a Friedel- Crafts acylation of R ² -H with acetylchloride in the presence of a Lewis acid, such as AICb or FeCb, under reaction conditions customary for this reaction type. Compounds of formula I, wherein R ⁵ is different from hydrogen and m is 0, can be prepared from compounds I (wherein R ⁵ = H and m = 0).

Compounds of formula I, wherein m is 0 and R ⁵ is Ci-Cio-alkyl, Ci-Cio-haloalkyl, C2- Cio-alkenyl, C2-Cio-haloalkenyl, C2-Cio-alkynyl, C2-Cio-haloalkynyl, C3-Cio-cycloalkyl, C3-Cio-halocycloalkyl, phenyl, phenyl-Ci-C4-alkyl, where the phenyl moiety in the 2 last- mentioned radicals may be substituted as described above, and a 5- or 6-membered saturated, partially unsaturated or aromatic heterocyclic ring containing 1 , 2 or 3 het- eroatoms selected from N, O and S as ring members, where the heterocyclic ring may be substituted as described above, may be prepared in analogy to the method described in DE-A-19520098 by reacting a compound I, wherein m is 0 and R ⁵ is H, with a compound R ⁵ -LG, where R ⁵ has one of the above meanings and LG is a leaving group, such as a halide (e.g. Cl, Br, I), a tosylate or a mesylate, in the presence of a base. Suitable bases are, for example, alkali metal hydrides (e.g. sodium hydride, po- tassium hydride), alkali metal hydroxides (e.g. sodium hydroxide, potassium hydroxide), alkali metal carbonates (e.g. sodium carbonate, potassium carbonate, caesium carbonate), alkali metal alkoxides (e.g. sodium methoxide, potassium methoxide, sodium ethoxide, potassium ethoxide, potassium tert-butoxide) or organolithium bases (e.g. n-butyl lithium, sec-butyl lithium, tert-butyl lithium and lithium diisopropylamine.). The reaction is generally carried out in a suitable solvent. Suitable solvents are, for example, toluene, N-methylpyrrolidinone, ethers (e.g. diethyl ether, tetrahydrofuran, dioxane, 1 ,2-dimethoxyethane), acetonitrile, N,N-dimethylformamide or dimethylsulfox- ide.

Alternatively, compounds of formula I, wherein m is 0 and R ⁵ is Ci-Cio-alkyl, Ci-Cio- haloalkyl, C2-Cio-alkenyl, C2-Cio-haloalkenyl, C2-Cio-alkynyl, C2-Cio-haloalkynyl, C3-C10- cycloalkyl, C3-Cio-halocycloalkyl, phenyl, phenyl-Ci-C4-alkyl, where the phenyl moiety in the 2 last-mentioned radicals may be substituted as described above, and a 5- or 6- membered saturated, partially unsaturated or aromatic heterocyclic ring containing 1 , 2 or 3 heteroatoms selected from N, O and S as ring members, where the heterocyclic ring may be substituted as described above, may be prepared in analogy to the method described in Heterocycles, 23(7), 1645-1649, 1985 by reacting compound IV with a disulfide R ⁵ -S-S-R ⁵ in the presence of a strong base under conditions similar to those described for scheme 1.

Compounds of formulae I, wherein m is 0 and R ⁵ is -C(=O)R ¹³ or -C(=S)R ¹³ , may be prepared in analogy to the method described in DE-A-19617461 by reacting a compound I, wherein m is 0 and R ⁵ is H, with a compound R ¹³ -C(=O)-W, R ¹³ -C(=S)-W, R ¹³ '- N=C=O or R ¹³ '-N=C=S, wherein R ¹³ has one of the above meanings, R ¹³ ' is C1-C10- alkyl or Ci-Cio-haloalkyl and W is a good leaving group, such as a halide (e.g. Cl, Br, I), an alkoxide (e.g. methoxide, ethoxide) or pentafluorophenoxide, in the presence of a base. Suitable bases are, for example, alkali metal hydrides (e.g. sodium hydride, potassium hydride), alkali metal hydroxides (e.g. sodium hydroxide, potassium hydrox- ide), alkali metal carbonates (e.g. sodium carbonate, potassium carbonate, caesium carbonate), alkali metal alkoxides (e.g. sodium methoxide, potassium methoxide, sodium ethoxide, potassium ethoxide, potassium tert-butoxide) or organolithium bases (e.g. n-butyl lithium, sec-butyl lithium, tert-butyl lithium, lithium diisopropylamine). The reaction is generally carried out in a suitable solvent. Suitable solvents are, for exam- pie, toluene, N-methylpyrrolidinone, ethers (e.g. diethyl ether, tetrahydrofuran, dioxane, 1 ,2-dimethoxyethane), acetonitrile, N,N-dimethylformamide or dimethylsulfoxide.

Compounds of formula I, wherein m is 0 and R ⁵ is -SO2R ¹³ , may be prepared in analogy to the method described in DE-A-19620590 by reacting a compound I, wherein m is 0 and R ⁵ is H, with a compound R ¹³ -Sθ2-W, wherein R ¹³ has one of the above meanings and W is a good leaving group, such as a halide (e.g. Cl, Br, I), an alkoxide (e.g. methoxide, ethoxide) or pentafluorophenoxide, in the presence of a base. Suitable bases are, for example, alkali metal hydrides (e.g. sodium hydride, potassium hydride), alkali metal hydroxides (e.g. sodium hydroxide, potassium hydroxide), alkali metal car- bonates (e.g. sodium carbonate, potassium carbonate, caesium carbonate), alkali metal alkoxides (e.g. sodium methoxide, potassium methoxide, sodium ethoxide, potassium ethoxide, potassium tert-butoxide) or organolithium bases (e.g. n-butyl lithium, sec-butyl lithium, tert-butyl lithium, lithium diisopropylamine). The reaction is generally carried out in a suitable solvent. Suitable solvents are, for example, toluene, N- methylpyrrolidinone, ethers (e.g. diethyl ether, tetrahydrofuran, dioxane, 1 ,2- dimethoxyethane), acetonitrile, N,N-dimethylformamide or dimethylsulfoxide.

Compounds of formula I, wherein m is 0 and R ⁵ is -CN, may be prepared in analogy to the method described in DE-A-19620407 by reacting a compound I, wherein m is 0 and R ⁵ is H, with a compound CN-W, wherein W is a good leaving group, such as a halide (e.g. Cl, Br, I), in the presence of a base. Suitable bases are, for example, alkali metal hydrides (e.g. sodium hydride, potassium hydride), alkali metal hydroxides (e.g. sodium hydroxide, potassium hydroxide), alkali metal carbonates (e.g. sodium carbonate, potassium carbonate, caesium carbonate), alkali metal alkoxides (e.g. sodium methoxide, potassium methoxide, sodium ethoxide, potassium ethoxide, potassium tert-butoxide) or organolithium bases (e.g. n-butyl lithium, sec-butyl lithium, tert-butyl lithium, lithium diisopropylamine). The reaction is generally carried out in a suitable solvent. Suitable solvents are, for example, toluene, N-methylpyrrolidinone, ethers (e.g. diethyl ether, tetrahydrofuran, dioxane, 1 ,2-dimethoxyethane), acetonitrile, N,N-dimethylformamide or dimethylsulfoxide.

Compounds of formula I, wherein m is 0 and R ⁵ is M, may be prepared in analogy to the method described in DE-A-19617282 by reacting a compound I with an amine NR ^a R ^b R ^c , wherein R ^a , R ^b and R ^c are as defined above, or with a metal salt, such as sodium hydroxide, potassium hydroxide or copper acetate.

Compounds of formula I, wherein m is 0 and R ⁵ is a group of formula III, may be pre- pared in analogy to the method described in WO 97/43269 by reacting a compound I, wherein m is O and R ⁵ is H, with a halogen, especially iodine, in the presence of a base. Suitable bases are, for example, alkali metal hydrides (e.g. sodium hydride, potassium hydride), alkali metal hydroxides (e.g. sodium hydroxide, potassium hydroxide), alkali metal carbonates (e.g. sodium carbonate, potassium carbonate, caesium carbonate), alkali metal alkoxides (e.g. sodium methoxide, potassium methoxide, sodium ethoxide, potassium ethoxide, potassium tert-butoxide) or organolithium bases (e.g. n-butyl lithium, sec-butyl lithium, tert-butyl lithium, lithium diisopropylamine). The reaction is generally carried out in a suitable solvent. Suitable solvents are, for example, toluene, N-methylpyrrolidinone, ethers (e.g. diethyl ether, tetrahydrofuran, dioxane, 1 ,2-dimethoxyethane), acetonitrile, N,N-dimethylformamide or dimethylsulfoxide.

Compounds of formula I, wherein m is 0 and R ⁵ is -P(=Q)R ¹⁴ R ¹⁵ , may be prepared in analogy to the method described in WO 99/05149.

Compounds of formula II, wherein R ^5a is hydrogen (or compounds of formula I, wherein m is 0 and R ⁵ is hydrogen), can be prepared in analogy to the method described in WO 99/18087 by reacting a triazolidinthione 9 with an oxidizing agent, optionally in the presence of a catalyst. Suitable oxidizing agents are, for example, oxygen, sulfur and potassium superoxide. Especially in case oxygen is used as oxidizing agent, it is ad- vantageous to carry out the oxidation reaction in the presence of a catalyst. A suitable catalyst is, for example, a mixture of powdery sulfur and KOH. The reaction is generally carried out in a suitable solvent. Suitable solvents are, for example, aliphatic hydrocarbons (e.g. pentane, hexane), cycloaliphatic hydrocarbons (e.g. cyclohexane), aromatic hydrocarbons (e.g. bemzene, toluene, the xylenes), ethers (e.g. diethylether, methyl- tert-butylether), and esters (e.g. ethylecetate, propylacetate, n-butylacetate).

The oxidation of the triazolidinthione 9 may also be carried out with ferric chloride (FeCb) in an acidic aqueous solution in analogy to the method described in WO 01/46158. The reaction is generally carried out in a suitable solvent. Suitable solvents are, for example, ethanol, ethylacetate and mixtures of ethanol with toluene.

The oxidation of the triazolidinthione 9 may also be carried out with formic acid, option- ally in the presence of a catalyst, in analogy to the method described in WO 99/18086 or WO 99/18088. Suitable catalysts are, for example, acids, like hydrochloric acid, sulfuric acid or p-toluenesulfonic acid, and metal oxides, like amorphous titanium dioxide. The reaction is generally carried out in a suitable solvent. Suitable solvents are weakly polar solvents like, for example, alcohols such as propanol, butanol and pentanol, es- ters, like ethyl acetate, butyl acetate and isobutyl formate, ethers, like 1 ,2- dimethoxyethane, methyl-tert-butyl ether and methyl-tert-amylether, and formic acid used in excess.

Compounds of formula II, wherein R ^5a is different from hydrogen, can be prepared by reacting the NR ^5a group, wherein R ^5a is H, in analogy to the above-described conversion of compounds I, wherein R ⁵ is H, into compounds, wherein R ⁵ is different from H.

Compounds I, wherein m is 1 or 2, can be prepared from respective compounds I, wherein m is 0, by oxidation. Alternatively, compounds I, wherein m is 2, can be pre- pared from compounds IV by first deprotonating the triazolyl ring and then reacting with a sulfonyl chloride R ⁵ Sθ2CI. Compounds I, wherein m is 3, can be prepared from compounds IV by first deprotonating the triazolyl ring and then reacting with sulfuric acid chloride or a sulfuric ester chloride of formula R ⁵ OSθ2CI, wherein R ⁵ is selected from hydrogen, Ci-Cio-alkyl, Ci-Cio-haloalkyl, C2-Cio-alkenyl, C2-Cio-haloalkenyl, C2-C10- alkynyl, C2-Cio-haloalkynyl, C3-Cio-cycloalkyl, C3-Cio-halocycloalkyl, phenyl, phenyl-Ci- C4-alkyl, where the phenyl moiety in the 2 last-mentioned radicals may be substituted as mentioned above, and a 5- or 6-membered saturated, partially unsaturated or aromatic heterocyclic ring containing 1 , 2 or 3 heteroatoms selected from N, O and S, wherein the heterocyclic ring may be substituted as mentioned above.

If individual compounds cannot be prepared via the above-described routes, they can be prepared by derivatization of other compounds I and Il or by customary modifications of the synthesis routes described.

The reaction mixtures are worked up in the customary manner, for example by mixing with water, separating the phases, and, if appropriate, purifying the crude products by chromatography, for example on alumina or silica gel. Some of the intermediates and end products may be obtained in the form of colorless or pale brown viscous oils, which are freed or purified from volatile components under reduced pressure and at moder- ately elevated temperature. If the intermediates and end products are obtained as solids, they may be purified by recrystallization or digestion.

A further aspect of the invention relates to compounds of formula IV

Λ— N

// W

N

> N

R' (IV)

wherein R ¹ has one of the general or, in particular, one of the preferred meanings given above for compounds I and II.

Compounds IV are on the one side valuable intermediates in the preparation of compounds I and Il (see above schemes), but on the other side show a remarkable fungicidal activity, too.

The invention further refers to an agricultural composition comprising at least one com- pound of formula I and/or Il as defined above or an agriculturally acceptable salt thereof and a liquid or solid carrier. Suitable carriers, as well as auxiliaries and further active compounds which may also be contained in the composition of the invention are defined below.

The compounds I and Il and the compositions according to the invention, respectively, are suitable as fungicides. They are distinguished by an outstanding effectiveness against a broad spectrum of phytopathogenic fungi, including soil-borne fungi, which derive especially from the classes of the Plasmodiophoromycetes, Peronosporomy- cetes (syn. Oomycetes), Chytridiomycetes, Zygomycetes, Ascomycetes, Basidiomy- cetes and Deuteromycetes (syn. Fungi imperfecti). Some are systemically effective and they can be used in crop protection as foliar fungicides, fungicides for seed dressing and soil fungicides. Moreover, they are suitable for controlling harmful fungi, which inter alia occur in wood or roots of plants.

The compounds I and Il and the compositions according to the invention are particularly important in the control of a multitude of phytopathogenic fungi on various cultivated plants, such as cereals, e. g. wheat, rye, barley, triticale, oats or rice; beet, e. g. sugar beet or fodder beet; fruits, such as pomes, stone fruits or soft fruits, e. g. apples, pears, plums, peaches, almonds, cherries, strawberries, raspberries, blackberries or gooseberries; leguminous plants, such as lentils, peas, alfalfa or soybeans; oil plants, such as rape, mustard, olives, sunflowers, coconut, cocoa beans, castor oil plants, oil palms, ground nuts or soybeans; cucurbits, such as squashes, cucumber or melons; fiber plants, such as cotton, flax, hemp or jute; citrus fruit, such as oranges, lemons, grapefruits or mandarins; vegetables, such as spinach, lettuce, asparagus, cabbages, carrots, onions, tomatoes, potatoes, cucurbits or paprika; lauraceous plants, such as avocados, cinnamon or camphor; energy and raw material plants, such as corn, soybean, rape, sugar cane or oil palm; corn; tobacco; nuts; coffee; tea; bananas; vines (table grapes and grape juice grape vines); hop; turf; natural rubber plants or ornamental and forestry plants, such as flowers, shrubs, broad-leaved trees or evergreens, e. g. conifers; and on the plant propagation material, such as seeds, and the crop material of these plants.

Preferably, compounds I and Il and compositions thereof, respectively are used for controlling a multitude of fungi on field crops, such as potatoes sugar beets, tobacco, wheat, rye, barley, oats, rice, corn, cotton, soybeans, rape, legumes, sunflowers, coffee or sugar cane; fruits; vines; ornamentals; or vegetables, such as cucumbers, tomatoes, beans or squashes.

The term "plant propagation material" is to be understood to denote all the generative parts of the plant such as seeds and vegetative plant material such as cuttings and tubers (e. g. potatoes), which can be used for the multiplication of the plant. This includes seeds, roots, fruits, tubers, bulbs, rhizomes, shoots, sprouts and other parts of plants, including seedlings and young plants, which are to be transplanted after germination or after emergence from soil. These young plants may also be protected before transplantation by a total or partial treatment by immersion or pouring.

Preferably, treatment of plant propagation materials with compounds I and Il and compositions thereof, respectively, is used for controlling a multitude of fungi on cereals, such as wheat, rye, barley and oats; rice, corn, cotton and soybeans.

The term "cultivated plants" is to be understood as including plants which have been modified by breeding, mutagenesis or genetic engineering including but not limiting to agricultural biotech products on the market or in development (cf. http://www.bio.org/speeches/pubs/er/agrLproducts.asp). Genetically modified plants are plants, which genetic material has been so modified by the use of recombinant DNA techniques that under natural circumstances cannot readily be obtained by cross breeding, mutations or natural recombination. Typically, one or more genes have been integrated into the genetic material of a genetically modified plant in order to improve certain properties of the plant. Such genetic modifications also include but are not limited to targeted post-translational modification of protein(s), oligo- or polypeptides e. g. by glycosylation or polymer additions such as prenylated, acetylated or farnesylated moieties or PEG moieties.

Plants that have been modified by breeding, mutagenesis or genetic engineering, e. g. have been rendered tolerant to applications of specific classes of herbicides, such as hydroxyphenylpyruvate dioxygenase (HPPD) inhibitors; acetolactate synthase (ALS) inhibitors, such as sulfonyl ureas (see e. g. US 6,222,100, WO 01/82685, WO 00/26390, WO 97/41218, WO 98/02526, WO 98/02527, WO 04/106529, WO 05/20673, WO 03/14357, WO 03/13225, WO 03/14356, WO 04/16073) or imida- zolinones (see e. g. US 6,222,100, WO 01/82685, WO 00/026390, WO 97/41218, WO 98/002526, WO 98/02527, WO 04/106529, WO 05/20673, WO 03/014357, WO 03/13225, WO 03/14356, WO 04/16073); enolpyruvylshikimate-3-phosphate synthase (EPSPS) inhibitors, such as glyphosate (see e. g. WO 92/00377); glutamine synthetase (GS) inhibitors, such as glufosinate (see e.g. EP-A 242 236, EP-A 242 246) or oxynil herbicides (see e. g. US 5,559,024) as a result of conventional methods of breeding or genetic engineering. Several cultivated plants have been rendered tolerant to herbicides by conventional methods of breeding (mutagenesis), e. g. Clearfield ^® summer rape (Canola, BASF SE, Germany) being tolerant to imidazolinones, e. g. imazamox. Genetic engineering methods have been used to render cultivated plants, such as soybean, cotton, corn, beets and rape, tolerant to herbicides such as glyphosate and glufosinate, some of which are commercially available under the trade names RoundupReady ^® (glyphosate-tolerant, Monsanto, U.S.A.) and LibertyLink ^® (glufosinate- tolerant, Bayer CropScience, Germany).

Furthermore, plants are also covered that, by the use of recombinant DNA techniques, are capable to synthesize one or more insecticidal proteins, especially those known from the bacterial genus Bacillus, particularly from Bacillus thuringiensis, such as δ-endotoxins, e. g. CrylA(b), CrylA(c), CrylF, CrylF(a2), CryllA(b), CrylllA, CrylllB(bi ) or Cryθc; vegetative insecticidal proteins (VIP), e. g. VIP1 , VIP2, VIP3 or VIP3A; insec- ticidal proteins of bacteria colonizing nematodes, e. g. Photorhabdus spp. or Xenor- habdus spp.; toxins produced by animals, such as scorpion toxins, arachnid toxins, wasp toxins, or other insect-specific neurotoxins; toxins produced by fungi, such Strep- tomycetes toxins, plant lectins, such as pea or barley lectins; agglutinins; proteinase inhibitors, such as trypsin inhibitors, serine protease inhibitors, patatin, cystatin or pa- pain inhibitors; ribosome-inactivating proteins (RIP), such as ricin, maize-RIP, abrin, luffin, saporin or bryodin; steroid metabolism enzymes, such as 3-hydroxysteroid oxidase, ecdysteroid-IDP-glycosyl-transferase, cholesterol oxidases, ecdysone inhibitors or HMG-CoA-reductase; ion channel blockers, such as blockers of sodium or calcium channels; juvenile hormone esterase; diuretic hormone receptors (helicokinin recep- tors); stilben synthase, bibenzyl synthase, chitinases or glucanases. In the context of the present invention these insecticidal proteins or toxins are to be understood expressly also as pre-toxins, hybrid proteins, truncated or otherwise modified proteins. Hybrid proteins are characterized by a new combination of protein domains, (see, e. g. WO 02/015701 ). Further examples of such toxins or genetically modified plants capable of synthesizing such toxins are disclosed, e. g., in EP-A 374 753, WO 93/007278, WO 95/34656, EP-A 427 529, EP-A 451 878, WO 03/18810 und WO 03/52073. The methods for producing such genetically modified plants are generally known to the person skilled in the art and are described, e. g., in the publications mentioned above. These insecticidal proteins contained in the genetically modified plants impart to the plants producing these proteins tolerance to harmful pests from all taxonomic groups of arthropods, especially to beetles (Coleoptera), two-winged insects (Diptera), and moths (Lepidoptera) and to nematodes (Nematoda). Genetically modified plants capable to synthesize one or more insecticidal proteins are, e. g., described in the publications mentioned above, and some of them are commercially available such as YieldGard ^® (corn cultivars producing the CryiAb toxin), YieldGard ^® Plus (corn cultivars producing Cry1 Ab and Cry3Bb1 toxins), Starlink ^® (corn cultivars producing the Cry9c toxin), Her- culex ^® RW (corn cultivars producing Cry34Ab1 , Cry35Ab1 and the enzyme Phosphi- nothricin-N-Acetyltransferase [PAT]); NuCOTN ^® 33B (cotton cultivars producing the Cry1 Ac toxin), Bollgard ^® I (cotton cultivars producing the CryiAc toxin), Bollgard ^® Il (cotton cultivars producing CryiAc and Cry2Ab2 toxins); VIPCOT ^® (cotton cultivars producing a VIP-toxin); NewLeaf ^® (potato cultivars producing the Cry3A toxin); Bt- Xtra ^® , NatureGard ^® , KnockOut ^® , BiteGard ^® , Protecta ^® , Bt 1 1 (e. g. Agrisure ^® CB) and Bt176 from Syngenta Seeds SAS, France, (corn cultivars producing the CryiAb toxin and PAT enyzme), MIR604 from Syngenta Seeds SAS, France (corn cultivars producing a modified version of the Cry3A toxin, c.f. WO 03/018810), MON 863 from Monsanto Europe S.A., Belgium (corn cultivars producing the Cry3Bb1 toxin), IPC 531 from Monsanto Europe S.A., Belgium (cotton cultivars producing a modified version of the CryiAc toxin) and 1507 from Pioneer Overseas Corporation, Belgium (corn cultivars producing the Cry1 F toxin and PAT enzyme).

Furthermore, plants are also covered that, by the use of recombinant DNA techniques, are capable to synthesize one or more proteins to increase the resistance or tolerance of those plants to bacterial, viral or fungal pathogens. Examples of such proteins are the so-called "pathogenesis-related proteins" (PR proteins, see, e. g. EP-A 392 225), plant disease resistance genes (e. g. potato cultivars, which express resistance genes acting against Phytophthora infestans derived from the Mexican wild potato Solanum bulbocastanum) or T4-lysozym (e. g. potato cultivars capable of synthesizing these proteins with increased resistance against bacteria such as Erwinia amylvora). The methods for producing such genetically modified plants are generally known to the person skilled in the art and are described, e. g., in the publications mentioned above.

Furthermore, plants are also covered that, by the use of recombinant DNA techniques, are capable to synthesize one or more proteins to increase the productivity (e. g. bio mass production, grain yield, starch content, oil content or protein content), tolerance to drought, salinity or other growth-limiting environmental factors or tolerance to pests and fungal, bacterial or viral pathogens of those plants.

Furthermore, plants are also covered that, by the use of recombinant DNA techniques, contain a modified amount of substances of content or new substances of content, specifically to improve human or animal nutrition, e. g. oil crops that produce health- promoting long-chain omega-3 fatty acids or unsaturated omega-9 fatty acids (e. g. Nexera ^® rape, DOW Agro Sciences, Canada).

Furthermore, plants are also covered that, by the use of recombinant DNA techniques, contain a modified amount of substances of content or new substances of content, specifically to improve raw material production, e. g. potatoes that produce increased amounts of amylopectin (e. g. Amflora ^® potato, BASF SE, Germany).

The compounds I and Il and compositions thereof, respectively, are particularly suitable for controlling the following plant diseases:

Albugo spp. (white rust) on ornamentals, vegetables (e. g. A. Candida) and sunflowers (e. g. A. tragopogonis); Altemaria spp. (Alternaria leaf spot) on vegetables, rape {A. brassicola or brassicae), sugar beets {A. tenuis), fruits, rice, soybeans, potatoes (e. g. A. solani or A. alternata), tomatoes (e. g. A. solani or A. alternata) and wheat; Aphano- myces spp. on sugar beets and vegetables; Ascochyta spp. on cereals and vegetables, e. g. A. tritici (anthracnose) on wheat and A. hordei on barley; Bipolaris and Drechslera spp. (teleomorph: Cochliobolus spp.), e. g. Southern leaf blight (D. maydis) or Northern leaf blight (β. zeicola) on corn, e. g. spot blotch (β. sorokiniana) on cereals and e.g. B. oryzae on rice and turfs; Blumeria (formerly Erysiphe) graminis (powdery mildew) on cereals (e. g. on wheat or barley); Botrytis cinerea (teleomorph: Botryotinia fuckeliana: grey mold) on fruits and berries (e. g. strawberries), vegetables (e. g. lettuce, carrots, celery and cabbages), rape, flowers, vines, forestry plants and wheat; Bremia lactucae (downy mildew) on lettuce; Ceratocystis (syn. Ophiostoma) spp. (rot or wilt) on broad- leaved trees and evergreens, e. g. C. ulmi (Dutch elm disease) on elms; Cercospora spp. (Cercospora leaf spots) on corn (e.g. Gray leaf spot: C. zeae-maydis), rice, sugar beets (e. g. C. beticola), sugar cane, vegetables, coffee, soybeans (e. g. C. sojina or C. kikuchii) and rice; Cladosporium spp. on tomatoes (e. g. C. fulvum: leaf mold) and cereals, e. g. C. herbarum (black ear) on wheat; Claviceps purpurea (ergot) on cereals; Cochliobolus (anamorph: Helminthosporium of Bipolaris) spp. (leaf spots) on corn (C. carbonum), cereals (e. g. C. sativus, anamorph: B. sorokiniana) and rice (e. g. C. miy- abeanus, anamorph: H. oryzae); Colletotrichum (teleomorph: Glomerella) spp. (an- thracnose) on cotton (e. g. C. gossypii), corn (e. g. C. graminicola: Anthracnose stalk rot), soft fruits, potatoes (e. g. C. coccodes: black dot), beans (e. g. C. lindemuthianum) and soybeans (e. g. C. truncatum or C. gloeosporioides); Corticium spp., e. g. C. sa- sakii (sheath blight) on rice; Corynespora cassiicola (leaf spots) on soybeans and or- namentals; Cycloconium spp., e. g. C. oleaginum on olive trees; Cylindrocarpon spp. (e. g. fruit tree canker or young vine decline, teleomorph: Nectria or Neonectria spp.) on fruit trees, vines (e. g. C. liriodendri, teleomorph: Neonectria liriodendrϊ. Black Foot Disease) and ornamentals; Dematophora (teleomorph: Rosellinia) necatrix (root and stem rot) on soybeans; Diaporthe spp., e. g. D. phaseolorum (damping off) on soy- beans; Drechslera (syn. Helminthosporium, teleomorph: Pyrenophora) spp. on corn, cereals, such as barley (e. g. D. teres, net blotch) and wheat (e. g. D. tritici-repentis: tan spot), rice and turf; Esca (dieback, apoplexy) on vines, caused by Formitiporia (syn. Phellinus) punctata, F. mediterranea, Phaeomoniella chlamydospora (earlier Phaeo- acremonium chlamydosporum), Phaeoacremonium aleophilum and/or Botryosphaeria obtusa; Elsinoe spp. on pome fruits (E. pyri), soft fruits (E. veneta: anthracnose) and vines (E ampelina: anthracnose); Entyloma oryzae (leaf smut) on rice; Epicoccum spp. (black mold) on wheat; Erysiphe spp. (powdery mildew) on sugar beets (E. betae), vegetables (e. g. E. pisi), such as cucurbits (e. g. E. cichoracearum), cabbages, rape (e. g. E. cruciferarum); Eutypa lata (Eutypa canker or dieback, anamorph: Cytosporina lata, syn. Libertella blepharis) on fruit trees, vines and ornamental woods; Exserohilum (syn. Helminthosporium) spp. on corn (e. g. E. turcicum); Fusarium (teleomorph: Gib- berella) spp. (wilt, root or stem rot) on various plants, such as F. graminearum or F. culmorum (root rot, scab or head blight) on cereals (e. g. wheat or barley), F. oxy- sporum on tomatoes, F. solani on soybeans and F. verticillioides on corn; Gaeumanno- myces graminis (take-all) on cereals (e. g. wheat or barley) and corn; Gibberella spp. on cereals (e. g. G. zeae) and rice (e. g. G. fujikuroi: Bakanae disease); Glomerella cingulata on vines, pome fruits and other plants and G. gossypii on cotton; Grain- staining complex on rice; Guignardia bidwellii (black rot) on vines; Gymnosporangium spp. on rosaceous plants and junipers, e. g. G. sabinae (rust) on pears; Helmintho- sporium spp. (syn. Drechslera, teleomorph: Cochliobolus) on corn, cereals and rice; Hemileia spp., e. g. H. vastatrix (coffee leaf rust) on coffee; lsariopsis clavispora (syn. Cladosporium vitis) on vines; Macrophomina phaseolina (syn. phaseoli) (root and stem rot) on soybeans and cotton; Microdochium (syn. Fusarium) nivale (pink snow mold) on cereals (e. g. wheat or barley); Microsphaera diffusa (powdery mildew) on soybeans; Monilinia spp., e. g. M. laxa, M. fructicola and M. fructigena (bloom and twig blight, brown rot) on stone fruits and other rosaceous plants; Mycosphaerella spp. on cereals, bananas, soft fruits and ground nuts, such as e. g. M. graminicola (anamorph: Septoria tritici, Septoria blotch) on wheat or M. fijiensis (black Sigatoka disease) on bananas; Peronospora spp. (downy mildew) on cabbage (e. g. P. brassicae), rape (e. g. P. parasitica), onions (e. g. P. destructor), tobacco (P. tabacina) and soybeans (e. g. P. manshurica); Phakopsora pachyrhizi and P. meibomiae (soybean rust) on soybeans; Phialophora spp. e. g. on vines (e. g. P. tracheiphila and P. tetraspora) and soybeans (e. g. P. gregata: stem rot); Phoma lingam (root and stem rot) on rape and cabbage and P. betae (root rot, leaf spot and damping-off) on sugar beets; Phomopsis spp. on sunflowers, vines (e. g. P. viticola: can and leaf spot) and soybeans (e. g. stem rot: P. phaseoli, teleomorph: Diaporthe phaseolorum); Physoderma maydis (brown spots) on corn; Phytophthora spp. (wilt, root, leaf, fruit and stem root) on various plants, such as paprika and cucurbits (e. g. P. capsici), soybeans (e. g. P. megasperma, syn. P. sojae), potatoes and tomatoes (e. g. P. infestans: late blight) and broad-leaved trees (e. g. P. ramorum: sudden oak death); Plasmodiophora brassicae (club root) on cabbage, rape, radish and other plants; Plasmopara spp., e. g. P. viticola (grapevine downy mildew) on vines and P. halstediiou sunflowers; Podosphaera spp. (powdery mildew) on rosaceous plants, hop, pome and soft fruits, e. g. P. leucotricha on apples; Polymyxa spp., e. g. on cereals, such as barley and wheat (P. graminis) and sugar beets (P. betae) and thereby transmitted viral diseases; Pseudocercosporella herpotrichoides (eyespot, teleomorph: Tapesia yallundae) on cereals, e. g. wheat or barley; Pseudoperonospora (downy mildew) on various plants, e. g. P. cubensis on cucurbits or P. humili on hop; Pseudopezicula tracheiphila (red fire disease or , rotbrenner' , anamorph: Phialo- phora) on vines; Puccinia spp. (rusts) on various plants, e. g. P. triticina (brown or leaf rust), P. striiformis (stripe or yellow rust), P. hordei (dwarf rust), P. graminis (stem or black rust) or P. recondita (brown or leaf rust) on cereals, such as e. g. wheat, barley or rye, and asparagus (e. g. P. asparagi); Pyrenophora (anamorph: Drechslera) tritici- repentis (tan spot) on wheat or P. feres (net blotch) on barley; Pyricularia spp., e. g. P. oryzae (teleomorph: Magnaporthe grisea, rice blast) on rice and P. grisea on turf and cereals; Pythium spp. (damping-off) on turf, rice, corn, wheat, cotton, rape, sunflowers, soybeans, sugar beets, vegetables and various other plants (e. g. P. ultimum or P. aphanidermatum); Ramularia spp., e. g. R. collo-cygni (Ra mu Ia ria leaf spots, Physiological leaf spots) on barley and R. beticola on sugar beets; Rhizoctonia spp. on cotton, rice, potatoes, turf, corn, rape, potatoes, sugar beets, vegetables and various other plants, e. g. R. solani (root and stem rot) on soybeans, R. so/an/ (sheath blight) on rice or R. cerealis (Rhizoctonia spring blight) on wheat or barley; Rhizopus stolonifer (black mold, soft rot) on strawberries, carrots, cabbage, vines and tomatoes; Rhynchosporium secalis (scald) on barley, rye and triticale; Sarocladium oryzae and S. attenuatum (sheath rot) on rice; Sclerotinia spp. (stem rot or white mold) on vegetables and field crops, such as rape, sunflowers (e. g. S. sclerotiorum) and soybeans (e. g. S. rolfsii or S. sclerotiorum); Septoria spp. on various plants, e. g. S. glycines (brown spot) on soybeans, S. tritici (Septoria blotch) on wheat and S. (syn. Stagonospora) nodorum (Stagonospora blotch) on cereals; Uncinula (syn. Erysiphe) necator (powdery mildew, anamorph: Oidium tuckeri) on vines; Setospaeria spp. (leaf blight) on corn (e. g. S. turcicum, syn. Helminthosporium turcicum) and turf; Sphacelotheca spp. (smut) on corn, (e. g. S. miliaria: head smut), sorghum und sugar cane; Sphaerotheca fuliginea (powdery mildew) on cucurbits; Spongospora subterranea (powdery scab) on potatoes and thereby transmitted viral diseases; Stagonospora spp. on cereals, e. g. S. nodorum (Stagonospora blotch, teleomorph: Leptosphaeria [syn. Phaeosphaeria] nodorum) on wheat; Synchytrium endobioticum on potatoes (potato wart disease); Taphrina spp., e. g. T. deformans (leaf curl disease) on peaches and T. pruni (plum pocket) on plums; Thielaviopsis spp. (black root rot) on tobacco, pome fruits, vegetables, soybeans and cotton, e. g. T. basicola (syn. Chalara elegans); Tilletia spp. (common bunt or stinking smut) on cereals, such as e. g. T. tritici (syn. T. caries, wheat bunt) and T. controversa (dwarf bunt) on wheat; Typhula incamata (grey snow mold) on barley or wheat; Uro- cystis spp., e. g. U. occulta (stem smut) on rye; Uromyces spp. (rust) on vegetables, such as beans (e. g. U. appendiculatus, syn. U. phaseoli) and sugar beets (e. g. U. betae); Ustilago spp. (loose smut) on cereals (e. g. U. nuda and U. avaenae), corn (e. g. U. maydis: corn smut) and sugar cane; Venturia spp. (scab) on apples (e. g. V. inaequalis) and pears; and Verticillium spp. (wilt) on various plants, such as fruits and ornamentals, vines, soft fruits, vegetables and field crops, e. g. V. dahliae on strawberries, rape, potatoes and tomatoes.

The compounds I and Il and compositions thereof, respectively, are also suitable for controlling harmful fungi in the protection of stored products or harvest and in the protection of materials. The term "protection of materials" is to be understood to denote the protection of technical and non-living materials, such as adhesives, glues, wood, paper and paperboard, textiles, leather, paint dispersions, plastics, colling lubricants, fiber or fabrics, against the infestation and destruction by harmful microorganisms, such as fungi and bacteria. As to the protection of wood and other materials, the particular attention is paid to the following harmful fungi: Ascomycetes such as Ophio- stoma spp., Ceratocysf/s spp., Aureobasidium pullulans, Sclerophoma spp., Chae- tomium spp., Humicola spp., Petriella spp., Trichurus spp.; Basidiomycetes such as

Coniophora spp., Coriolus spp., Gloeophyllum spp., Lentinus spp., Pleurotus spp., Po- ria spp., Serpula spp. and Tyromyces spp., Deuteromycetes such as Aspergillus spp., Cladosporium spp., Penicillium spp., Trichorma spp., Altemaria spp., Paecilomyces spp. and Zygomycetes such as Mucorspp., and in addition in the protection of stored products and harvest the following yeast fungi are worthy of note: Candida spp. and Saccharomyces cerevisae.

The compounds I and Il and compositions thereof, respectively, may be used for impro- ving the health of a plant. The invention also relates to a method for improving plant health by treating a plant, its propagation material and/or the locus where the plant is growing or is to grow with an effective amount of compounds I and/or Il and compositions thereof, respectively.

The term "plant health" is to be understood to denote a condition of the plant and/or its products which is determined by several indicators alone or in combination with each other such as yield (e. g. increased biomass and/or increased content of valuable ingredients), plant vigor [e. g. improved plant growth and/or greener leaves ("greening effect")], quality (e. g. improved content or composition of certain ingredients) and tol- erance to abiotic and/or biotic stress. The above identified indicators for the health condition of a plant may be interdependent or may result from each other.

The compounds of formula I and Il can be present in different crystal modifications whose biological activity may differ. They are likewise subject matter of the present invention.

The compounds I and Il are employed as such or in form of compositions by treating the fungi or the plants, plant propagation materials, such as seeds, soil, surfaces, materials or rooms to be protected from fungal attack with a fungicidally effective amount of the active substances. The application can be carried out both before and after the infection of the plants, plant propagation materials, such as seeds, soil, surfaces, materials or rooms by the fungi.

Plant propagation materials may be treated with compounds I and/or Il as such or a composition comprising at least one compound I and/or Il prophylactically either at or before planting or transplanting.

The invention also relates to agrochemical compositions comprising a solvent or solid carrier and at least one compound I and/or Il and to the use for controlling harmful fungi.

An agrochemical composition comprises a fungicidally effective amount of a compound I and/or II. The term "effective amount" denotes an amount of the composition or of the compounds I and/or II, which is sufficient for controlling harmful fungi on cultivated plants or in the protection of materials and which does not result in a substantial damage to the treated plants. Such an amount can vary in a broad range and is dependent on various factors, such as the fungal species to be controlled, the treated cultivated plant or material, the climatic conditions and the specific compound I used.

The compounds I and/or Il and salts thereof can be converted into customary types of agrochemical compositions, e. g. solutions, emulsions, suspensions, dusts, powders, pastes and granules. The composition type depends on the particular intended purpose; in each case, it should ensure a fine and uniform distribution of the compound according to the invention.

Examples for composition types are suspensions (SC, OD, FS), emulsifiable concentrates (EC), emulsions (EW, EO, ES), pastes, pastilles, wettable powders or dusts (WP, SP, SS, WS, DP, DS) or granules (GR, FG, GG, MG), which can be water- soluble or wettable, as well as gel formulations for the treatment of plant propagation materials such as seeds (GF).

Usually the composition types (e. g. SC, OD, FS, EC, WG, SG, WP, SP, SS, WS, GF) are employed diluted. Composition types such as DP, DS, GR, FG, GG and MG are usually used undiluted.

The compositions are prepared in a known manner (cf. US 3,060,084, EP-A 707 445 (for liquid concentrates), Browning: "Agglomeration", Chemical Engineering, Dec. 4, 1967, 147-48, Perry's Chemical Engineer's Handbook, 4 ^th Ed., McGraw-Hill, New York, 1963, pp. 8-57 et seq., WO 91/13546, US 4,172,714, US 4,144,050, US 3,920,442, US 5,180,587, US 5,232,701 , US 5,208,030, GB 2,095,558, US 3,299,566, Klingman: Weed Control as a Science (J. Wiley & Sons, New York, 1961), Hance et al.: Weed Control Handbook (8 ^th Ed., Blackwell Scientific, Oxford, 1989) and Mollet, H. and Grubemann, A.: Formulation technology (Wiley VCH Verlag, Weinheim, 2001 ).

The agrochemical compositions may also comprise auxiliaries which are customary in agrochemical compositions. The auxiliaries used depend on the particular application form and active substance, respectively.

Examples for suitable auxiliaries are solvents, solid carriers, dispersants or emulsifiers (such as further solubilizers, protective colloids, surfactants and adhesion agents), organic and inorganic thickeners, bactericides, anti-freezing agents, anti-foaming agents, if appropriate colorants and tackifiers or binders (e. g. for seed treatment formulations). Suitable solvents are water, organic solvents such as mineral oil fractions of medium to high boiling point, such as kerosene or diesel oil, furthermore coal tar oils and oils of vegetable or animal origin, aliphatic, cyclic and aromatic hydrocarbons, e.g. toluene, xylene, paraffin, tetrahydronaphthalene, alkylated naphthalenes or their derivatives, alcohols such as methanol, ethanol, propanol, butanol and cyclohexanol, glycols, ketones such as cyclohexanone and gamma-butyrolactone, fatty acid dimethylamides, fatty acids and fatty acid esters and strongly polar solvents, e. g. amines such as N- methylpyrrolidone.

Solid carriers are mineral earths such as silicates, silica gels, talc, kaolins, limestone, lime, chalk, bole, loess, clays, dolomite, diatomaceous earth, calcium sulfate, magnesium sulfate, magnesium oxide, ground synthetic materials, fertilizers, such as, e. g., ammonium sulfate, ammonium phosphate, ammonium nitrate, ureas, and products of vegetable origin, such as cereal meal, tree bark meal, wood meal and nutshell meal, cellulose powders and other solid carriers.

Suitable surfactants (adjuvants, wtters, tackifiers, dispersants or emulsifiers) are alkali metal, alkaline earth metal and ammonium salts of aromatic sulfonic acids, such as ligninsoulfonic acid (Borresperse ^® types, Borregard, Norway) phenolsulfonic acid, naphthalenesulfonic acid (Morwet ^® types, Akzo Nobel, U.S.A.), dibutylnaphthalene- sulfonic acid (Nekal ^® types, BASF, Germany), and fatty acids, alkylsulfonates, alkyl- arylsulfonates, alkyl sulfates, laurylether sulfates, fatty alcohol sulfates, and sulfated hexa-, hepta- and octadecanolates, sulfated fatty alcohol glycol ethers, furthermore condensates of naphthalene or of naphthalenesulfonic acid with phenol and formal- dehyde, polyoxy-ethylene octylphenyl ether, ethoxylated isooctylphenol, octylphenol, nonylphenol, alkylphenyl polyglycol ethers, tributylphenyl polyglycol ether, tristearyl- phenyl polyglycol ether, alkylaryl polyether alcohols, alcohol and fatty alcohol/ethylene oxide condensates, ethoxylated castor oil, polyoxyethylene alkyl ethers, ethoxylated polyoxypropylene, lauryl alcohol polyglycol ether acetal, sorbitol esters, lignin-sulfite waste liquors and proteins, denatured proteins, polysaccharides (e. g. methylcellulose), hydrophobically modified starches, polyvinyl alcohols (Mowiol ^® types, Clariant, Switzerland), polycarboxylates (Sokolan ^® types, BASF, Germany), polyalkoxylates, polyvinyl- amines (Lupasol ^® types, BASF, Germany), polyvinylpyrrolidone and the copolymers therof.

Examples for thickeners (i. e. compounds that impart a modified flowability to compositions, i. e. high viscosity under static conditions and low viscosity during agitation) are polysaccharides and organic and anorganic clays such as Xanthan gum (Kelzan ^® , CP Kelco, U.S.A.), Rhodopol ^® 23 (Rhodia, France), Veegum ^® (RT. Vanderbilt, U.S.A.) or Attaclay ^® (Engelhard Corp., NJ, USA).

Bactericides may be added for preservation and stabilization of the composition. Ex- amples for suitable bactericides are those based on dichlorophene and benzylalcohol hemi formal (Proxel ^® from ICI or Acticide ^® RS from Thor Chemie and Kathon ^® MK from Rohm & Haas) and isothiazolinone derivatives such as alkylisothiazolinones and ben- zisothiazolinones (Acticide ^® MBS from Thor Chemie).

Examples for suitable anti-freezing agents are ethylene glycol, propylene glycol, urea and glycerin.

Examples for anti-foaming agents are silicone emulsions (such as e. g. Silikon ^® SRE, Wacker, Germany or Rhodorsil ^® , Rhodia, France), long chain alcohols, fatty acids, salts of fatty acids, fluoroorganic compounds and mixtures thereof.

Suitable colorants are pigments of low water solubility and water-soluble dyes. Examples to be mentioned und the designations rhodamin B, C. I. pigment red 112, C. I. solvent red 1 , pigment blue 15:4, pigment blue 15:3, pigment blue 15:2, pigment blue 15:1 , pigment blue 80, pigment yellow 1 , pigment yellow 13, pigment red 112, pigment red 48:2, pigment red 48:1 , pigment red 57:1 , pigment red 53:1 , pigment orange 43, pigment orange 34, pigment orange 5, pigment green 36, pigment green 7, pigment white 6, pigment brown 25, basic violet 10, basic violet 49, acid red 51 , acid red 52, acid red 14, acid blue 9, acid yellow 23, basic red 10, basic red 108.

Examples for tackifiers or binders are polyvinylpyrrolidons, polyvinylacetates, polyvinyl alcohols and cellulose ethers (Tylose ^® , Shin-Etsu, Japan).

Powders, materials for spreading and dusts can be prepared by mixing or conco- mitantly grinding the compounds I and, if appropriate, further active substances, with at least one solid carrier.

Granules, e. g. coated granules, impregnated granules and homogeneous granules, can be prepared by binding the active substances to solid carriers. Examples of solid carriers are mineral earths such as silica gels, silicates, talc, kaolin, attaclay, limestone, lime, chalk, bole, loess, clay, dolomite, diatomaceous earth, calcium sulfate, magnesium sulfate, magnesium oxide, ground synthetic materials, fertilizers, such as, e. g., ammonium sulfate, ammonium phosphate, ammonium nitrate, ureas, and products of vegetable origin, such as cereal meal, tree bark meal, wood meal and nutshell meal, cellulose powders and other solid carriers.

Examples for composition types are:

1. Composition types for dilution with water

i) Water-soluble concentrates (SL, LS)

10 parts by weight of a compound I or Il according to the invention are dissolved in 90 parts by weight of water or in a water-soluble solvent. As an alternative, wetting agents or other auxiliaries are added. The active substance dissolves upon dilution with water. In this way, a composition having a content of 10% by weight of active substance is obtained.

ii) Dispersible concentrates (DC)

20 parts by weight of a compound I or Il according to the invention are dissolved in 70 parts by weight of cyclohexanone with addition of 10 parts by weight of a dispersant, e. g. polyvinylpyrrolidone. Dilution with water gives a dispersion. The active substance content is 20% by weight.

iii) Emulsifiable concentrates (EC)

15 parts by weight of a compound I or Il according to the invention are dissolved in 75 parts by weight of xylene with addition of calcium dodecylbenzenesulfonate and castor

011 ethoxylate (in each case 5 parts by weight). Dilution with water gives an emulsion. The composition has an active substance content of 15% by weight.

iv) Emulsions (EW, EO, ES)

25 parts by weight of a compound I or Il according to the invention are dissolved in 35 parts by weight of xylene with addition of calcium dodecylbenzenesulfonate and castor oil ethoxylate (in each case 5 parts by weight). This mixture is introduced into 30 parts by weight of water by means of an emulsifying machine (Ultraturrax) and made into a homogeneous emulsion. Dilution with water gives an emulsion. The composition has an active substance content of 25% by weight.

v) Suspensions (SC, OD, FS)

In an agitated ball mill, 20 parts by weight of a compound I or Il according to the invention are comminuted with addition of 10 parts by weight of dispersants and wetting agents and 70 parts by weight of water or an organic solvent to give a fine active sub- stance suspension. Dilution with water gives a stable suspension of the active substance. The active substance content in the composition is 20% by weight.

vi) Water-dispersible granules and water-soluble granules (WG, SG) 50 parts by weight of a compound I or Il according to the invention are ground finely with addition of 50 parts by weight of dispersants and wetting agents and prepared as water-dispersible or water-soluble granules by means of technical appliances (e. g. extrusion, spray tower, fluidized bed). Dilution with water gives a stable dispersion or solution of the active substance. The composition has an active substance content of 50% by weight.

vii) Water-dispersible powders and water-soluble powders (WP, SP, SS, WS) 75 parts by weight of a compound I or Il according to the invention are ground in a ro- tor-stator mill with addition of 25 parts by weight of dispersants, wetting agents and silica gel. Dilution with water gives a stable dispersion or solution of the active substance. The active substance content of the composition is 75% by weight.

viii) Gel (GF)

In an agitated ball mill, 20 parts by weight of a compound I or Il according to the inven- tion are comminuted with addition of 10 parts by weight of dispersants, 1 part by weight of a gelling agent wetters and 70 parts by weight of water or of an organic solvent to give a fine suspension of the active substance. Dilution with water gives a stable suspension of the active substance, whereby a composition with 20% (w/w) of active substance is obtained.

2. Composition types to be applied undiluted

ix) Dustable powders (DP, DS)

5 parts by weight of a compound I or Il according to the invention are ground finely and mixed intimately with 95 parts by weight of finely divided kaolin. This gives a dustable composition having an active substance content of 5% by weight.

x) Granules (GR, FG, GG, MG)

0.5 parts by weight of a compound I or Il according to the invention is ground finely and associated with 99.5 parts by weight of carriers. Current methods are extrusion, spray- drying or the fluidized bed. This gives granules to be applied undiluted having an active substance content of 0.5% by weight.

xi) ULV solutions (UL) 10 parts by weight of a compound I or Il according to the invention are dissolved in 90 parts by weight of an organic solvent, e. g. xylene. This gives a composition to be applied undiluted having an active substance content of 10% by weight.

The agrochemical compositions generally comprise between 0.01 and 95%, preferably between 0.1 and 90%, most preferably between 0.5 and 90%, by weight of active substance. The active substances are employed in a purity of from 90% to 100%, preferably from 95% to 100% (according to NMR spectrum).

Water-soluble concentrates (LS), flowable concentrates (FS), powders for dry treatment (DS), water-dispersible powders for slurry treatment (WS), water-soluble powders (SS), emulsions (ES) emulsifiable concentrates (EC) and gels (GF) are usually employed for the purposes of treatment of plant propagation materials, particularly seeds. These compositions can be applied to plant propagation materials, particularly seeds, diluted or undiluted. The compositions in question give, after two-to-tenfold dilution, active substance concentrations of from 0.01 to 60% by weight, preferably from 0.1 to 40% by weight, in the ready-to-use preparations. Application can be carried out before or during sowing. Methods for applying or treating agrochemical compounds and compositions thereof, respectively, on to plant propagation material, especially seeds, are known in the art, and include dressing, coating, pelleting, dusting, soaking and in- furrow application methods of the propagation material. In a preferred embodiment, the compounds or the compositions thereof, respectively, are applied on to the plant propagation material by a method such that germination is not induced, e. g. by seed dressing, pelleting, coating and dusting.

In a preferred embodiment, a suspension-type (FS) composition is used for seed treatment. Typcially, a FS composition may comprise 1-800 g/l of active substance, 1-200 g/l Surfactant, 0 to 200 g/l antifreezing agent, 0 to 400 g/l of binder, 0 to 200 g/l of a pigment and up to 1 liter of a solvent, preferably water.

The active substances can be used as such or in the form of their compositions, e. g. in the form of directly sprayable solutions, powders, suspensions, dispersions, emulsions,

011 dispersions, pastes, dustable products, materials for spreading, or granules, by means of spraying, atomizing, dusting, spreading, brushing, immersing or pouring. The application forms depend entirely on the intended purposes; it is intended to ensure in each case the finest possible distribution of the active substances according to the invention. Aqueous application forms can be prepared from emulsion concentrates, pastes or wettable powders (sprayable powders, oil dispersions) by adding water. To prepare emulsions, pastes or oil dispersions, the substances, as such or dissolved in an oil or solvent, can be homogenized in water by means of a wetter, tackifier, dispersant or emulsifier. Alternatively, it is possible to prepare concentrates composed of active substance, wetter, tackifier, dispersant or emulsifier and, if appropriate, solvent or oil, and such concentrates are suitable for dilution with water.

The active substance concentrations in the ready-to-use preparations can be varied within relatively wide ranges. In general, they are from 0.0001 to 10%, preferably from 0.001 to 1 % by weight of active substance.

The active substances may also be used successfully in the ultra-low-volume process (ULV), it being possible to apply compositions comprising over 95% by weight of active substance, or even to apply the active substance without additives.

When employed in plant protection, the amounts of active substances applied are, depending on the kind of effect desired, from 0.001 to 2 kg per ha, preferably from 0.005 to 2 kg per ha, more preferably from 0.05 to 0.9 kg per ha, in particular from 0.1 to 0.75 kg per ha.

In treatment of plant propagation materials such as seeds, e. g. by dusting, coating or drenching seed, amounts of active substance of from 0.1 to 1000 g, preferably from 1 to 1000 g, more preferably from 1 to 100 g and most preferably from 5 to 100 g, per 100 kilogram of plant propagation material (preferably seed) are generally required.

When used in the protection of materials or stored products, the amount of active substance applied depends on the kind of application area and on the desired effect. Amounts customarily applied in the protection of materials are, e. g., 0.001 g to 2 kg, preferably 0.005 g to 1 kg, of active substance per cubic meter of treated material.

Various types of oils, wetters, adjuvants, herbicides, bactericides, other fungicides and/or pesticides may be added to the active substances or the compositions comprising them, if appropriate not until immediately prior to use (tank mix). These agents can be admixed with the compositions according to the invention in a weight ratio of 1 :100 to 100:1 , preferably 1 :10 to 10:1.

Adjuvants which can be used are in particular organic modified polysiloxanes such as Break Thru S 240 ^® ; alcohol alkoxylates such as Atplus 245 ^® , Atplus MBA 1303 ^® , PIu- rafac LF 300 ^® and Lutensol ON 30 ^® ; EO/PO block polymers, e. g. Pluronic RPE 2035 ^® and Genapol B ^® ; alcohol ethoxylates such as Lutensol XP 80 ^® ; and dioctyl sulfosucci- nate sodium such as Leophen RA ^® .

The compositions according to the invention can, in the use form as fungicides, also be present together with other active substances, e. g. with herbicides, insecticides, growth regulators, fungicides or else with fertilizers, as pre-mix or, if appropriate, not until immediately prior to use (tank mix).

Mixing the compounds I and/or Il or the compositions comprising them in the use form as fungicides with other fungicides results in many cases in an expansion of the fungicidal spectrum of activity being obtained or in a prevention of fungicide resistance development. Furthermore, in many cases, synergistic effects are obtained.

The following list of active substances, in conjunction with which the compounds according to the invention can be used, is intended to illustrate the possible combinations but does not limit them:

A) strobilurins azoxystrobin, dimoxystrobin, enestroburin, fluoxastrobin, kresoxim-methyl, meto- minostrobin, orysastrobin, picoxystrobin, pyraclostrobin, pyribencarb, triflox- ystrobin, 2-(2-(6-(3-chloro-2-methyl-phenoxy)-5-fluoro-pyrimidin-4-ylo xy)-phenyl)- 2-methoxyimino-N-methyl-acetamide, 3-methoxy-2-(2-(N-(4-methoxy-phenyl)- cyclopropane-carboximidoylsulfanylmethyl)-phenyl)-acrylic acid methyl ester, methyl (2-chloro-5-[1-(3-methylbenzyloxyimino)ethyl]benzyl)carbamat e and 2-(2-

(3-(2,6-dichlorophenyl)-1-methyl-allylideneaminooxymethyl )-phenyl)-2- methoxyimino-N-methyl-acetamide;

B) carboxamides carboxanilides: benalaxyl, benalaxyl-M, benodanil, bixafen, boscalid, carboxin, fenfuram, fenhexamid, flutolanil, furametpyr, isopyrazam, isotianil, kiralaxyl, me- pronil, metalaxyl, metalaxyl-M (mefenoxam), ofurace, oxadixyl, oxycarboxin, pen- thiopyrad, sedaxane, tecloftalam, thifluzamide, tiadinil, 2-amino-4-methyl- thiazole-5-carboxanilide, 2-chloro-N-(1 ,1 ,3-trimethyl-indan-4-yl)-nicotinamide, N- (3',4',5'-trifluorobiphenyl-2-yl)-3-difluoromethyl-1-methyl- 1 H-pyrazole- 4-carboxamide, N-(4'-trifluoromethylthiobiphenyl-2-yl)-3-difluoromethyl-1 -methyl-

1 H-pyrazole-4-carboxamide, N-(2-(1 ,3-dimethyl-butyl)-phenyl)-1 ,3-dimethyl-5- fluoro-1 H-pyrazole-4-carboxamide and N-(2-(1 ,3,3-trimethyl-butyl)-phenyl)-1 ,3- dimethyl-5-fluoro-1 H-pyrazole-4-carboxamide; carboxylic morpholides: dimethomorph, flumorph, pyrimorph; benzoic acid amides: flumetover, fluopicolide, fluopyram, zoxamide, N-(3-Ethyl- 3,5,5-trimethyl-cyclohexyl)-3-formylamino-2-hydroxy-benzamid e; other carboxamides: carpropamid, dicyclomet, mandiproamid, oxytetracyclin, silthiofarm and N-(6-methoxy-pyτidin-3-yl) cyclopropanecarboxylic acid amide; C) azoles triazoles: azaconazole, bitertanol, bromuconazole, cyproconazole, difenocona- zole, diniconazole, diniconazole-M, epoxiconazole, fenbuconazole, fluquincona- zole, flusilazole, flutriafol, hexaconazole, imibenconazole, ipconazole, metcona- zole, myclobutanil, oxpoconazole, paclobutrazole, penconazole, propiconazole, prothioconazole, simeconazole, tebuconazole, tetraconazole, triadimefon, triadi- menol, triticonazole, uniconazole, 1-(4-chloro-phenyl)-2-([1 ,2,4]triazol-1-yl)- cycloheptanol; imidazoles: cyazofamid, imazalil, pefurazoate, prochloraz, triflumizol; benzimidazoles: benomyl, carbendazim, fuberidazole, thiabendazole; - others: ethaboxam, etridiazole, hymexazole and 2-(4-chloro-phenyl)-N-[4-(3,4-di- methoxy-phenyl)-isoxazol-5-yl]-2-prop-2-ynyloxy-acetamide; D) heterocyclic compounds pyridines: fluazinam, pyrifenox, 3-[5-(4-chloro-phenyl)-2,3-dimethyl-isoxazolidin- 3-yl]-pyridine, 3-[5-(4-methyl-phenyl)-2,3-dimethyl-isoxazolidin-3-yl]-pyrid ine, 2,3,5,6-tetra-chloro-4-methanesulfonyl-pyridine, 3,4,5-trichloropyridine-2,6-di- carbonitrile, N-(1-(5-bromo-3-chloro-pyridin-2-yl)-ethyl)-2,4-dichloronico tinamide, N-[(5-bromo-3-chloro-pyridin-2-yl)-methyl]-2,4-dichloro-nico tinamide; pyrimidines: bupirimate, cyprodinil, diflumetorim, fenarimol, ferimzone, mepani- pyrim, nitrapyrin, nuarimol, pyrimethanil; - piperazines: triforine; pyrroles: fenpiclonil, fludioxonil; morpholines: aldimorph, dodemorph, dodemorph-acetate, fenpropimorph, tride- morph; piperidines: fenpropidin; - dicarboximides: fluoroimid, iprodione, procymidone, vinclozolin; non-aromatic 5-membered heterocycles: famoxadone, fenamidone, flutianil, oc- thilinone, probenazole, 5-amino-2-isopropyl-3-oxo-4-ortho-tolyl-2,3-dihydro- pyrazole-1-carbothioic acid S-allyl ester; others: acibenzolar-S-methyl, amisulbrom, anilazin, blasticidin-S, captafol, cap- tan, chinomethionat, dazomet, debacarb, diclomezine, difenzoquat, difenzoquat- methylsulfate, fenoxanil, Folpet, oxolinic acid, piperalin, proquinazid, pyroquilon, quinoxyfen, triazoxide, tricyclazole, 2-butoxy-6-iodo-3-propylchromen-4-one, 5- chloro-1 -(4,6-dimethoxy-pyrimidin-2-yl)-2-methyl-1 H-benzoimidazole, 5-chloro- 7-(4-methylpiperidin-1 -yl)-6-(2,4,6-trifluorophenyl)-[1 ,2,4]triazolo[1 ,5-a]pyrimidine and 5-ethyl-6-octyl-[1 ,2,4]triazolo[1 ,5-a]pyrimidine-7-ylamine;

E) carbamates thio- and dithiocarbamates: ferbam, mancozeb, maneb, metam, methasulpho- carb, metiram, propineb, thiram, zineb, ziram; carbamates: benthiavalicarb, diethofencarb, iprovalicarb, propamocarb, propamo- carb hydrochlorid, valiphenal and N-(1-(1-(4-cyano-phenyl)ethanesulfonyl)-but-2- yl) carbamic acid-(4-fluorophenyl) ester;

F) other active substances - guanidines: guanidine, dodine, dodine free base, guazatine, guazatine-acetate, iminoctadine, iminoctadine-triacetate, iminoctadine-tris(albesilate); antibiotics: kasugamycin, kasugamycin hydrochloride-hydrate, streptomycin, pol- yoxine, validamycin A; nitrophenyl derivates: binapacryl, dinobuton, dinocap, nitrthal-isopropyl, tecna- zen, organometal compounds: fentin salts, such as fentin-acetate, fentin chloride or fentin hydroxide; sulfur-containing heterocyclyl compounds: dithianon, isoprothiolane; organophosphorus compounds: edifenphos, fosetyl, fosetyl-aluminum, iproben- fos, phosphorous acid and its salts, pyrazophos, tolclofos-methyl; organochlorine compounds: chlorothalonil, dichlofluanid, dichlorophen, flusul- famide, hexachlorobenzene, pencycuron, pentachlorphenole and its salts, phthalide, quintozene, thiophanate-methyl, tolylfluanid, N-(4-chloro-2-nitro- phenyl)-N-ethyl-4-methyl-benzenesulfonamide; - inorganic active substances: Bordeaux mixture, copper acetate, copper hydroxide, copper oxychloride, basic copper sulfate, sulfur; others: biphenyl, bronopol, cyflufenamid, cymoxanil, diphenylamin, metrafenone, mildiomycin, oxin-copper, prohexadione-calcium, spiroxamine, tolylfluanid, N- (cyclopropylmethoxyimino-(6-difluoro-methoxy-2,3-difluoro-ph enyl)-methyl)-2- phenyl acetamide, N'-(4-(4-chloro-3-trifluoromethyl-phenoxy)-2,5-dimethyl- phenyl)-N-ethyl-N-methyl formamidine, N'-(4-(4-fluoro-3-trifluoromethyl-phenoxy)- 2,5-dimethyl-phenyl)-N-ethyl-N-methyl formamidine, N'-(2-methyl-5- trifluoromethyl-4-(3-trimethylsilanyl-propoxy)-phenyl)-N-eth yl-N-methyl formamidine, N'-(5-difluoromethyl-2-methyl-4-(3-trimethylsilanyl-propoxy) -phenyl)-N- ethyl-N-methyl formamidine,

2-{1-[2-(5-methyl-3-trifluoromethyl-pyrazole-1-yl)-acetyl ]-piperidin-4-yl}-thiazole-4- carboxylic acid methyl-(1 ,2,3,4-tetrahydro-naphthalen-1-yl)-amide, 2-{1-[2-(5- methyl-S-trifluoromethyl-pyrazole-i-yO-acety^-piperidin^-ylJ -thiazole^-carboxylic acid methyl-(R)-1 ,2,3,4-tetrahydro-naphthalen-1-yl-amide, acetic acid 6-tert-butyl- 8-fluoro-2,3-dimethyl-quinolin-4-yl ester and methoxy-acetic acid 6-tert-butyl-8- fluoro-2,3-dimethyl-quinolin-4-yl ester. G) growth regulators abscisic acid, amidochlor, ancymidol, 6-benzylaminopurine, brassinolide, butralin, chlormequat (chlormequat chloride), choline chloride, cyclanilide, daminozide, dikegulac, dimethipin, 2,6-dimethylpuridine, ethephon, flumetralin, flurprimidol, fluthiacet, forchlorfenuron, gibberellic acid, inabenfide, indole-3-acetic acid , maleic hydrazide, mefluidide, mepiquat (mepiquat chloride), naphthaleneacetic acid, N-6-benzyladenine, paclobutrazol, prohexadione (prohexadione-calcium), prohydrojasmon, thidiazuron, triapenthenol, tributyl phosphorotrithioate,

2,3,5-tri-iodobenzoic acid , trinexapac-ethyl and uniconazole; H) herbicides acetamides: acetochlor, alachlor, butachlor, dimethachlor, dimethenamid, flufen- acet, mefenacet, metolachlor, metazachlor, napropamide, naproanilide, pethox- amid, pretilachlor, propachlor, thenylchlor; amino acid derivatives: bilanafos, glyphosate, glufosinate, sulfosate; aryloxyphenoxypropionates: clodinafop, cyhalofop-butyl, fenoxaprop, fluazifop, haloxyfop, metamifop, propaquizafop, quizalofop, quizalofop-P-tefuryl;

Bipyridyls: diquat, paraquat; - (thio)carbamates: asulam, butylate, carbetamide, desmedipham, dimepiperate, eptam (EPTC), esprocarb, molinate, orbencarb, phenmedipham, prosulfocarb, pyributicarb, thiobencarb, triallate; cyclohexanediones: butroxydim, clethodim, cycloxydim, profoxydim, sethoxydim, tepraloxydim, tralkoxydim; - dinitroanilines: benfluralin, ethalfluralin, oryzalin, pendimethalin, prodiamine, triflu- ralin; diphenyl ethers: acifluorfen, aclonifen, bifenox, diclofop, ethoxyfen, fomesafen, lactofen, oxyfluorfen; hydroxybenzonitriles: bomoxynil, dichlobenil, ioxynil; - imidazolinones: imazamethabenz, imazamox, imazapic, imazapyr, imazaquin, imazethapyr; phenoxy acetic acids: clomeprop, 2,4-dichlorophenoxyacetic acid (2,4-D), 2,4-

DB, dichlorprop, MCPA, MCPA-thioethyl, MCPB, Mecoprop; pyrazines: chloridazon, flufenpyr-ethyl, fluthiacet, norflurazon, pyridate; - pyridines: aminopyralid, clopyralid, diflufenican, dithiopyr, fluridone, fluroxypyr, picloram, picolinafen, thiazopyr; sulfonyl ureas: amidosulfuron, azimsulfuron, bensulfuron, chlorimuron-ethyl, chlorsulfuron, cinosulfuron, cyclosulfamuron, ethoxysulfuron, flazasulfuron, fluce- tosulfuron, flupyrsulfuron, foramsulfuron, halosulfuron, imazosulfuron, iodosulfu- ron, mesosulfuron, metsulfuron-methyl, nicosulfuron, oxasulfuron, primisulfuron, prosulfuron, pyrazosulfuron, rimsulfuron, sulfometuron, sulfosulfuron, thifensulfu- ron, triasulfuron, tribenuron, trifloxysulfuron, triflusulfuron, tritosulfuron, 1-((2- chloro-6-propyl-imidazo[1 ,2-b]pyridazin-3-yl)sulfonyl)-3-(4,6-dimethoxy-pyπmidin- 2-yl)urea; triazines: ametryn, atrazine, cyanazine, dimethametryn, ethiozin, hexazinone, metamitron, metribuzin, prometryn, simazine, terbuthylazine, terbutryn, triaziflam; ureas: chlorotoluron, daimuron, diuron, fluometuron, isoproturon, linuron, metha- benzthiazuron,tebuthiuron; - other acetolactate synthase inhibitors: bispyribac-sodium, cloransulam-methyl, diclosulam, florasulam, flucarbazone, flumetsulam, metosulam, ortho-sulfamuron, penoxsulam, propoxycarbazone, pyribambenz-propyl, pyribenzoxim, pyriftalid, pyriminobac-methyl, pyrimisulfan, pyrithiobac, pyroxasulfone, pyroxsulam; others: amicarbazone, aminotriazole, anilofos, beflubutamid, benazolin, bencar- bazone,benfluresate, benzofenap, bentazone, benzobicyclon, bromacil, bromo- butide, butafenacil, butamifos, cafenstrole, carfentrazone, cinidon-ethlyl, chlor- thal, cinmethylin, clomazone, cumyluron, cyprosulfamide, dicamba, difenzoquat, diflufenzopyr, Drechslera monoceras, endothal, ethofumesate, etobenzanid, fen- trazamide, flumiclorac-pentyl, flumioxazin, flupoxam, flurochloridone, flurtamone, indanofan, isoxaben, isoxaflutole, lenacil, propanil, propyzamide, quinclorac, quinmerac, mesotrione, methyl arsonic acid, naptalam, oxadiargyl, oxadiazon, oxaziclomefone, pentoxazone, pinoxaden, pyraclonil, pyraflufen-ethyl, pyrasulfo- tole, pyrazoxyfen, pyrazolynate, quinoclamine, saflufenacil, sulcotrione, sulfentra- zone, terbacil, tefuryltrione, tembotrione, thiencarbazone, topramezone, 4- hydroxy-3-[2-(2-methoxy-ethoxymethyl)-6-trifluoromethyl-pyri dine-3-carbonyl]- bicyclo[3.2.1]oct-3-en-2-one, (3-[2-chloro-4-fluoro-5-(3-methyl-2,6-dioxo-4- trifluoromethyl-3,6-dihydro-2H-pyrimidin-1-yl)-phenoxy]-pyri din-2-yloxy)-acetic a- cid ethyl ester, 6-amino-5-chloro-2-cyclopropyl-pyrimidine-4-carboxylic acid methyl ester, 6-chloro-3-(2-cyclopropyl-6-methyl-phenoxy)-pyridazin-4-ol, 4- amino-3-chloro-6-(4-chloro-phenyl)-5-fluoro-pyridine-2-carbo xylic acid, 4-amino-

3-chloro-6-(4-chloro-2-fluoro-3-methoxy-phenyl)-pyridine- 2-carboxylic acid methyl ester, and 4-amino-3-chloro-6-(4-chloro-3-dimethylamino-2-fluoro-phenyl )- pyridine-2-carboxylic acid methyl ester. I) insecticides - organo(thio)phosphates: acephate, azamethiphos, azinphos-methyl, chlorpyrifos, chlorpyrifos-methyl, chlorfenvinphos, diazinon, dichlorvos, dicrotophos, dimethoa- te, disulfoton, ethion, fenitrothion, fenthion, isoxathion, malathion, methamido- phos, methidathion, methyl-parathion, mevinphos, monocrotophos, oxydemeton- methyl, paraoxon, parathion, phenthoate, phosalone, phosmet, phosphamidon, phorate, phoxim, pirimiphos-methyl, profenofos, prothiofos, sulprophos, tetra- chlorvinphos, terbufos, triazophos, trichlorfon; carbamates: alanycarb, aldicarb, bendiocarb, benfuracarb, carbaryl, carbofuran, carbosulfan, fenoxycarb, furathiocarb, methiocarb, methomyl, oxamyl, pirimicarb, propoxur, thiodicarb, triazamate; pyrethroids: allethrin, bifenthrin, cyfluthrin, cyhalothrin, cyphenothrin, cyperme- thrin, alpha-cypermethrin, beta-cypermethrin, zeta-cypermethrin, deltamethrin, esfenvalerate, etofenprox, fenpropathrin, fenvalerate, imiprothrin, lambda- cyhalothrin, permethrin, prallethrin, pyrethrin I and II, resmethrin, silafluofen, tau- fluvalinate, tefluthrin, tetramethrin, tralomethrin, transfluthrin, profluthrin, dimeflu- thrin; insect growth regulators: a) chitin synthesis inhibitors: benzoylureas: chlorfluazu- ron, cyramazin, diflubenzuron, flucycloxuron, flufenoxuron, hexaflumuron, lufenu- ron, novaluron, teflubenzuron, triflumuron; buprofezin, diofenolan, hexythiazox, etoxazole, clofentazine; b) ecdysone antagonists: halofenozide, methoxyfenozi- de, tebufenozide, azadirachtin; c) juvenoids: pyriproxyfen, methoprene, fenoxycarb; d) lipid biosynthesis inhibitors: spirodiclofen, spiromesifen, spirotetramat; nicotinic receptor agonists/antagonists compounds: clothianidin, dinotefuran, imi- dacloprid, thiamethoxam, nitenpyram, acetamiprid, thiacloprid, 1-(2-chloro- thiazol-5-ylmethyl)-2-nitrimino-3,5-dimethyl-[1 ,3,5]triazinane;

GABA antagonist compounds: endosulfan, ethiprole, fipronil, vaniliprole, pyraflu- prole, pyriprole, 5-amino-1 -(2,6-dichloro-4-methyl-phenyl)-4-sulfinamoyl-

1 H-pyrazole-3-carbothioic acid amide; macrocyclic lactone insecticides: abamectin, emamectin, milbemectin, lepimectin, spinosad, spinetoram; mitochondrial electron transport inhibitor (METI) I acaricides: fenazaquin, pyrida- ben, tebufenpyrad, tolfenpyrad, flufenerim;

METI Il and III compounds: acequinocyl, fluacyprim, hydramethylnon; Uncouplers: chlorfenapyr; - oxidative phosphorylation inhibitors: cyhexatin, diafenthiuron, fenbutatin oxide, propargite; moulting disruptor compounds: cryomazine; mixed function oxidase inhibitors: piperonyl butoxide; sodium channel blockers: indoxacarb, metaflumizone; - others: benclothiaz, bifenazate, cartap, flonicamid, pyridalyl, pymetrozine, sulfur, thiocyclam, flubendiamide, chlorantraniliprole, cyazypyr (HGW86), cyenopyrafen, flupyrazofos, cyflumetofen, amidoflumet, imicyafos, bistrifluron, and pyrifluquina- zon. The present invention furthermore relates to agrochemical compositions comprising a mixture of at least one compound I and/or Il (component 1 ) and at least one further active substance useful for plant protection, e. g. selected from the groups A) to I) (component 2), in particular one further fungicide, e. g. one or more fungicide from the groups A) to F), as described above, and if desired one suitable solvent or solid carrier. Those mixtures are of particular interest, since many of them at the same application rate show higher efficiencies against harmful fungi. Furthermore, combating harmful fungi with a mixture of compounds I and/or Il and at least one fungicide from groups A) to F), as described above, is more efficient than combating those fungi with individual compounds I or Il or individual fungicides from groups A) to F). By applying compounds

1 and/or Il together with at least one active substance from groups A) to I) a synergistic effect can be obtained, i.e. more then simple addition of the individual effects is obtained (synergistic mixtures).

According to this invention, applying the compounds I and/or Il together with at least one further active substance is to be understood to denote that at least one compound of formula I and/or Il and at least one further active substance occur simultaneously at the site of action (i.e. the harmful fungi to be controlled or their habitats such as infected plants, plant propagation materials, particularly seeds, surfaces, materials or the soil as well as plants, plant propagation materials, particularly seeds, soil, surfaces, materials or rooms to be protected from fungal attack) in a fungicidally effective amount. This can be obtained by applying the compounds I and/or Il and at least one further active substance simultaneously, either jointly (e. g. as tank-mix) or sperately, or in succession, wherein the time interval between the individual applications is selected to ensure that the active substance applied first still occurs at the site of action in a sufficient amount at the time of application of the further active substance(s). The order of application is not essential for working of the present invention.

In binary mixtures, i.e. compositions according to the invention comprising one com- pound I or Il (component 1 ) and one further active substance (component 2), e. g. one active substance from groups A) to I), the weight ratio of component 1 and component

2 generally depends from the properties of the active substances used, usually it is in the range of from 1 :100 to 100:1 , regularly in the range of from 1 :50 to 50:1 , preferably in the range of from 1 :20 to 20:1 , more preferably in the range of from 1 :10 to 10:1 and in particular in the range of from 1 :3 to 3:1.

In ternary mixtures, i.e. compositions according to the invention comprising one compound I (component 1 ) and a first further active substance (component 2) and a second further active substance (component 3), e. g. two active substances from groups A) to I), the weight ratio of component 1 and component 2 depends from the properties of the active substances used, preferably it is in the range of from 1 :50 to 50:1 and particularly in the range of from 1 :10 to 10:1 , and the weight ratio of component 1 and component 3 preferably is in the range of from 1 :50 to 50:1 and particularly in the range of from 1 :10 to 10:1.

The components can be used individually or already partially or completely mixed with one another to prepare the composition according to the invention. It is also possible for them to be packaged and used further as combination composition such as a kit of parts.

In one embodiment of the invention, the kits may include one or more, including all, components that may be used to prepare a subject agrochemical composition. E. g., kits may include one or more fungicide component(s) and/or an adjuvant component and/or an insecticide component and/or a growth regulator component and/or a her- bicde. One or more of the components may already be combined together or pre- formulated. In those embodiments where more than two components are provided in a kit, the components may already be combined together and as such are packaged in a single container such as a vial, bottle, can, pouch, bag or canister. In other embodi- ments, two or more components of a kit may be packaged separately, i. e., not pre- formulated. As such, kits may include one or more separate containers such as vials, cans, bottles, pouches, bags or canisters, each container containing a separate component for an agrochemical composition. In both forms, a component of the kit may be applied separately from or together with the further components or as a component of a combination composition according to the invention for preparing the composition according to the invention.

The user applies the composition according to the invention usually from a predosage device, a knapsack sprayer, a spray tank or a spray plane. Here, the agrochemical composition is made up with water and/or buffer to the desired application concentration, it being possible, if appropriate, to add further auxiliaries, and the ready-to-use spray liquor or the agrochemical composition according to the invention is thus obtained. Usually, 50 to 500 liters of the ready-to-use spray liquor are applied per hectare of agricultural useful area, preferably 100 to 400 liters.

According to one embodiment, individual components of the composition according to the invention such as parts of a kit or parts of a binary or ternary mixture may be mixed by the user himself in a spray tank and further auxiliaries may be added, if appropriate (tank mix). In a further embodiment, either individual components of the composition according to the invention or partially premixed components, e. g. components comprising compounds I and/or Il and/or active substances from the groups A) to I), may be mixed by the user in a spray tank and further auxiliaries and additives may be added, if appropriate (tank mix).

In a further embodiment, either individual components of the composition according to the invention or partially premixed components, e. g. components comprising com- pounds I and/or Il and/or active substances from the groups A) to I), can be applied jointly (e. .g. after tankmix) or consecutively.

Preference is also given to mixtures comprising a compound I and/or Il (component 1 ) and at least one active substance selected from the strobilurines of group A) (compo- nent 2) and particularly selected from azoxystrobin, dimoxystrobin, fluoxastrobin, kresoxim-methyl, orysastrobin, picoxystrobin, pyraclostrobin and trifloxystrobin.

Preference is also given to mixtures comprising a compound I and/or Il (component 1 ) and at least one active substance selected from the carboxamides of group B) (com- ponent 2) and particularly selected from bixafen, boscalid, sedaxane, fenhexamid, metalaxyl, isopyrazam, mefenoxam, ofurace, dimethomorph, flumorph, fluopicolid (pi- cobenzamid), zoxamide, carpropamid, mandipropamid and N-(3',4',5'-trifluorobiphenyl- 2-yl)-3-difluoromethyl-1 -methyl-1 H-pyrazole-4-carboxamide.

Preference is given to mixtures comprising a compound of formula I and/or Il (component 1 ) and at least one active substance selected from the azoles of group C) (component 2) and particularly selected from cyproconazole, difenoconazole, epoxicona- zole, fluquinconazole, flusilazole, flutriafol, metconazole, myclobutanil, penconazole, propiconazole, prothioconazole, triadimefon, triadimenol, tebuconazole, tetraconazole, triticonazole, prochloraz, cyazofamid, benomyl, carbendazim and ethaboxam.

Preference is also given to mixtures comprising a compound I and/or Il (component 1 ) and at least one active substance selected from the heterocyclic compounds of group D) (component 2) and particularly selected from fluazinam, cyprodinil, fenarimol, me- panipyrim, pyrimethanil, triforine, fludioxonil, dodemorph, fenpropimorph, tridemorph, fenpropidin, iprodione, vinclozolin, famoxadone, fenamidone, probenazole, proquina- zid, acibenzolar-S-methyl, captafol, folpet, fenoxanil, quinoxyfen and 5-ethyl-6-octyl- [1 ,2,4]triazolo[1 ,5-a]pyrimidine-7-ylamine. Preference is also given to mixtures comprising a compound I and/or Il (component 1 ) and at least one active substance selected from the carbamates of group E) (component 2) and particularly selected from mancozeb, metiram, propineb, thiram, iprovali- carb, benthiavalicarb and propamocarb.

Preference is also given to mixtures comprising a compound I and/or Il (component 1 ) and at least one active substance selected from the fungicides given in group F) (component 2) and particularly selected from dithianon, fentin salts, such as fentin acetate, fosetyl, fosetyl-aluminium, H3PO3 and salts thereof, chlorthalonil, dichlofluanid, thio- phanat-methyl, copper acetate, copper hydroxide, copper oxychloride, copper sulfate, sulfur, cymoxanil, metrafenone and spiroxamine.

Accordingly, the present invention furthermore relates to compositions comprising one compound I and/or Il (component 1 ) and one further active substance (component 2), which further active substance is selected from the column "Component 2" of the lines B-1 to B-346 of Table B.

A further embodiment relates to the compositions B-1 to B-346 listed in Table B, where a row of Table B corresponds in each case to a fungicidal composition comprising one of the in the present specification individualized compounds of formula I or Il (component 1 ) and the respective further active substance from groups A) to I) (component 2) stated in the row in question. Preferably, the compositions described comprise the active substances in synergistically effective amounts.

Table B: Composition comprising one indiviualized compound I or Il and one further active substance from groups A) to I)

The active substances referred to as component 2, their preparation and their activity against harmful fungi is known (cf.: http://www.alanwood.net/pesticides/); these substances are commercially available. The compounds described by IUPAC nomencla- ture, their preparation and their fungicidal activity are also known (cf. Can. J. Plant Sci. 48(6), 587-94, 1968; EP-A 141 317; EP-A 152 031 ; EP-A 226 917; EP-A 243 970; EP-A 256 503; EP-A 428 941 ; EP-A 532 022; EP-A 1 028 125; EP-A 1 035 122; EP-A 1 201 648; EP-A 1 122 244, JP 2002316902; DE 19650197; DE 10021412; DE 102005009458; US 3,296,272; US 3,325,503; WO 98/46608; WO 99/14187; WO 99/24413; WO 99/27783; WO 00/29404; WO 00/46148; WO 00/65913; WO 01/54501 ; WO 01/56358; WO 02/22583; WO 02/40431 ; WO 03/10149; WO 03/1 1853; WO 03/14103; WO 03/16286; WO 03/53145; WO 03/61388; WO 03/66609; WO 03/74491 ; WO 04/49804; WO 04/83193; WO 05/120234; WO 05/123689; WO 05/123690; WO 05/63721 ; WO 05/87772; WO 05/87773; WO 06/15866; WO 06/87325; WO 06/87343; WO 07/82098; WO 07/90624).

The mixtures of active substances can be prepared as compositions comprising besides the active ingredients at least one inert ingredient by usual means, e. g. by the means given for the compositions of compounds I and/or II.

Concerning usual ingredients of such compositions reference is made to the explanations given for the compositions containing compounds I and/or II.

The mixtures of active substances according to the present invention are suitable as fungicides, as are the compounds of formula I and II. They are distinguished by an outstanding effectiveness against a broad spectrum of phytopathogenic fungi, especially from the classes of the Ascomycetes, Basidiomycetes, Deuteromycetes and Perono- sporomycetes (syn. Oomycetes ). In addition, it is referred to the explanations regarding the fungicidal activity of the compounds and the compositions containing com- pounds I and/or Il respectively.

The compounds I, Il and IV and pharmaceutically acceptable salts thereof are also suitable for treating diseases in men and animals, especially as antimycotics, for treat- ing cancer and for treating virus infections. The term "antimycotic", as distinguished from the term "fungicide", refers to a medicament for combating zoopathogenic or hu- manpathogenic fungi, i.e. for combating fungi in animals, especially in mammals (including humans) and birds.

Thus, a further aspect of the present invention relates to a medicament comprising at least one compound of the formulae I, Il and/or IV and/or at least one pharmaceutically acceptable salt thereof and a pharmaceutically acceptable carrier.

Suitable pharmaceutically acceptable salts are especially physiologically tolerated salts of the compound I, Il and/or IV, in particular the acid addition salts with physiologically acceptable acids. Examples of suitable organic and inorganic acids are hydrochloric acid, hydrobromic acid, phosphoric acid, sulfuric acid, Ci-C4-alkylsulfonic acids, such as methanesulfonic acid, aromatic sulfonic acids, such as benzenesulfonic acid and toluenesulfonic acid, oxalic acid, maleic acid, fumaric acid, lactic acid, tartaric acid, adipic acid and benzoic acid. Further suitable acids are described, for example, in Fortschritte der Arzneimittelforschung, Volume 10, pages 224 ff., Birkhauser Verlag, Basle and Stuttgart, 1966, the entire contents of which is expressly incorporated herein by way of reference.

Suitable carriers are, for example, solvents, carriers, excipients, binders and the like customarily used for pharmaceutical formulations, which are described below in an exemplary manner for individual types of administration.

A further aspect of the present invention relates to the use of compounds I, Il and IV or of pharmaceutically acceptable salts thereof for preparing an antimycotic medicament; i.e. for preparing a medicament for the treatment and/or prophylaxis of infections with humanpathogenic and/or zoopathogenic fungi. Another aspect of the present invention relates to the use of compounds of formulae I, Il and/or IV or of pharmaceutically ac- ceptable salts thereof for preparing a medicament for the treatment of cancer. Another aspect of the present invention relates to the use of compounds of formulae I, Il and/or IV or of pharmaceutically acceptable salts thereof for preparing a medicament for the treatment or prophylaxis of virus infections.

The compounds of formulae I, Il and IV and/or their pharmaceutically acceptable salts are suitable for the treatment, inhibiton or control of growth and/or propagation of tumor cells and the disorders associated therewith. Accordingly, they are suitable for cancer therapy in warm-blooded vertebrates, for example mammals and birds, in particular man, but also other mammals, in particular useful and domestic animals, such as dogs, cats, pigs, ruminants (cattle, sheep, goats, bison, etc.), horses and birds, such as chicken, turkey, ducks, geese, guineafowl and the like.

The compounds of formulae 1, 11 and IV and/or their pharmaceutically acceptable salts are suitable for the therapy of cancer or cancerous disorders of the following organs: breast, lung, intestine, prostate, skin (melanoma), kidney, bladder, mouth, larynx, oesophagus, stomach, ovaries, pancreas, liver and brain or CNS.

The compounds of formulae 1, 11 and IV and/or their pharmaceutically acceptable salts are suitable for the treatment of virus infections in warm-blooded vertebrates, for example mammals and birds, in particular man, but also other mammals, in particular useful and domestic animals, such as dogs, cats, pigs, ruminants (cattle, sheep, goats, bison, etc.), horses and birds, such as chicken, turkey, ducks, geese, guineafowl and the like. They are suitable for treating virus infections like retrovirus infections such as HIV and HTLV, influenza virus infection, rhinovirus infections, herpes and the like.

The compounds according to the invention can be administered in a customary manner, for example orally, intravenously, intramuscularly or subcutaneously. For oral administration, the active compound can be mixed, for example, with an inert diluent or with an edible carrier; it can be embedded into a hard or soft gelatin capsule, it can be compressed to tablets or it can be mixed directly with the food/feed. The active compound can be mixed with excipients and administered in the form of indigestible tablets, buccal tablets, pastilles, pills, capsules, suspensions, potions, syrups and the like. Such preparations should contain at least 0.1 % of active compound. The composition of the preparation may, of course, vary. It usually comprises from 2 to 60% by weight of active compound, based on the total weight of the preparation in question (dosage unit). Preferred preparations of the compound I according to the invention comprise from 10 to 1000 mg of active compound per oral dosage unit.

The tablets, pastilles, pills, capsules and the like may furthermore comprise the following components: binders, such as traganth, gum arabic, corn starch or gelatin, excipients, such as dicalcium phosphate, disintegrants, such as corn starch, potato starch, alginic acid and the like, glidants, such as magnesium stearate, sweeteners, such as sucrose, lactose or saccharin, and/or flavors, such as peppermint, vanilla and the like. Capsules may furthermore comprise a liquid carrier. Other substances which modify the properties of the dosage unit may also be used. For example, tablets, pills and capsules may be coated with schellack, sugar or mixtures thereof. In addition to the active compound, syrups or potions may also comprise sugar (or other sweeteners), methyl- or propylparaben as preservative, a colorant and/or a flavor. The components of the active compound preparations must, of course, be pharmaceutically pure and nontoxic at the quantities employed. Furthermore, the active compounds can be formulated as preparations with a controlled release of active compound, for example as delayed-release preparations.

The active compounds can also be administered parenterally or intraperitoneal^. Solutions or suspensions of the active compounds or their salts can be prepared with water using suitable wetting agents, such as hydroxypropylcellulose. Dispersions can also be prepared using glycerol, liquid polyethylene glycols and mixtures thereof in oils. Frequently, these preparations furthermore comprise a preservative to prevent the growth of microorganisms.

Preparations intended for injections comprise sterile aqueous solutions and dispersions and also sterile powders for preparing sterile solutions and dispersions. The preparation has to be sufficiently liquid for injection. It has to be stable under the preparation and storage conditions and it has to be protected against contamination by microorganisms. The carrier may be a solvent or a dispersion medium, for example, water, etha- nol, a polyol (for example glycerol, propylene glycol or liquid polyethylene glycol), a mixture thereof and/or a vegetable oil.

The invention is further illustrated by the following, non-limiting examples.

I. Synthesis examples

Proton and carbon NMR spectra were obtained on a Bruker AC 300 spectrometer at 300 MHz. Proton spectra were referenced to tetramethylsilane as an internal standard and the carbon spectra were referenced to CDCb (purchased from Aldrich or Cambridge Isotope Laboratories, unless otherwise specified). Melting points were obtained on a Mel-Temp Il apparatus and are uncorrected. ESI Mass spectra were obtained on a Shimadzu LCMS-2010 EV Mass Spectrometer. HPLC analyses were obtained using an Alltech Alltima C18 Rocket Column utilizing PDA detection at 254 nm (unless otherwise specified) on a Shimadzu Prominence HPLC system. The following time program was utilized (flow rate of 2.5 mL per minute):

1. Preparation of 1 -{[2-(2,4-Difluorophenyl)-4-propyl-1 ,3-dioxolan-2-yl]methyl}-1 H- 1 ,2,4-triazole-5(4/-/)-thione (compound E6)

1.1 2-Bromo-1-(2,4-difluorophenyl)ethanone

To a stirred solution of 1-(2,4-difluorophenyl)ethanone (7.1 g, 45.5 mmol) in MeOH (200 ml_), Br2 (7.3 g, 45.5 mmol) was added dropwise at 0 ⁰ C. The mixture was then stirred for 8 h at room temperature. The reaction mixture was diluted with EtOAc (1 L) and washed with brine (2x200 ml_). The organic layer was separated, dried with sodium sulfate, and concentrated in vacuum to afford crude 2-bromoehtanone 2 (1O g, 93%) as red oil.

1.2 2-(Bromomethyl)-2-(2,4-difluorophenyl)-4-propyl-1 ,3-dioxolane

To a solution of 2-bromo-1-(2,4-difluorophenyl)ethanone (3.8 g, 16.2 mmol) and pen- tane-1 ,2-diol (21.0 mmol) in toluene (50 ml_), was added PTSA (279 mg, 1.62 mmol). The solution was stirred and heated at reflux with a Dean-Stark trap for 5 h, collecting water to facilitate the ketal formation. The reaction mixture was diluted with EtOAc (ethylacetate; 100 ml.) and washed with brine (2x50 ml_). The organic layer was separated, dried with sodium sulfate, and concentrated in vacuum. The residue was purified by column chromatography (silica gel, eluents: hexanes/EtOAc 4:1 ) to afford the title ketal compound (2.3 g, 44%) as clear oil.

1.3 1 -{[2-(2,4-Difluorophenyl)-4-propyl-1 ,3-dioxolan-2-yl]methyl}- 7H-1 ,2,4-triazole

To a stirred mixture of 1 ,2,4-triazole (193 mg, 2.8 mmol) and CS2CO3 (1.43 g, 4.4 mmol) in DMF (20 ml_), a solution of the ketal obtained in step 1.2 (1.3 g, 4.0 mmol) in DMF (10 ml.) was added dropwise at 0 ⁰ C. The reaction mixture was heated at 100 ⁰ C and stirred for 24 h. Ice-water (200 ml.) was added, and the product was extracted with EtOAc (2x50 ml_). The combined organic layers were dried with sodium sulfate and concentrated in vacuum. The residue was purified by column chromatography (silica gel, eluents: hexanes/EtOAc 3:2) to afford the title compound (150 mg, 17%) as clear oil.

1.4 1 -{[2-(2,4-Difluorophenyl)-4-propyl-1 ,3-dioxolan-2-yl]methyl}-1 H- 1 ,2,4-triazole- 5(4H)-thione To a stirred solution of triazole ketal obtained in step 1.3 (170 mg, 0.55 mmol) in DMF (10 ml), Ss (176 mg, 5.5 mmol) was added. The mixture was heated at reflux and stirring for 3 days. The reaction mixture was quenched with brine (50 ml.) and extracted with EtOAc (50 ml_). The organic layer was additionally washed with brine (50 ml_), separated, dried with sodium sulfate and concentrated in vacuum. The residue was then purified by column chromatography (silica gel, eluents: EtOAc/hexanes 1 :9 to 2:3) to afford the titled triazole thione as white solid (70 mg, 38%).

m.p. = 135-136 ⁰ C.

The following compounds were prepared in an analogous manner.

2. Preparation of 1 -{[2-(4-chlorophenyl)-4-propyl-1 ,3-dioxolan-2-yl]methyl}- 7H-1 ,2,4- triazole-5(4H)-thione (compound E5)

In this case, the ethanone (2-bromo-1-(4-chlorophenyl)ethanone) was commercially available.

m.p. = 133-134 ⁰ C

3. Preparation of 1 -{[2-(4-chloro-2-fluorophenyl)-4-propyl-1 ,3-dioxolan-2-yl)methyl)- 7H-1 ,2,4-triazole-5(4H)-thione (compound E2)

m.p. = 115-116 ⁰ C

4. Preparation of 1-{[2-(2-chloro-4-fluorophenyl)-4-propyl-1 ,3-dioxolan-2-yl]methyl}- 7H-1 ,2,4-triazole-5(4H)-thione (compound E3)

m.p. = 107-108 ⁰ C

5. Preparation of 1 -{[2-(3,4-difluorophenyl)-4-propyl-1 ,3-dioxolan-2-yl]methyl}- 7H- 1 ,2,4-triazole-5(4H)-thione (compound E4)

m.p. = 145-146 ⁰ C

II. Examples of the action against harmful fungi The fungicidal action of the compounds of the formulae I and Il was demonstrated by the following experiments:

A) Microtiter tests

The active substances were formulated separately as a stock solution in dimethyl sulfoxide (DMSO) at a concentration of 10 000 ppm.

Use example 1 : Activity against the late blight pathogen Phytophthora infestans in the microtiter test

The stock solution was pipetted into a microtiter plate (MTP) and diluted to the stated active substance concentration using a pea juice-based aqueous nutrient medium for fungi. An aqueous zoospore suspension of Phytophthora infestans was then added. The plates were placed in a water vapor-saturated chamber at temperatures of 18°C. Using an absorption photometer, the MTPs were measured at 405 nm on day 7 after the inoculation. The measured parameters were compared to the growth of the active substance-free control variant (= 100 %) and the fungus- and active substance-free blank value to determine the relative growth in % of the pathogens in the individual active substances.

Use example 2: Activity against the rice blast pathogen caused by Pyricularia oryzae in the microtiter test

The stock solution was pipetted into a microtiter plate (MTP) and diluted to the stated active substance concentration using a malt-based aqueous nutrient medium for fungi. An aqueous spore suspension of Pyricularia oryzae was then added. The plates were placed in a water vapor-saturated chamber at temperatures of 18°C. Using an absorption photometer, the microtiter plates were measured at 405 nm on day 7 after the in- oculation. The measured parameters were compared to the growth of the active substance-free control variant (= 100%) and the fungus- and active substance-free blank value to determine the relative growth in % of the pathogens in the individual active substances.

Use example 3: Activity against the Septoria blotch pathogen caused by Septoria tritici in the microtiter test

The stock solution was pipetted into a microtiter plate (MTP) and diluted to the stated active substance concentration using a malt-based aqueous nutrient medium for fungi. An aqueous spore suspension of Septoria tritici was then added. The plates were placed in a water vapor-saturated chamber at temperatures of 18°C. Using an absorption photometer, the microtiter plates were measured at 405 nm on day 7 after the inoculation. The measured parameters were compared to the growth of the active sub- stance-free control variant (= 100%) and the fungus- and active substance-free blank value to determine the relative growth in % of the pathogens in the individual active substances.

B) Greenhouse tests

The active substances were formulated separately or together as a stock solution comprising 25 mg of active substance which was made up to 10 ml using a mixture of acetone and/or dimethyl sulfoxide (DMSO) and the emulsifier Wettol EM 31 (wetting agent having emulsifying and dispersing action based on ethoxylated alkylphenols) in a vol- ume ratio of solvent/emulsifier of 99 to 1. This solution was then made up to 100 ml using water. This stock solution was diluted with the solvent/emulsifier/water mixture described to the active substance concentration given below.

Use example 4: Activity against early blight on tomatoes caused by Phytophthora in- festans with protective application

Young seedlings of tomato plants were grown in pots. The plants were sprayed to runoff with an aqueous suspension containing the concentration of active substance stated below. The next day, the treated plants were inoculated with an aqueous suspension of sporangia of Phytophthora infestans. After inoculation, the trial plants were immediately transferred to a humid chamber. After 6 days at 18 to 20 ⁰ C and a relative humidity close to 100%, the extent of fungal attack on the leaves was visually assessed as % diseased leaf area.

Use example 5: Curative action against Puccinia recondita on wheat (brown rust of wheat)

Leaves of potted wheat seedlings of the cultivar "Kanzler" were dusted with a suspension of spores of brown rust of wheat (Puccinia recondita). The plants were then placed in a chamber with high atmospheric humidity (90 to 95%), at 20-22 ⁰ C, for 24 hours.

During this time, the spores germinated and the germinal tubes penetrated into the leaf tissue. The next day, the infected plants were sprayed to runoff point with an aqueous suspension having the concentration of active substance stated below. After drying of the sprayed suspension, the test plants were returned into the greenhouse and culti- vated at temperatures between 20 and 22°C and at 65 to 70% relative atmospheric humidity for a further 7 days. The extent of the rust development on the leaves was then determined visually.

Use example 6: Protective action against Puccinia recondita on wheat (brown rust of wheat)

Leaves of potted wheat seedlings of the cultivar "Kanzler" were sprayed to runoff point with an aqueous suspension having the concentration of active substance stated be- low. The next day, the treated plants were dusted with a suspension of spores of brown rust of wheat (Puccinia recondita). The plants were then placed in a chamber with high atmospheric humidity (90 to 95%), at 20-22 ⁰ C, for 24 hours. During this time, the spores germinated and the germinal tubes penetrated into the leaf tissue. The next day, the test plants were returned into the greenhouse and cultivated at temperatures between 20 and 22°C and at 65 to 70% relative atmospheric humidity for a further 7 days. The extent of the rust development on the leaves was then determined visually.

Use example 7: Protective action against Blumeria graminis triticiou wheat (mildew of wheat)

Leaves of potted wheat seedlings of the cultivar "Kanzler" were sprayed to runoff point with an aqueous suspension having the concentration of active substance stated below. The next day, the treated plants were dusted with a suspension of spores of mildew of wheat (Blumeria graminis tritici). The plants were then returned into the green- house and cultivated at temperatures between 20 and 24°C and at 60 to 90% relative atmospheric humidity for a further 7 days. The extent of the mildew development on the leaves was then determined visually.

Use example 8: Protective action against Sphaerotheca fuliginea on cucumber (mildew of cucumber)

Leaves of potted cucumber seedlings (in the germ layer stage) were sprayed to runoff point with an aqueous suspension having the concentration of active substance stated below. The next day, the treated plants were dusted with a suspension of spores of mildew of cucumber (Sphaerotheca fuliginea). The plants were then returned into the greenhouse and cultivated at temperatures between 20 and 24°C and at 60 to 80% relative atmospheric humidity for a further 7 days. The extent of the mildew development on the seed leaves was then determined visually.