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Title:
ANTIHYPERLIPEMIC AGENTS
Document Type and Number:
WIPO Patent Application WO/1999/027965
Kind Code:
A1
Abstract:
Remedies for hypercholesterolemia, hyperlipemia and arteriosclerosis containing as the active ingredient neuropeptide Y Y5 receptor antagonists typified by, for example, a compound represented by formula [I-f-1].

Inventors:
FUKAMI TAKEHIRO (JP)
F KURODA TAKAHIRO (JP)
KANATANI AKIO (JP)
IHARA MASAKI (JP)
Application Number:
PCT/JP1998/005358
Publication Date:
June 10, 1999
Filing Date:
November 27, 1998
Export Citation:
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Assignee:
BANYU PHARMA CO LTD (JP)
FUKAMI TAKEHIRO (JP)
KURODA TAKAHIRO F (JP)
KANATANI AKIO (JP)
IHARA MASAKI (JP)
International Classes:
A61K31/352; C07D311/82; (IPC1-7): A61K45/00; A61K31/35; A61K31/44; A61K31/495
Domestic Patent References:
WO1997019682A11997-06-05
WO1997020820A11997-06-12
WO1997020821A11997-06-12
WO1997020822A11997-06-12
WO1997020823A21997-06-12
Other References:
MASSICOT F., ET AL.: "ANTIOBESITY ACTIVITY OF A NEW CYCLIC AMINO ARYLOXYACETATE IN OBESE MICE AND RATS.", EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY., EDITIONS SCIENTIFIQUE ELSEVIER, PARIS., FR, vol. 20., no. 06., 1 January 1985 (1985-01-01), FR, pages 559 - 562., XP002920020, ISSN: 0223-5234
GOLDSTEIN J. L., BROWN M. S.: "REGULATION OF THE MEVALONATE PATHWAY.", NATURE, NATURE PUBLISHING GROUP, UNITED KINGDOM, vol. 343., no. 6257., 1 February 1990 (1990-02-01), United Kingdom, pages 425 - 430., XP002920021, ISSN: 0028-0836, DOI: 10.1038/343425a0
Attorney, Agent or Firm:
BANYU PHARMACEUTICAL CO., LTD. (2-3 Nihombashi Honcho 2-chome Chuo-ku Tokyo, JP)
BANYU PHARMACEUTICAL CO., LTD. (2-3 Nihombashi Honcho 2-chome Chuo-ku Tokyo, JP)
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