Title:
AZEPIN-DERIVATIVES AS DERIVATIVES AS G- PROTEIN COUPLED RECEPTOR (GPR43) AGONISTS
Document Type and Number:
WIPO Patent Application WO/2011/151436
Kind Code:
A3
Abstract:
The present invention is directed to novel compounds of formula (I) Ar1__L1__R__Ar2__Ar3 and their use in treating and/or preventing inflammatory, gastrointestinal and/or metabolic disorders.
Inventors:
HOVEYDA HAMID (BE)
ZOUTE LUDIVINE (BE)
LENOIR FRANCOIS (BE)
ZOUTE LUDIVINE (BE)
LENOIR FRANCOIS (BE)
Application Number:
PCT/EP2011/059181
Publication Date:
February 02, 2012
Filing Date:
June 03, 2011
Export Citation:
Assignee:
EUROSCREEN SA (BE)
HOVEYDA HAMID (BE)
ZOUTE LUDIVINE (BE)
LENOIR FRANCOIS (BE)
HOVEYDA HAMID (BE)
ZOUTE LUDIVINE (BE)
LENOIR FRANCOIS (BE)
International Classes:
C07D223/10; A61K31/55; A61K31/551; A61P3/10; C07D225/02; C07D417/04; C07D417/14
Domestic Patent References:
| WO2005118573A1 | 2005-12-15 | |||
| WO2009055357A1 | 2009-04-30 | |||
| WO2006024815A1 | 2006-03-09 |
Foreign References:
| EP1698624A1 | 2006-09-06 | |||
| US20060160869A1 | 2006-07-20 |
Other References:
COVINGTON D K ET AL: "The G-protein-coupled receptor 40 family (GPR40-GPR43) and its role in nutrient sensing", BIOCHEMICAL SOCIETY TRANSACTIONS, PORTLAND PRESS LTD, GB LNKD- DOI:10.1042/BST0340770, vol. 34, no. 5, 1 November 2006 (2006-11-01), pages 770 - 773, XP008106357, ISSN: 0300-5127, Retrieved from the Internet
Attorney, Agent or Firm:
SCHREIBER, Ina et al. (96/98 Boulevard Carnot, Lille cedex, FR)
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