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Title:
AZOLE DERIVATIVE
Document Type and Number:
WIPO Patent Application WO/2013/062027
Kind Code:
A1
Abstract:
The invention according to the present application provides a therapeutic or prophylactic agent for diseases including mood disorders, anxiety disorders, schizophrenia, Alzheimer's disease, Parkinson's disease, Huntington's chorea, eating disorder, hypertension, digestive diseases, drug dependence, epilepsy, cerebral infarction, cerebral ischemia, cerebral edema, head injury, inflammations, immune-related diseases and alopecia. Specifically provided is an azole derivative having an arginine-vasopressin 1b receptor antagonistic activity and represented by general formula (I) or a pharmaceutically acceptable salt thereof.

Inventors:
YOSHINAGA MITSUKANE (JP)
KUWADA TAKESHI (JP)
MIYAKOSHI NAOKI (JP)
ISHIZAKA TOMOKO (JP)
WAKASUGI DAISUKE (JP)
SHIROKAWA SHIN-ICHI (JP)
HATTORI NOBUTAKA (JP)
SHIMAZAKI YOUICHI (JP)
Application Number:
JP2012/077541
Publication Date:
May 02, 2013
Filing Date:
October 25, 2012
Export Citation:
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Assignee:
TAISHO PHARMACEUTICAL CO., LTD. (24-1, Takada 3-chome Toshima-k, Tokyo 33, 〒1708633, JP)
International Classes:
C07D207/444; A61K31/4164; A61K31/4178; A61K31/4196; A61K31/4439; A61K31/444; A61K31/454; A61K31/4545; A61K31/46; A61K31/4725; A61K31/496; A61K31/537; A61K31/5377; A61K31/5386; A61K31/541; A61K31/553; A61P1/04; A61P9/10; A61P9/12; A61P17/14; A61P25/00; A61P25/08; A61P25/14; A61P25/16; A61P25/18; A61P25/22; A61P25/28; A61P25/30; A61P29/00; A61P37/02; A61P43/00; C07D231/12; C07D233/64; C07D233/70; C07D249/08; C07D249/10; C07D263/32; C07D277/20; C07D277/30; C07D401/04; C07D401/10; C07D403/04; C07D403/06; C07D403/10; C07D413/10; C07D451/06; C07D491/107; C07D498/08
Domestic Patent References:
WO2011104322A12011-09-01
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Foreign References:
JP2009537581A2009-10-29
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Other References:
See also references of EP 2772482A4
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Attorney, Agent or Firm:
ONO, SHINJIRO et al. (YUASA AND HARA, Section 206 New Ohtemachi Bldg., 2-1, Ohtemachi 2-chome, Chiyoda-k, Tokyo 04, 〒1000004, JP)
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