Title:
BENZOTRIAZOLE-DERIVED Α AND Β UNSATURATED AMIDE COMPOUND USED AS TGF-ΒR1 INHIBITOR
Document Type and Number:
WIPO Patent Application WO/2017/215506
Kind Code:
A1
Abstract:
A benzotriazole-derived α and β unsaturated amide compound used as TGF-βR1 inhibitor or a pharmaceutically acceptable salt thereof, the structure of the compound being as shown in formula (I).
Inventors:
SUN FEI (CN)
WU LIFANG (CN)
DING CHARLES Z (CN)
HU GUOPING (CN)
LI JIAN (CN)
CHEN SHUHUI (CN)
LU JIANYU (CN)
WU LIFANG (CN)
DING CHARLES Z (CN)
HU GUOPING (CN)
LI JIAN (CN)
CHEN SHUHUI (CN)
LU JIANYU (CN)
Application Number:
PCT/CN2017/087546
Publication Date:
December 21, 2017
Filing Date:
June 08, 2017
Export Citation:
Assignee:
MEDSHINE DISCOVERY INC (CN)
International Classes:
A61K31/4155; C07D401/14; A61K31/4439; A61P35/00; C07D471/04
Domestic Patent References:
WO2004050659A1 | 2004-06-17 |
Foreign References:
CN1681501A | 2005-10-12 | |||
CN103025731A | 2013-04-03 | |||
CN1511157A | 2004-07-07 |
Other References:
See also references of EP 3470409A4
Attorney, Agent or Firm:
SHANGHAI BESHINING LAW OFFICE (CN)
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