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Patent Searching and Data


Title:
BICYCLIC DERIVATIVES OF MORPHINE-6-GLUCURONIDE, PREPARATION METHOD THEREOF AND USE OF SAME IN THERAPEUTICS
Document Type and Number:
WIPO Patent Application WO/2010/067008
Kind Code:
A3
Abstract:
The invention relates to compounds having formula (I) wherein: R1 represents a hydrogen atom or a (C1-C4)alkyl group; R2 represents a hydroxyl group, a thiol group, a (C1-C4)alkyloxy group or a thio(C1-C4)alkyl group; and n is an integer equal to 1 or 2, in the form of a base or acid addition salt, as well as in hydrate or solvate form. The invention also relates to the preparation method thereof and to the use of same in therapeutics.

Inventors:
DLUBALA, Alain (Patent Department17, avenue de France Paris, F-75013, FR)
RIPOCHE, Isabelle (Ecole Nationale Supérieure de Clermont-Ferrand, Campus Cezeaux - BP 187, Aubière Cedex, F-63174, FR)
TRECANT, Claire (16 rue de Copenhague, Strasbourg, Strasbourg, F-67000, FR)
Application Number:
FR2009/052446
Publication Date:
July 07, 2011
Filing Date:
December 08, 2009
Export Citation:
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Assignee:
SANOFI (174 avenue de France, Paris, Paris, F-75013, FR)
DLUBALA, Alain (Patent Department17, avenue de France Paris, F-75013, FR)
RIPOCHE, Isabelle (Ecole Nationale Supérieure de Clermont-Ferrand, Campus Cezeaux - BP 187, Aubière Cedex, F-63174, FR)
TRECANT, Claire (16 rue de Copenhague, Strasbourg, Strasbourg, F-67000, FR)
International Classes:
C07H15/24; A61K31/485; A61K31/519; A61K31/7042; A61P25/04; C07H7/06; C07H17/00
Domestic Patent References:
WO1998046618A11998-10-22
Foreign References:
FR2864082A12005-06-24
Attorney, Agent or Firm:
PIGASSE, Caroline (Département Brevets17, avenue de France Paris, F-75013, FR)
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