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Title:
BISPHOSPHONIC ACID AND COFORMERS WITH LYSIN, GLYCIN, NICOTINAMIDE FOR TREATING PSORIATIC ARTHRITIS
Document Type and Number:
WIPO Patent Application WO/2017/208070
Kind Code:
A1
Abstract:
Preparation, in-vitro and in vivo characterization of novel forms of (1-hydroxy - 2-imidazol-1-yl-1-phosphono-ethyl) phosphonic acid, suitable for pharmaceutical compositions in drug delivery systems for humans.

Inventors:
HANNA MAZEN (US)
Application Number:
PCT/IB2017/000746
Publication Date:
December 07, 2017
Filing Date:
May 31, 2017
Export Citation:
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Assignee:
GRUENENTHAL GMBH (DE)
International Classes:
A61K31/198; A61K31/662; A61P17/06; A61P19/02
Domestic Patent References:
WO2015051327A12015-04-09
WO2006002009A22006-01-05
WO2007093226A12007-08-23
WO2003007916A12003-01-30
WO2006080780A12006-08-03
WO2007032808A12007-03-22
WO2005005447A22005-01-20
WO2008064849A12008-06-05
Foreign References:
US9169279B22015-10-27
US20160016982A12016-01-21
US20150306116A12015-10-29
US20060068010A12006-03-30
US20070014319A12007-01-18
US20070238707A12007-10-11
US20060178439A12006-08-10
Other References:
COLEMAN ET AL., BRITISH J CANCER, vol. 102, no. 7, 2010, pages 1099 - 1105
GNANT ET AL., NEW ENGLAND J MEDICINE., vol. 360, no. 17, 2009, pages 679 - 691
DAVIES ET AL., J CLINICAL ONCOLOGY, vol. 28, no. 7s, 2010
SORBERA ET AL., DRUGS OF THE FUTURE, vol. 25, no. 3, 2000
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