Title:
C20 THROUGH C26 AMINO STEROIDS
Document Type and Number:
WIPO Patent Application WO1987001706
Kind Code:
A3
Inventors:
MCCALL JOHN M (US)
AYER DONALD E (US)
JACOBSEN E JON (US)
VAN DOORNIK FREDERICK J (US)
PALMER JOHN R (US)
KARNES HAROLD A (US)
AYER DONALD E (US)
JACOBSEN E JON (US)
VAN DOORNIK FREDERICK J (US)
PALMER JOHN R (US)
KARNES HAROLD A (US)
Application Number:
PCT/US1986/001797
Publication Date:
July 16, 1987
Filing Date:
August 28, 1986
Export Citation:
Assignee:
UPJOHN CO (US)
MCCALL JOHN M (US)
AYER DONALD E (US)
JACOBSEN E JON (US)
DOORNIK FREDERICK J VAN (US)
PALMER JOHN R (US)
KARNES HAROLD A (US)
MCCALL JOHN M (US)
AYER DONALD E (US)
JACOBSEN E JON (US)
DOORNIK FREDERICK J VAN (US)
PALMER JOHN R (US)
KARNES HAROLD A (US)
International Classes:
C07D213/65; C07D213/74; C07D239/50; C07D249/14; C07D251/70; C07D295/135; C07D307/68; C07D333/66; C07D401/14; C07J3/00; C07J5/00; C07J7/00; C07J21/00; C07J31/00; C07J41/00; C07J43/00; (IPC1-7): C07J41/00; A61K31/56; A61K31/58; C07C93/14; C07D213/02; C07D239/24; C07D251/12; C07D253/06; C07D307/68; C07D333/52; C07D401/04; C07J5/00; C07J7/00; C07J43/00
Foreign References:
| GB954146A | 1964-04-02 | |||
| DE1087598B | 1960-08-25 | |||
| US3144446A | 1964-08-11 | |||
| US2665274A | 1954-01-05 | |||
| GB1390014A | 1975-04-09 | |||
| FR1413722A | 1965-10-08 | |||
| GB1345640A | 1974-01-30 |
Other References:
Journal of the Chemical Society, Perkin Transaction I, 1972 (London, GB), G. RAPI et al., "Amino- and Dienamino-Derivatives Formed from Adrenocortical Steroids and Heterocyclic Bases", pages 502-507, see the whole document cited in the application
Journal of Organic Chemistry, Vol. 26, No. 4, 18 April 1961 (Washington DC, USA), R.E. SCHAUB et al., "The Synthesis of Certain C-21-Substituted Derivatives of 21-Deoxyhydrocortisone, 21-Deoxy-9 alpha-Fluorhydrocortisone, and Progesterone", pages 1223-1227, see the whole document cited in the application
CHEMICAL ABSTRACTS, Vol. 70, No. 25, 23 June 1969 (Columbus, Ohio, USA), E.M. GOL'DBERG et al., "Nucleophilic Substitution of Iodine at Position 21 in 21-Iodo-17-alpha-Hydroxyprogesterone", see page 380, Abstract No. 115402v, Khim.-Farm. Zh. 1968, 2 (11), 26-9
CHEMICAL ABSTRACTS, Vol. 85, No. 11, 13 September 1976 (Columbus, Ohio, USA), D. MAHESH et al., " A Convenient Preparation of 1-Aroylpiperazines", see page 542, Abstract No. 78082c, Org. Prep. Proced. Int. 1976, 8 (1-2), 85-6
Journal of Organic Chemistry, Vol. 26, No. 4, 18 April 1961 (Washington DC, USA), R.E. SCHAUB et al., "The Synthesis of Certain C-21-Substituted Derivatives of 21-Deoxyhydrocortisone, 21-Deoxy-9 alpha-Fluorhydrocortisone, and Progesterone", pages 1223-1227, see the whole document cited in the application
CHEMICAL ABSTRACTS, Vol. 70, No. 25, 23 June 1969 (Columbus, Ohio, USA), E.M. GOL'DBERG et al., "Nucleophilic Substitution of Iodine at Position 21 in 21-Iodo-17-alpha-Hydroxyprogesterone", see page 380, Abstract No. 115402v, Khim.-Farm. Zh. 1968, 2 (11), 26-9
CHEMICAL ABSTRACTS, Vol. 85, No. 11, 13 September 1976 (Columbus, Ohio, USA), D. MAHESH et al., " A Convenient Preparation of 1-Aroylpiperazines", see page 542, Abstract No. 78082c, Org. Prep. Proced. Int. 1976, 8 (1-2), 85-6
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