Title:
CARBOXYLIC ACID DERIVATIVE AS AT2R RECEPTOR ANTAGONIST
Document Type and Number:
WIPO Patent Application WO/2018/224037
Kind Code:
A1
Abstract:
The present invention relates to a compound shown in formula (II) or a pharmaceutically acceptable salt thereof and an application of the same in preparing a drug for treating a disease related to angiotensin II receptor type 2 (AT2R). (II)
Inventors:
ZHANG YANG (CN)
WU WENTAO (CN)
LI ZHIXIANG (CN)
TENG MINGXING (CN)
YANG GUANGWEN (CN)
LI JIE (CN)
LI JIAN (CN)
CHEN SHUHUI (CN)
WU WENTAO (CN)
LI ZHIXIANG (CN)
TENG MINGXING (CN)
YANG GUANGWEN (CN)
LI JIE (CN)
LI JIAN (CN)
CHEN SHUHUI (CN)
Application Number:
PCT/CN2018/090432
Publication Date:
December 13, 2018
Filing Date:
June 08, 2018
Export Citation:
Assignee:
MEDSHINE DISCOVERY INC (CN)
International Classes:
C07D217/26; A61K31/47; A61P25/00
Domestic Patent References:
WO2011088504A1 | 2011-07-28 |
Foreign References:
CN102821765A | 2012-12-12 | |||
CN106478502A | 2017-03-08 | |||
CN103003244A | 2013-03-27 |
Other References:
PAIN. MEDICINE, vol. 14, 2013, pages 1557 - 1568
LANCET, vol. 383, 2014, pages 1637 - 1647
EXPERT OPIN. INVESTIG. DRUGS., vol. 23, 2014, pages 1 - 12
EXPERT. OPIN. THER. TARGETS., vol. 19, 2015, pages 25 - 35
BERGE ET AL.: "Pharmaceutical Salts", JOURNAL OF PHARMACEUTICAL SCIENCE, vol. 66, 1977, pages 1 - 19, XP002675560, DOI: 10.1002/jps.2600660104
See also references of EP 3620454A4
LANCET, vol. 383, 2014, pages 1637 - 1647
EXPERT OPIN. INVESTIG. DRUGS., vol. 23, 2014, pages 1 - 12
EXPERT. OPIN. THER. TARGETS., vol. 19, 2015, pages 25 - 35
BERGE ET AL.: "Pharmaceutical Salts", JOURNAL OF PHARMACEUTICAL SCIENCE, vol. 66, 1977, pages 1 - 19, XP002675560, DOI: 10.1002/jps.2600660104
See also references of EP 3620454A4
Attorney, Agent or Firm:
SHANGHAI BESHINING LAW OFFICE (CN)
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