Title:
COMPOUND, ANTI-ALLERGY DRUG, AND MEDIATOR RELEASE INHIBITOR
Document Type and Number:
WIPO Patent Application WO/2019/225035
Kind Code:
A1
Abstract:
The compound represented by the general formula exhibits strong anti-allergy activity. R1 represents a substituted or unsubstituted acyloxy group, or a substituted or unsubstituted acylamino group. R2 represents a substituted or unsubstituted alkyl group.
Inventors:
TAI AKIHIRO (JP)
MIURA KAORI (JP)
WAKAYAMA SACHIO (JP)
MIURA KAORI (JP)
WAKAYAMA SACHIO (JP)
Application Number:
PCT/JP2018/044160
Publication Date:
November 28, 2019
Filing Date:
November 30, 2018
Export Citation:
Assignee:
LAIMU CORP (JP)
International Classes:
C07D307/62; A61K31/366; A61P37/08
Domestic Patent References:
| WO2014050894A1 | 2014-04-03 | |||
| WO2009014343A2 | 2009-01-29 |
Foreign References:
| JP2017031083A | 2017-02-09 | |||
| JP2015003894A | 2015-01-08 | |||
| JPS61263969A | 1986-11-21 | |||
| JP2019006692A | 2019-01-17 |
Other References:
IWAOKA, Y. ET AL.: "Affinity resins as new tools for identifying target proteins of ascorbic acid", ANALYST, vol. 143, no. 4, 9 January 2018 (2018-01-09), pages 874 - 882, XP055655485
KATO, K. ET AL.: "Studies on Scavengers of Active Oxygen Species. 1.Synthesis and Biological Activity of 2-0-Alkylascorbic Acids", J. MED. CHEM., vol. 31, no. 4, 1988, pages 793 - 798, XP055655494
TAI, AKIHIRO ET AL.: "Antiallergic Effects of Ascorbic Acid Derivatives", VI TAMINS, vol. 91, no. 9, 2017, pages 579 - 580
KATO, K. ET AL.: "Studies on Scavengers of Active Oxygen Species. 1.Synthesis and Biological Activity of 2-0-Alkylascorbic Acids", J. MED. CHEM., vol. 31, no. 4, 1988, pages 793 - 798, XP055655494
TAI, AKIHIRO ET AL.: "Antiallergic Effects of Ascorbic Acid Derivatives", VI TAMINS, vol. 91, no. 9, 2017, pages 579 - 580
Attorney, Agent or Firm:
SIKS & CO. (JP)
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