Title:
CONDENSED HETEROCYCLIC COMPOUNDS AS ANTI-INFLAMMATORY AND IMMUNOMODULATORY AGENTS
Document Type and Number:
WIPO Patent Application WO1999045926
Kind Code:
B1
Abstract:
The present invention relates to use of a compound of formula (1) as an immunomodulatory or anti-inflammatory drug or for use in the treatment of a therapeutic indication in which inhibition of dehydro-orate dehydrogenase (DHODH) is beneficial and salts and physiologically functional salts thereof, wherein X, R<5>, R<6>, A, Z<1> and Z<2> have the meanings given in Claim 1.
Inventors:
SHANNON PATRICK VIVIAN RICHARD (GB)
EICHHOLTZ THOMAS (GB)
LINSTEAD DAVID (GB)
MASDIN PHILIP (GB)
SKINNER RICHARD (GB)
EICHHOLTZ THOMAS (GB)
LINSTEAD DAVID (GB)
MASDIN PHILIP (GB)
SKINNER RICHARD (GB)
Application Number:
PCT/GB1999/000580
Publication Date:
November 04, 1999
Filing Date:
February 25, 1999
Export Citation:
Assignee:
UNIV CARDIFF (GB)
SHANNON PATRICK VIVIAN RICHARD (GB)
EICHHOLTZ THOMAS (GB)
LINSTEAD DAVID (GB)
MASDIN PHILIP (GB)
SKINNER RICHARD (GB)
SHANNON PATRICK VIVIAN RICHARD (GB)
EICHHOLTZ THOMAS (GB)
LINSTEAD DAVID (GB)
MASDIN PHILIP (GB)
SKINNER RICHARD (GB)
International Classes:
A61K31/41; A61K31/422; A61K31/4245; A61K31/454; A61K31/7056; (IPC1-7): A61K31/44; A61K31/40; A61K31/41; A61K31/415; A61K31/42; A61K31/445; A61K31/535; A61K31/70
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