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Title:
CRYSTALLINE FORM OF(7-[4-(4-FLUOROPHENYL)-6-ISOPROPYL-2-(N- METHYL-N-METHYLSULFONYLAMINO)PYRIMIDIN-5-YL]-(3R,5S)- DIHYDROXY-(E)-6-HEPTENOIC ACID INTERMEDIATE, PROCESS FOR PREPARING THE SAME AND USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2009/128091
Kind Code:
A3
Abstract:
Disclosed herein is a crystalline form of methyl 7-[4-(4-flourophenyl)-6- isopropyl-2-(N-methyl-N-methylsulfonylamino)-pyrimidin-5-yl]-(3R)-3-hydroxy-5-oxo- (E)-6-heptenate (rosuvastatin intermediate), process for producing the same and using the same for producing rosuvastatin or pharmaceutically acceptable salts thereof.

Inventors:
MAHAJAN SANJAY (IN)
SETHI MADHURESH (IN)
RAY PURNA CHANDRA (IN)
DATTA DEBASHISH (IN)
Application Number:
PCT/IN2009/000116
Publication Date:
November 04, 2010
Filing Date:
February 20, 2009
Export Citation:
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Assignee:
MATRIX LAB LTD (IN)
MAHAJAN SANJAY (IN)
SETHI MADHURESH (IN)
RAY PURNA CHANDRA (IN)
DATTA DEBASHISH (IN)
International Classes:
C07D239/42
Domestic Patent References:
WO2008067440A22008-06-05
Foreign References:
CN1872841A2006-12-06
Attorney, Agent or Firm:
BABU, M.R., Ramesh (709/710 Tolstoy House,15-17 Tolstoy Marg, New Delhi 1, IN)
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