Title:
CYCLIC AMIDE DERIVATIVE
Document Type and Number:
WIPO Patent Application WO/2012/029942
Kind Code:
A1
Abstract:
Provided is a compound represented by formula (1) or a pharmacologically acceptable salt thereof. (In the formula, A represents a C6-10 arylene group or the like; R1a, R1b and R1c each independently represents a hydrogen atom, a halogen atom, a C1-4 alkyl group, a C1-4 alkoxy group or the like; R2 represents an optionally substituted C6-10 aryl group, an optionally substituted 5-12 membered monocyclic or polycyclic heteroaryl group, an optionally substituted C7-16 aralkyl group or the like; m represents 0 or the like; and n represents an integer of 0-2.)
Inventors:
HORIUCHI YOSHIHIRO (JP)
FUJIWARA HIROAKI (JP)
SUDA HITOSHI (JP)
SASAKI IZUMI (JP)
IWATA MITSUTAKA (JP)
SAWAMURA KIYOTO (JP)
FUJIWARA HIROAKI (JP)
SUDA HITOSHI (JP)
SASAKI IZUMI (JP)
IWATA MITSUTAKA (JP)
SAWAMURA KIYOTO (JP)
Application Number:
PCT/JP2011/070010
Publication Date:
March 08, 2012
Filing Date:
September 02, 2011
Export Citation:
Assignee:
DAINIPPON SUMITOMO PHARMA CO (JP)
HORIUCHI YOSHIHIRO (JP)
FUJIWARA HIROAKI (JP)
SUDA HITOSHI (JP)
SASAKI IZUMI (JP)
IWATA MITSUTAKA (JP)
SAWAMURA KIYOTO (JP)
HORIUCHI YOSHIHIRO (JP)
FUJIWARA HIROAKI (JP)
SUDA HITOSHI (JP)
SASAKI IZUMI (JP)
IWATA MITSUTAKA (JP)
SAWAMURA KIYOTO (JP)
International Classes:
C07C235/84; A61K31/166; A61K31/337; A61K31/341; A61K31/343; A61K31/351; A61K31/357; A61K31/36; A61K31/381; A61K31/40; A61K31/4025; A61K31/415; A61K31/4164; A61K31/421; A61K31/426; A61K31/44; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/5375; A61P3/04; A61P3/10; A61P9/08; A61P9/10; A61P9/12; A61P19/10; A61P25/18; A61P25/22; A61P25/24; A61P25/28; A61P27/06; A61P37/02; A61P43/00; C07C255/57; C07D207/335; C07D207/34; C07D213/50; C07D213/61; C07D213/82; C07D231/12; C07D233/64; C07D263/32; C07D277/20; C07D277/28; C07D277/30; C07D295/10; C07D305/08; C07D307/20; C07D307/78; C07D307/81; C07D309/12; C07D317/48; C07D319/18; C07D333/20; C07D333/58; C07D409/06; C07D409/14
Domestic Patent References:
WO2009001817A1 | 2008-12-31 |
Foreign References:
JP2010523692A | 2010-07-15 | |||
JP2010501578A | 2010-01-21 | |||
JP2009539937A | 2009-11-19 |
Other References:
See also references of EP 2612848A4
GREEN ET AL., JOURNAL OF NEUROSCIENCE, vol. 26, no. 35, 2006, pages 9047
YAU ET AL., THE JOURNAL OF NEUROSCIENCE, vol. 27, no. 39, 2007, pages 10487
GREEN ET AL., JOURNAL OF NEUROSCIENCE, vol. 26, no. 35, 2006, pages 9047
YAU ET AL., THE JOURNAL OF NEUROSCIENCE, vol. 27, no. 39, 2007, pages 10487
Attorney, Agent or Firm:
TANAKA, Mitsuo et al. (JP)
Mitsuo Tanaka (JP)
Mitsuo Tanaka (JP)
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