Title:
DERIVATIVES OF QUINAZOLINEDIONE PHTHALIMIDE, PREPARATIONS THEREOF AND THEIR THERAPEUTIC USES
Document Type and Number:
WIPO Patent Application WO2001044228
Kind Code:
A3
Abstract:
The invention relates to a compound of general formula (I), wherein R1 represents a C1-6 alkyl, C2-6 alkenyl, C3-6 cycloalkyl, hydroxy-C1-6 alkyl or C1-3alkoxy-C1-6 alkyl group, R2 represents a NR8R9, -O-C1-6 alkylene-NR4R5, -O-C1-6alkylene-CONR4R5 or -O-C1-6 alkylene-CO2R6 group or a group of formula (a), R3 represents a hydrogen atom, a hydroxy, a halogen atom, a cyano, a nitro, an amino or a C1-3 alkyl group, and W represents a C1-3 alkylene or C2-3 alkenylene group; and to their salts and hydrates. The invention also relates to the therapeutic uses of the inventive derivatives.
Inventors:
ALETRU MICHEL (FR)
BOVY PHILIPPE R (FR)
NAMANE CLAUDIE (FR)
BOVY PHILIPPE R (FR)
NAMANE CLAUDIE (FR)
Application Number:
PCT/FR2000/003534
Publication Date:
December 13, 2001
Filing Date:
December 14, 2000
Export Citation:
Assignee:
SANOFI SYNTHELABO (FR)
ALETRU MICHEL (FR)
BOVY PHILIPPE R (FR)
NAMANE CLAUDIE (FR)
ALETRU MICHEL (FR)
BOVY PHILIPPE R (FR)
NAMANE CLAUDIE (FR)
International Classes:
A61P1/00; A61P11/00; A61P15/06; C07D403/06; C07D403/14; (IPC1-7): C07D403/06; A61K31/517; A61P9/12; C07D403/14
Domestic Patent References:
| WO1998018781A2 | 1998-05-07 | |||
| WO1994019342A1 | 1994-09-01 |
Foreign References:
| FR2784379A1 | 2000-04-14 |
Other References:
Y.EGUCHI ET AL.: "studies on hypotensive agents.", CHEMICAL AND PHARMACEUTICAL BULLETIN., vol. 39, no. 7, 1991, PHARMACEUTICAL SOCIETY OF JAPAN. TOKYO., JP, pages 1753 - 9, XP002105928, ISSN: 0009-2363
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