Title:
DIPHENYLPYRAZOLE COMPOUND, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF
Document Type and Number:
WIPO Patent Application WO/2022/147993
Kind Code:
A1
Abstract:
Provided are a diphenylpyrazole compound as represented by formula (I) below or an agrochemically acceptable salt thereof, which is a novel inhibitor targeting pest GSTs, has a wide range of inhibitory activity on GSTs in various pests, can effectively delay in vivo metabolism of pest GSTs on pesticides, thereby reducing the metabolic resistance of pests to pesticides, and being suitable for use as a synergist for pesticides.
Inventors:
LIU JIYUAN (CN)
ZHANG YALIN (CN)
ZHANG YALIN (CN)
Application Number:
PCT/CN2021/105643
Publication Date:
July 14, 2022
Filing Date:
July 12, 2021
Export Citation:
Assignee:
UNIV NORTHWEST A&F (CN)
International Classes:
C07D401/12; A01N43/56; A01N43/78; A01P7/04; C07D231/14; C07D403/12; C07D405/12; C07D417/12
Foreign References:
| CN103483313A | 2014-01-01 | |||
| CN105968092A | 2016-09-28 | |||
| CN1654457A | 2005-08-17 | |||
| CN1654456A | 2005-08-17 |
Other References:
DATABASE REGISTRY 23 April 2021 (2021-04-23), "4-Pyridinecarboxylic acid, 1,2-dihydro-2-oxo-, 2-[(1,3-diphenyl-1H-pyrazol-5-yl)carbonyl]hydrazide (CA INDEX NAME)", XP055956641, retrieved from STN Database accession no. 2636891-44-4
DATABASE REGISTRY 24 February 2006 (2006-02-24), "1H-Pyrazole-5-carboxylic acid, 1,3-diphenyl-, 2-benzoylhydrazide (CA INDEX NAME)", XP055956634, retrieved from STN Database accession no. 875156-62-0
ZHOU YUNYUN, WEI WEI, ZHU LIANGLIANG, LI YUXIN, LI ZHENGMING: "Synthesis and insecticidal activity study of novel anthranilic diamides analogs containing a diacylhydrazine bridge as effective Ca 2+ modulators", CHEMICAL BIOLOGY & DRUG DESIGN, vol. 92, no. 5, 1 November 2018 (2018-11-01), pages 1914 - 1919, XP055949627, ISSN: 1747-0277, DOI: 10.1111/cbdd.13349
J. ORG. CHEM., vol. 75, no. 3, 2010, pages 984 - 987
DATABASE REGISTRY 24 February 2006 (2006-02-24), "1H-Pyrazole-5-carboxylic acid, 1,3-diphenyl-, 2-benzoylhydrazide (CA INDEX NAME)", XP055956634, retrieved from STN Database accession no. 875156-62-0
ZHOU YUNYUN, WEI WEI, ZHU LIANGLIANG, LI YUXIN, LI ZHENGMING: "Synthesis and insecticidal activity study of novel anthranilic diamides analogs containing a diacylhydrazine bridge as effective Ca 2+ modulators", CHEMICAL BIOLOGY & DRUG DESIGN, vol. 92, no. 5, 1 November 2018 (2018-11-01), pages 1914 - 1919, XP055949627, ISSN: 1747-0277, DOI: 10.1111/cbdd.13349
J. ORG. CHEM., vol. 75, no. 3, 2010, pages 984 - 987
Attorney, Agent or Firm:
BEIJING MOUNTAINWILL INTELLECTUAL PROPERTY AGENCY (CN)
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