Title:
DRUG COMPOSITION FOR PERCUTANEOUS ABSORPTION
Document Type and Number:
WIPO Patent Application WO/2000/053184
Kind Code:
A1
Abstract:
A drug composition for percutaneous absorption, comprising (a) an active ingredient selected from the group consisting of quinazoline derivatives having a $g(a)¿1?-receptor blocking effect and salts thereof, (b) a substance selected from the group consisting of C¿8?-C¿15? fatty acids, C¿8?-C¿16? fatty acid esters, C¿8?-C¿12? higher alcohols, and geraniol, (c) a substance selected from the group consisting of polyhydric alcohols and ethanol and, if necessary, (d) benzyl alcohol. This composition enables efficient percutaneous absorption of terazosin or other drugs.
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Inventors:
YAMAUCHI HITOSHI (JP)
NAKAJIMA NORIKO (JP)
NISHI HIROYOSHI (JP)
MATSUOKA YOSHINORI (JP)
YANO SHINJI (JP)
NAKAJIMA NORIKO (JP)
NISHI HIROYOSHI (JP)
MATSUOKA YOSHINORI (JP)
YANO SHINJI (JP)
Application Number:
PCT/JP2000/001429
Publication Date:
September 14, 2000
Filing Date:
March 09, 2000
Export Citation:
Assignee:
DAIICHI SEIYAKU SAITAMA (JP)
MITSUBISHI CHEM CORP (JP)
YAMAUCHI HITOSHI (JP)
NAKAJIMA NORIKO (JP)
NISHI HIROYOSHI (JP)
MATSUOKA YOSHINORI (JP)
YANO SHINJI (JP)
MITSUBISHI CHEM CORP (JP)
YAMAUCHI HITOSHI (JP)
NAKAJIMA NORIKO (JP)
NISHI HIROYOSHI (JP)
MATSUOKA YOSHINORI (JP)
YANO SHINJI (JP)
International Classes:
A61K9/00; A61K31/517; A61K47/10; A61P13/02; A61K47/12; A61K47/14; (IPC1-7): A61K31/517; A61K9/70; A61P9/12; A61P13/02
Foreign References:
JPH1045597A | 1998-02-17 | |||
JPS63246338A | 1988-10-13 | |||
EP0760238A1 | 1997-03-05 |
Attorney, Agent or Firm:
Imamura, Masazumi (KRF Building 5-5 Kyobashi 1-chome Chuo-ku, Tokyo, JP)
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