Title:
ENNIATINES AND ENNIATINE DERIVATES USED TO CONTROL ENDOPARASITES
Document Type and Number:
WIPO Patent Application WO1993025543
Kind Code:
A3
Abstract:
The present invention relates to the use of cyclic depsipeptides having 18 ring atoms of the general formula (I) (I) in which R1 to R6 have the meaning given in the description, and to their optical isomers and racemates, in medicine and veterinary medicine for combating endoparasites, to their preparation, and to new cyclic depsipeptides having 18 ring atoms.
Inventors:
BONSE, GERHARD
LONDERSHAUSEN, MICHAEL
BISCHOFF, ERWIN
MUELLER, HARTWIG
HARDER, ACHIM
MENCKE, NORBERT
KURKA, PETER
JESCHKE, PETER
SCHERKENBECK, JUERGEN
LONDERSHAUSEN, MICHAEL
BISCHOFF, ERWIN
MUELLER, HARTWIG
HARDER, ACHIM
MENCKE, NORBERT
KURKA, PETER
JESCHKE, PETER
SCHERKENBECK, JUERGEN
Application Number:
PCT/EP1993/001436
Publication Date:
May 26, 1994
Filing Date:
June 07, 1993
Export Citation:
Assignee:
BAYER AKTIENGESELLSCHAFT
International Classes:
A61K31/395; A61P31/00; A61P33/00; C07C227/18; C07C229/06; C07C229/12; C07C229/14; C07C229/22; C07C229/34; C07C231/02; C07C233/36; C07C235/12; C07C271/22; C07D273/00; (IPC1-7): C07D273/00; A61K31/395; C07C231/02; C07C235/12; C07C229/06; C07C227/18
Foreign References:
| EP0382173A2 | 1990-08-16 |
Other References:
ZH. OBSHCH.KHIM. Bd. 38, Nr. 6, 1968, Seiten 1228 - 1239 MIKHALEVA, I.I. ET AL. 'Relation between structure and biological action in a series of enniatin B and its analogs'
J. ANTIBIOTICS Bd. 45, Nr. 8, 1992, Seiten 1207 - 1215 TOMODA, H. ET AL. 'New cyclodepsipeptides, enniatins D, E and F produced by Fusarium sp. FO-1305' in der Anmeldung erwähnt
HELVETICA CHIMICA ACTA Bd. 46, 1963, Seiten 927 - 935 PLATTNER, P.A. ET AL. 'Synthesen in der Depsipeptid-Reihe'
HELVETICA CHIMICA ACTA Bd. 46, 1963, Seiten 1715 - 1720 QUITT, P. ET AL. 'Synthesen in der Depsipeptidreihe' in der Anmeldung erwähnt
TETRAHEDRON LETTERS Bd. 2, 1971, Seiten 159 - 162 OVCHINNIKOV, Y. ET AL. 'The synthesis and some properties of Beauvericin'
AGRIC.BIOL.CHEM. Bd. 43, Nr. 5, 1979, Seiten 1079 - 1083 KANAOKA, M. ET AL. 'Synthesis of Bassianolide and its two homologs, Enniatin C and Decabassianolide'
CHEM.BER. Bd. 101, 1968, Seiten 1532 - 1539 LOSSE, G. & RAUE, H. 'Synthese von Stereoisomeren des Enniatins B'
J. ANTIBIOTICS Bd. 45, Nr. 8, 1992, Seiten 1207 - 1215 TOMODA, H. ET AL. 'New cyclodepsipeptides, enniatins D, E and F produced by Fusarium sp. FO-1305' in der Anmeldung erwähnt
HELVETICA CHIMICA ACTA Bd. 46, 1963, Seiten 927 - 935 PLATTNER, P.A. ET AL. 'Synthesen in der Depsipeptid-Reihe'
HELVETICA CHIMICA ACTA Bd. 46, 1963, Seiten 1715 - 1720 QUITT, P. ET AL. 'Synthesen in der Depsipeptidreihe' in der Anmeldung erwähnt
TETRAHEDRON LETTERS Bd. 2, 1971, Seiten 159 - 162 OVCHINNIKOV, Y. ET AL. 'The synthesis and some properties of Beauvericin'
AGRIC.BIOL.CHEM. Bd. 43, Nr. 5, 1979, Seiten 1079 - 1083 KANAOKA, M. ET AL. 'Synthesis of Bassianolide and its two homologs, Enniatin C and Decabassianolide'
CHEM.BER. Bd. 101, 1968, Seiten 1532 - 1539 LOSSE, G. & RAUE, H. 'Synthese von Stereoisomeren des Enniatins B'
Download PDF:
Previous Patent: BENZOXAZINONE AND BENZOTHIAZINONE DERIVATIVES HAVING CARDIOVASCULAR ACTIVITY
Next Patent: PROCESS FOR PRODUCING AMINE-BORANES
Next Patent: PROCESS FOR PRODUCING AMINE-BORANES