Title:
FLUORINE-CONTAINING PYRIMIDINE COMPOUNDS, HARMFUL FUNGI CONTROL AGENT, AND METHOD FOR PRODUCING FLUORINE-CONTAINING PYRIMIDINE COMPOUNDS
Document Type and Number:
WIPO Patent Application WO/2023/085142
Kind Code:
A1
Abstract:
Provided are novel fluorine-containing pyrimidine compounds and a method for producing the same. Compounds represented by general formula (1), (2), or (3). (In the formula, W and X each independently represent a hydrogen atom, a halogen atom, a C1-10 hydrocarbon group, -CmF2m+1, a nitro group, -OA1, -SOlA1, -SA1, -NA1A2, -B(OA1)(OA2), -COA1, -COOA1, or -CONA1A2, Y represents a halogen atom or -OA3, Z represents a halogen atom, a C1-10 hydrocarbon group, -CmF2m+1, a nitro group, -OA1, -SOlA1, -SA1, or -NA1A2, A1 and A2 each independently represent a hydrogen atom or a C1-10 hydrocarbon group, A3 represents a C1-12 hydrocarbon group, m represents an integer of 1-10, l represents an integer of 1-3, and n represents an integer of 0-3.)
Inventors:
AOTSU RIE (JP)
SEINO JUNYA (JP)
KOKIN KEISUKE (JP)
SEINO JUNYA (JP)
KOKIN KEISUKE (JP)
Application Number:
PCT/JP2022/040603
Publication Date:
May 19, 2023
Filing Date:
October 31, 2022
Export Citation:
Assignee:
UNIMATEC CO LTD (JP)
International Classes:
C07D401/04; A01N43/54; A01P3/00
Domestic Patent References:
| WO2021235420A1 | 2021-11-25 |
Foreign References:
| US5250530A | 1993-10-05 | |||
| JP2008528473A | 2008-07-31 | |||
| US20030069239A1 | 2003-04-10 | |||
| JP2020532549A | 2020-11-12 |
Other References:
KISHOR CHANDAN, ARYA TARUN, REDDI RAVIKUMAR, CHEN XIAOCHUN, SADDANAPU VENKATESHWARLU, MARAPAKA ANIL KUMAR, GUMPENA RAJESH, MA DAWE: "Identification, Biochemical and Structural Evaluation of Species-Specific Inhibitors against Type I Methionine Aminopeptidases", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, US, vol. 56, no. 13, 11 July 2013 (2013-07-11), US , pages 5295 - 5305, XP093065988, ISSN: 0022-2623, DOI: 10.1021/jm400395p
Attorney, Agent or Firm:
EINSEL Felix-Reinhard et al. (JP)
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