A HERBAL PERFORMANCE ENHANCEMENT MIX AND ITS PRODUCTION PROCESS

Technical Field

The invention relates to a mixture of herbal and animal ingredients which enhances virility, increases sperm count and prevents cerebral arteriosclerosis in the user, and the production process of this mixture thereof.

More specifically, the invention relates to a mixture of organic herbal and animal ingredients which enhance virility, and increase sperm count and quality without any chemical ingredients that are detrimental to human health and any side effects, and the production process of this mixture thereof.

State of the Art

In the state of the art, there are medicines that enhance virility, and increase sperm count and quality. Although they achieve the desired outcome, they can have serious side effects. These side effects may manifest as vascular disorders such as risk of heart attack and risk of cerebral hemorrhage, as well as others.

Although organic mixtures are available, their effectiveness is limited and the desired outcome may not be achieved.

Although the patent application 2012/00176 submitted to the Turkish Patent and Trademark Institution contains 1-99% methylprotodioxin and 5-95% dioxin by weight, there are no common ingredients with the invented product.

Although panax ginseng is an ingredient of the USPTO application no. US6544563B2, the content of this ingredient is about 3.3% by weight. None of its other ingredients are linked to our invention.

The Object of the Invention In the context of the state of the art, the object of the invention is to present a mixture which increases the sperm count and quality without causing cerebral arteriosclerosis. Description of the Figures

Figure 1 schematically illustrates the ingredients of a version of the invented mixture.

Figure 2 schematically illustrates a production version of the invented mixture.

Figure 3 schematically illustrates the ingredients of another version of the invented mixture.

REFERENCE NUMBERS

1 Mixture

1.1 Organic honey

1.2 Carob molasse 1.3 Maca root

1.4 Panax ginseng red

1.5 Ginger

1.6 Cinnamon

1.7 Ferula root 1.8 Turmeric

1.9 Ginkgo biloba

1.10 Black pepper

1.11 Bitter melon extract

1.12 Black mulberry molasse 2 Black cumin seed oil

4 Rosemary oil

5 Fig seed oil

6 Oregano oil

7 Mustard oil 9 Clove oil

11 Royal jelly

14 Cinchona

15 Tribulus terrestris

16 Horny goat weed 17 Organic pollen

18 Soda

19 Yeast

13 Water

300 Production method 301 Holding phase

302 Preparation phase

303 Mixing phase 304 Second holding phase

305 Second mixing phase

306 Third holding phase The invented mixture (1) is a purely herbal product with low production cost, which is easy to ingest and use, increases the sperm count and mobility in men and prevents cerebral arteriosclerosis thanks to beneficial fatty acids it contains. It does not contain any colorant and/or coloring agent. Shelf life of the product is longer than regular medicines thanks to its improved production process (100). It is free of any side effects caused by chemical active substances and does not contain any chemical agent sweeteners such as glucose/sucrose/fructose syrup.

Propolis (10) is widely used as a general purpose medicine and it is indicated for the treatment of cardiovascular and blood circulatory system disorders (anemia), respiratory tract infections, dental problems, dermal problems (tissue renewal, ulcers, eczema), wound treatments -particularly burn wounds (mycosis), mucous membrane infections and lesions, cancer, immune system disorders and digestive system disorders. In women, it is used for the treatment of osteoporosis, joint rheumatism, inflammatory disorders, wounds, cuts and some skin diseases, gastric wounds, upper respiratory tract disorders, asthma, bronchitis, otitis media, bad breath as well as for treatments of cancer, thanks to its anti-cancer properties. In a study with rats, propolis (10) was able to stop the formation of early tooth decay and in this respect can be used for the treatment of and protection against tooth decay. Furthermore, its use in the treatment of foot and skin problems of pets, endometritis in cows and fowl typhoid as well as blocking the enzymatic activity of urease have been reported. Unlike synthetic antibiotics, prolonged use of propolis (10) does not cause resistance to harmful bacteria and does not adversely affect beneficial bacteria. Therefore, propolis (10) is considered a rare broad-spectrum antibiotic.

Black pepper (1.10), which is called “Piper Nigrum” in Latin, contains a powerful antioxidant called piperine and prevents free radicals from damaging the cells. Studies have shown that it lowers cholesterol and also enhances the effectiveness of cholesterol lowering supplements. Black pepper (1.10) is also reported to slow replication of cancer cells in experimental studies and lead to death of these cells. Black pepper (1.10) is a plant seed that can be safely consumed by adults and children.

Clove (9), which is called “Syzygium Aromaticum” in Latin, is used in traditional medicine for the symptomatic treatment of small inflammations in the mouth or throat. Clove (9) temporarily relieves toothache. It is suitable for use by adults and the elderly. There are not enough studies about its use in children and adolescents.

Mustard (7), which is called “Brassica Juncea” in Latin, has been shown to be protective against cancer as organic isothiocyanate. Cytotoxicity of mustard (7) derivatives on neuroblastoma cells was investigated. Mustard (7) is known to be a natural source of antioxidant alpha-tocopherol.

Aqueous mustard (7) extracts have been shown to inhibit lipid peroxidation induced by FeS04-ascorbate on human erythrocyte membranes.

Black cumin seed oil (2), which is called “Semen Nigellae Sativae” in Latin, contains many chemical compounds such as thymokinone (TQ) (30-48%), flavonoids, anthocyanins, alkaloids and essential fatty acids, particularly linoleic and oleic acid.

It has traditionally been used in the treatment of respiratory and digestive disorders, renal and hepatic dysfunction and rheumatic diseases in different ways. Many studies have demonstrated the medicinal properties of black cumin seeds including immunomodulatory activity as well as anti-inflammatory, antimicrobial and antioxidant activity.

Some studies show that black cumin seed powder can increase blood sugar levels in people with diabetes. Black cumin seed may also increase cholesterol levels in people with diabetes.

Fig seed (5), which is called “Ficus Carica” in Latin, may reduce insulin requirements in patients with type 1 diabetes. Figs have been shown to lower blood sugar levels after consumption. The fruits, roots and leaves of the fig plant are used in traditional medicine to treat gastrointestinal problems (colic, indigestion, loss of appetite and diarrhea), respiration problems (sore throat, cough and bronchial problems) and cardiovascular disorders as well as used as an anti-inflammatory and antispasmodic agent. Rosemary (4), which is called “Rosmarinus Officinalis” in Latin, provides symptomatic relief in dyspepsia and helps with gastrointestinal spasms. Rosemary (4) is helpful in alleviating mild muscle and joint pain and minor peripheral circulatory disorders.

Black mulberry (1.12), which is called “Morus Nigra” in Latin, helps to prevent cardiovascular and inflammatory diseases, and cancer thanks to the phytochemicals it contains. Its ingredients acts as beneficial antioxidants for human health. Black mulberry (1.12) is rich in flavonoids.

Ferula root (1.7), which is called “Ferula Communis” in Latin, has traditionally been used to treat hysteria and dysentery. The root-stem of the plant which is known as “Al-kalakh” in Saudi Arabia is locally used for the treatment of skin infections, while the roasted flower buds are used to treat fever and dysentery.

Oregano (6), which is called “Origanum vulgare” in Latin, is known for its antimicrobial and antioxidant activity and may also serve as an antispasmodic and antidiabetic.

Bitter melon extract (1.11) is used in the treatment of gastrointestinal system diseases such as colitis, ulcer, duodenal ulcer, gastritis and excess acid. It has been shown to be beneficial for eczema and psoriasis as well as supporting the liver. Other benefits of bitter melon extract include rapid healing of wounds and inflammations, relieving bowel laziness and cell renewal. It also contains high levels of vitamin E and high quality protein.

Tribulus terrestris extract (15) may increase virility and sperm quality, and reduce the risk of prostate cancer. Studies have shown that it alleviates atherosclerosis.

Horny goat weed extract (16) is one of the most effective natural remedies for reducing high blood pressure, it protects against cardiovascular diseases, it is used in liver disorders and is known for its immune-enhancing properties. It promotes sperm production in men. Horny goat extract (16) is a helpful supplement for men struggling with impotence and enhances orgasm in women.

Cinchona extract (14) is used to treat lack of appetite, digestive disorders, bloating and indigestion, as well as strengthening and revitalizing the body in cases of asthenia and weakness.

Cinnamon (1.6), which is called “Cinnamomum verum” in Latin, is used for the symptomatic treatment of mild, spasmodic gastrointestinal complaints, including gas and flatulence. Ginger (1.9), which is called “Zingiber officinale” in Latin, is used to prevent nausea and vomiting due to motion sickness, as well as for the symptomatic treatment of mild, spasmodic gastrointestinal complaints, including gas and bloating. The antioxidant effect explains its effectiveness in colds or in increasing body resistance. Turmeric (1.8), which is called “Curcuma longa” in Latin, is used in the treat digestive disorders such as bloating, slow digestion and gas in the stomach.

Many current studies show that curcumin in turmeric (1.8) has an antidepressant effect and reduces the symptoms of depression.

Carob (1.2), which is called “Ceratonia siliqua” in Latin, contains vitamins A, C and B6 as well as the minerals iron, selenium, sodium, potassium and magnesium. 100gr of carob contains about 40gr of fiber. Some studies report that consumption of carob (1.2) pod powder or the juice extracted from raw carob (1.2) just before a standard oral rehydration solution (ORS), shortens the duration of diarrhea and reduces symptoms in children with acute diarrhea. Preliminary studies show that oral consumption of carob (1.2) or a specific carob (1.2) product for up to six weeks reduces the total and low-density lipoprotein (LDL or “bad cholesterol”) cholesterol in patients with high cholesterol. Other studies showed that carob (1.2) increased libido and sexual pleasure, as well as the viability of sperms thanks its vitamin and mineral content.

Royal jelly (11), which is called “Apis mellifera I.” in Latin, has been studied in terms of antibiotic, antitumor, blood pressure lowering and immune system regulating activity. Royal Jelly (11) has some female hormonal activity. In addition, it has been shown to have a cholesterol, insulin-like activity, and certain effect on the nervous system. In a study where the therapeutical properties of royal jelly was investigated by creating sperm abnormalities in terms of count and shape, and observing the DNA modifications in the hepatic and testicular tissue, royal jelly (11 ) was found to have alleviated the toxic activity of cyclosporin A in a dosage and time dependent manner when royal jelly and cyclosporin A are taken together compared to cyclosporine A alone. Therefore, royal jelly (11) was claimed to be a protective agent. In another study, it was reported that 0.05, 0.1 , 0.2, 0.3 and 0.4% royal jelly (11) added to the media during buffalo sperm freezing could increase in vitro fertilization capacity and viability of sperm.

Organic honey (1.1), which is called "Apis Mellifera" in Latin, is used to reduce stress and fatigue. Studies have shown that 15ml of organic honey (1.1) facilitates a healthy sleep. Organic honey (1.1) can be used alone or in combination with other ingredients in the treatment of some diseases. It can also increase the activity and effectiveness of the combined medicinal ingredients. Organic honey (1.1) is a common food and there is no dose limitation on its use. Organic honey (1.1) is an easy to digest, nourishing, protective, therapeutic and functional food thanks to the vitamins, minerals, organic acids, flavonoids, phenolic acids, amino acids and enzymes it contains. The antioxidant, antimicrobial and anticarcinogenic effects of organic honey (1.1) have been shown in many studies.

Ginseng panax (1.4), which is called “Panax quinquefolius” in Latin is traditionally used for symptoms of asthenia such as fatigue and weakness. Ginseng root is widely used to increase daily performance and for its adaptogenic, immunomodulatory, antineoplastic, cardiovascular, central nervous system and endocrine activity. Ginseng panax (1.4) is thought to improve adrenal and thyroid functions, especially in stressful situations. Ginseng panax (1.4) is widely used in the treatment of metabolic diseases such as hyperglycemia, hyperlipidemia and hepatosteatosis. Unless otherwise stated, a standardized ginseng panax (1.4) product is considered to contain 4% ginsenoside and these amounts are used as a comparison standard. Ginsenosides have various pharmacological and physiological effects such as anticancer, antidiabetic, immunomodulatory, neuroprotective, radioprotective, antiamnestic and antistress activity.

Ginkgo biloba (1.9), which is called “Salisburia adiantifolia” in Latin, is used to improve cognitive impairment and quality of life in mild age-related dementia. The main active compounds of Ginkgo biloba (1.9) are flavonoids and terpenic lactones. Ginkgo biloba (1.9) leaves contain 22-27% flavone glycosides (quercetin, campherol, isorhamnetin; biflavonelaramentoflavone), terpenic lactones 5-7% (2.8-3.4% ginkgolite A, B, C, J and M; 2, 6-3, 2% bilobalite), as well as other compounds, 8-12% proanthocyanidins, organic acids (hydroxycinurenic acid, quinurenic acid, protocolatechic acid and vanylic acid), oses, polysaccharides, ginkgolic acid (=anacardic acid), D-glucaric acid, alkylphenols (cardanols, cardols), phytosterols and carotenoids. The use of ginkgo biloba (1.9) extract for indications such as dizziness, dementia, functional heart complaints, tinnitus and peripheral artery occlusive disease has been approved by Commission E, WHO, ESCOP, NIH. It is used in traditional herbal therapy to relieve the weight of the legs, and alleviate the symptoms of cold hands and feet related to minor circulatory disorders. The increase in the bleeding tendency can be counted as one of the side effects. Propolis 10 has been used both internally and externally. It is known to kill bacteria, viruses and fungi; provide with local anesthetic, antiulcer and anti-inflammatory activity; lower blood pressure; and stimulate the immune system.

Propolis (10) is particularly effective as an antimicrobial agent against gram-positive bacteria, yeasts and certain viruses.

Cytotoxicity of propolis (10) and its chemical components has been shown to inhibit growth of tumor cells.

According to experimental scientific evidence, maca root (1.3), which is called “Lepidium meyenii” in Latin, has nutritious, energizing and fertility enhancing activity. Maca root (1.3) is also effective in the treatment sexual dysfunction, osteoporosis and prostate hyperplasia. Macaene and macamide, which are thought to have important bioactive properties, are merely maca plant related compounds. They have positive effects on sexual activity. Maca extracts contain carbohydrates that play a role in the energy metabolism and are readily hydrolyzable in more than 50% of dry matter. In published studies, maca has been shown to increase physical and mental energy levels. It has been reported to improve physical performance even in ovariectomized rats, as well as to reduce immobility time caused by depression. Maca was observed to increase dose-dependent locomotor activities in another study. At an oral dose of 2000mg per day, the performance of the athletes increased and their lap times decreased. In swimming tests, the physical activity of the mice increased and their serum lactic acid levels decreased. Total serum Fe, RBC and hematocrit levels of ovariectomized mice increased. It has been reported to reduce blood glucose, plasma and hepatic VLDL, LDL, total cholesterol and triachylglycerol levels when added to the diet of rats and mice with hereditary hypertriglyceridemia (HHTg). In the conclusion of this study, it was stated that maca and maca root (1.3) can be used in the treatment and prevention of chronic diseases.

Figure 1 illustrates a version of the mixture. Figure 3 illustrates a version with increased effectiveness thanks to added ingredients.

Figure 2 illustrates the production process (100) of the mixture (1) version with basic ingredients. The mixture (1) must be produced under nitrogen gas. In another version, however, it can be produced without nitrogen gas. It can also be produced by taking out some of the less important ingredients. In another version of the mixture (1), carob molasse (1.2) may be replaced by some other molasse.

Pine honey is the preferred organic honey (1.1). If pine honey is replaced with flower honey, the mixture (1) may crystallize in cold ambient temperatures.

The invented mixture (1) contains the ingredients listed in Table 1 by weight. The mixture (1) contains 27-33% (preferably 30%) organic honey (1.1) by weight that is comprised of 10% chestnut honey, 50% pine honey and 40% flower honey, 32-28% (preferably 35%) carob molasse (1.2) by weight, 1.2-1.8% (preferably 1.5%) maca root (1.3) by weight, 1.2- 1.8% (preferably 1.5%) panax ginseng (1.4) by weight, 1.2-18% (preferably 1.5%) ginger (1.5) by weight, 1.2-1.8% (preferably 1.5%) cinnamon (1.6) by weight, 1.2-1.8% (preferably 1.5%) ferula root (1.7) by weight, 1.2-1.8% (preferably 1.5%) turmeric (1.8) by weight, 1.2- 1.8% (preferably 1.5%) Ginkgo biloba (1.9) by weight, 0.2-1% (preferably 0.5%) black pepper (1.10) by weight, 1.2-1.8% (preferably 1.5%) bitter melon (1.11) by weight, 3-5% (preferably 5%) black mulberry molasse (1.12) by weight as well as 16-20% (preferably 17.5%) water (13) by weight to complete the formulation. Water (13) displays alkaline water property preferably in pH 8.0 ratio. Table 1

Another version of the mixture (1 ) contains black cumin seed oil (2), rosemary oil (4), fig seed oil (5), thyme oil (6), mustard oil (7), clove oil (9), royal jelly (11), cinchona (14), tribulus terrestris (15), organic pollen (17), soda (18) yeast in addition to the ingredients. Table 2 below lists percentages in relation to the weight of the mixture (1). In this version, the mixture (1) contains 27-33% (preferably 30% by weight) organic honey (1.1) that is comprised of 10% chestnut honey, 50% pine honey and 40% flower honey, 32-28% (preferably 35% by weight) carob molasse (1.2), 1.2-1.8% (preferably 1.5% by weight) maca root (1.3), 1.2-1.8% (preferably 1.5% by weight) panax ginseng (1.4), 1.2-18% (preferably 1.5% by weight) ginger (1.5), 1.2-1.8% (preferably 1.5% by weight) cinnamon (1.6), 1.2-1.8% (preferably 1.5% by weight) ferula root (1.7), 1.2-1.8% (preferably 1.5% by weight) turmeric (1.8), 1.2-1.8% (preferably 1.5% by weight) Ginkgo biloba (1.9), 0.2-1% (preferably 0.5% by weight) black pepper (1.10), 1.2-1.8% (preferably 1.5% by weight) bitter melon (1.11), 3-5% (preferably 5% by weight) black mulberry molasse (1.12), 1.2- 1.8% (preferably 1.5% by weight) black cumin seed oil (2), 1.2-1.8% (preferably 1.5% by weight) cinchona (14), 0.3-0.7% (preferably 0.5% by weight) rosemary oil (4), 0.3-0.7% (preferably 0.5% by weight) fig seed oil (5), 0.3-0.7% (preferably 0.5% by weight) thyme oil (6), 0.3-0.7% (preferably 0.5% by weight) mustard oil (7), 0.3-0.7% (preferably 0.5% by weight) clove oil (9), 0.3-0.7% (preferably 0.5% by weight) royal jelly (11), 1.2-1.8% (preferably 1.5% by weight) horny goat weed (16), 1.2-1.8% (preferably 1.5% by weight) organic pollen (17), 0.3-0.7% (preferably 0.5% by weight) soda (18), 1.2-1.8% (preferably 1.5% by weight) yeast (19) as well as 3-7% (preferably 4.5% by weight) water (13) to complete the formulation. Water (13) displays alkaline water property preferably in pH 8.0 ratio.

Table 2

The invention is a special mixture production method (300) and it is characterized by:

-the holding phase where extracted panax ginseng (1.4), ginkgo biloba (1.9), ferula root (1.7), bitter melon (1.11), turmeric (1.8), ginger (1.5), black pepper (1.10), maca root extract (1.3) and cinnamon (1.6) are held in pH 8.0 alkaline water in separate containers at 35-40ºC for at least two hours (301 ) in ratios d esignated for the mixture (1 ),

-the preparation phase (302) where organic honey (1.1), carob molasse (1.2) and black mulberry molasse (1.12) are placed in a vessel with agitator in ratios designated for the mixture (1), -the mixing phase (303), where each extract prepared in the holding phase (301) are added one by one and mixed, following the preparation phase (302)

-the second holding phase (304), where the temperature is increased to 70ºC and the mixture is held for hour, following the mixing phase (303)

-the second mixing phase (305), where there is another mixing process at 30-35ºC for at least 8 hours, following the second holding phase (304)

-the third holding phase (306), where there is a minimum of 6 hours of holding time, following the second mixing phase (305)

The holding phase (301), whereby extracted royal jelly (11) is added which has been held in pH 8.0 alkaline water at 35-40ºC for at least two h ours in the ratio designated for the mixture (1).

The holding phase (301), whereby extracted cinchona (14) is added which has been held in pH 8.0 alkaline water at 35-40ºC for at least two h ours in the ratio designated for the mixture (1).

The holding phase (301), whereby extracted horny goat weed (16) is added which has been held in pH 8.0 alkaline water at 35-40ºC f or at least two hours in the ratio designated for the mixture (1).

The holding phase (301), whereby extracted horny goat weed (16) is added which has been held in pH 8.0 alkaline water at 35-40ºC f or at least two hours in the ratio designated for the mixture (1).

The holding phase (301), whereby extracted organic pollen (17) is added which has been held in pH 8.0 alkaline water at 35-40ºC for at least two hours in the ratio designated for the mixture (1).

The holding phase (301), whereby extracted tribulus terrestris (15) is added which has been held in pH 8.0 alkaline water at 35-40ºC f or at least two hours in the ratio designated for the mixture (1).

The mixing phase (301), whereby soda (18) and yeast (19) is added in the ratio designated for the mixture (1). The second mixing phase (305), whereby black cumin seed oil (2) is added in the ratio designated for the mixture (1).

The second mixing phase (305), whereby clove oil (9) is added in the ratio designated for the mixture (1).

The second mixing phase (305), whereby mustard oil (7) is added in the ratio designated for the mixture (1).

The second mixing phase (305), whereby fig seed oil (5) is added in the ratio designated for the mixture (1).

The second mixing phase (305), whereby Oregon oil (6) is added in the ratio designated for the mixture (1).