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Title:
HETEROARYL COMPOUND HAVING PHARMACEUTICAL ACTIVITY
Document Type and Number:
WIPO Patent Application WO/2018/233655
Kind Code:
A1
Abstract:
The present invention provides a novel compound having selective inhibitory activity against Btk and better metabolic stability.

Inventors:
LIU XIN (CN)
YUAN ZHEDONG (CN)
KONG RUI (CN)
CHEN SHAN (CN)
Application Number:
PCT/CN2018/092122
Publication Date:
December 27, 2018
Filing Date:
June 21, 2018
Export Citation:
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Assignee:
SHANGHAI DUDE MEDICAL TECH CO LTD (CN)
International Classes:
C07D487/04; A61P29/00; A61P35/00; C07D473/34
Domestic Patent References:
WO2014130856A22014-08-28
WO2016010926A12016-01-21
WO2008121742A22008-10-09
WO2010009342A22010-01-21
Foreign References:
CN107501270A2017-12-22
CN106279172A2017-01-04
CN101674834A2010-03-17
CN103917545A2014-07-09
JP2010504324A2010-02-12
CN201180026837A2011-05-30
CN201280045383A2012-07-11
Other References:
NATURE, vol. 361, 1993, pages 226 - 233
ANTICANCER AGENTS IN MEDICINAL CHEMISTRY, vol. 7, no. 6, 2007, pages 624 - 632
LCK-DELETION MICE, vol. 16, 1998, pages 2351 - 2356
See also references of EP 3643716A4
Attorney, Agent or Firm:
TUO YING LAW OFFICES (SHANGHAI) (CN)
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