HETEROARYL DERIVATIVES AS SUPERIOR LIGANDS FOR NOCICEPTIN RECEPTOR ORL-1

Title:

HETEROARYL DERIVATIVES AS SUPERIOR LIGANDS FOR NOCICEPTIN RECEPTOR ORL-1

Document Type and Number:

WIPO Patent Application WO2003039469

Kind Code:

A3

Abstract:

Novel compounds of the formula (I), wherein R is optionally substituted heteroaryl or (a); R<1> is H or C1-C6 alkyl; and R<2> and R<3> are -CH3, -OCH3 or halo; or a pharmaceutically acceptable salt or solvate thereof, pharmaceutical compositions therefore, and the use of said compounds in the treatment of pain, anxiety, cough, asthma, depression and alcohol abuse are disclosed.

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Inventors:

TULSHIAN DEEN
HO GINNY D
NG FAY W

Application Number:

PCT/US2002/035539

Publication Date:

October 16, 2003

Filing Date:

November 06, 2002

Export Citation:

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Assignee:

SCHERING CORP (US)

International Classes:

A61K31/506; A61K45/00; A61P11/06; A61P11/14; A61P25/04; A61P25/22; A61P25/24; A61P25/32; A61P29/00; A61P37/08; A61P43/00; C07D451/06; (IPC1-7): C07D451/06; A61K31/46; A61P43/00

Domestic Patent References:

WO2001007050A1

2001-02-01

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