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Title:
HETEROCYCLIC COMPOUND OR SALT THEREOF, GPR35 AGONIST, AND PHARMACEUTICAL COMPOSITION
Document Type and Number:
WIPO Patent Application WO/2019/054386
Kind Code:
A1
Abstract:
Provided is a heterocyclic compound represented by general formula (I), or a pharmacologically acceptable salt of the heterocyclic compound. In general formula (I): X represents O or NH; R1 represents a substituted or unsubstituted aryl group, or a substituted or unsubstituted aromatic heterocyclic group; R2 represents a substituted or unsubstituted alkyl group, etc.; R3 represents COOR (where R is a hydrogen atom, an alkyl group, etc.); and the n appended to R2 represents the number of R2, and is an integer of 0-3.

Inventors:
MATSUNO KENJI (JP)
OHNO OSAMU (JP)
TANAKA SATOSHI (JP)
FURUTA KAZUYUKI (JP)
Application Number:
JP2018/033694
Publication Date:
March 21, 2019
Filing Date:
September 11, 2018
Export Citation:
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Assignee:
UNIV KOGAKUIN (JP)
NAT UNIV CORPORATION OKAYAMA UNIV (JP)
International Classes:
C07D215/48; A61K31/352; A61K31/435; A61K31/4433; A61P1/00; A61P3/10; A61P9/10; A61P37/08; C07D311/24; C07D405/04; C07D407/04; C07D409/04
Domestic Patent References:
WO2017015221A12017-01-26
WO2017139274A12017-08-17
WO2015162538A12015-10-29
Foreign References:
US20120115751A12012-05-10
JP2006520361A2006-09-07
JP2001139571A2001-05-22
CN1382688A2002-12-04
US3786071A1974-01-15
JP2010529996A2010-09-02
US3673218A1972-06-27
US20150265561A12015-09-24
CN105769846A2016-07-20
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Attorney, Agent or Firm:
TAIYO, NAKAJIMA & KATO (JP)
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