Title:
HETEROCYCLIC COMPOUND SERVING AS SYK INHIBITOR AND/OR SYK-HDAC DUAL INHIBITOR
Document Type and Number:
WIPO Patent Application WO/2016/197987
Kind Code:
A1
Abstract:
The present invention provides a heterocyclic compound serving as a Syk inhibitor and/or a Syk-HDAC dual inhibitor. Specifically, the present invention provides a compound represented by formula (I), wherein each group is defined by a description in the specification. The compound in the present invention has Syk inhibitory activity and/or Syk-HDAC dual-inhibitory activity, thereby being capable of treating diseases related to Syk and/or HDAC activity or expression level.
Inventors:
ZHANG HANCHENG (CN)
LIU SHIFENG (CN)
LIU SHIFENG (CN)
Application Number:
PCT/CN2016/085505
Publication Date:
December 15, 2016
Filing Date:
June 12, 2016
Export Citation:
Assignee:
HANGZHOU INNOGATE PHARMA CO LTD (CN)
International Classes:
C07D519/00; A61K31/4985; A61K31/5383; A61P9/00; A61P9/10; A61P19/08; A61P25/28; A61P35/00; A61P35/02; A61P37/02; A61P37/08; C07D487/04
Foreign References:
CN102307474A | 2012-01-04 | |||
US20130338142A1 | 2013-12-19 | |||
CN104059073A | 2014-09-24 |
Attorney, Agent or Firm:
XU & PARTNERS,LLC. (CN)
上海一平知识产权代理有限公司 (CN)
上海一平知识产权代理有限公司 (CN)
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