Title:
HYDROGENATION ANNULE [12] AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR
Document Type and Number:
WIPO Patent Application WO/2021/012478
Kind Code:
A1
Abstract:
Provided are a hydrogenation annule [12] aromatic compound and a preparation method therefor. The hydrogenation annule [12] aromatic compound is a stereoisomer of a represented compound or a compound as represented by formula (I), (I)
Inventors:
WANG MEIXIANG (CN)
SHI TANHAO (CN)
TONG SHUO (CN)
SHI TANHAO (CN)
TONG SHUO (CN)
Application Number:
PCT/CN2019/116305
Publication Date:
January 28, 2021
Filing Date:
November 07, 2019
Export Citation:
Assignee:
UNIV TSINGHUA (CN)
International Classes:
C07C13/70; C07C1/20; C07C17/395; C07C19/04; G01N1/28; G01N33/00
Foreign References:
| CN110372469A | 2019-10-25 | |||
| CN110372468A | 2019-10-25 | |||
| CN109384780A | 2019-02-26 |
Other References:
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WANG, QIUAN, CHIEF EDITOR: "Calixarene Chemistry", PHYSICAL ORGANIC CHEMISTRY, 30 June 2010 (2010-06-30)
HIROSE TOMOYASU, KOJIMA YASUHIRO, MATSUI HIDEHITO, HANAKI HIDEAKI, IWATSUKI MASATO, SHIOMI KAZURO, ŌMURA SATOSHI, SUNAZUKA TOSHIAK: "Total synthesis of (±)-naphthacemycin A9, possessing both antibacterial activity against methicillin-resistant Staphylococcus aureus and circumventing effect of β-lactam resistance", THE JOURNAL OF ANTIBIOTICS, NATURE PUBLISHING GROUP, GB, vol. 70, no. 5, 1 May 2017 (2017-05-01), GB, pages 574 - 581, XP055774986, ISSN: 0021-8820, DOI: 10.1038/ja.2016.141
R. SHAH, J. ET AL.: "9-Aminomethyl-9, 10-dihydroanthracene (AMDA) Analogs as Structural Probes for Steric Tolerance in 5-HT2A and H1 Receptor Binding Sites", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 20, no. 3, 31 December 2009 (2009-12-31), XP026861837, ISSN: 0960-894X, DOI: 20200422153829Y
JANA ANUPAM, MISZTAL KASJAN, ŻAK ANNA, GRELA KAROL: "Synthesis of Selectively Substituted or Deuterated Indenes via Sequential Pd and Ru Catalysis", JOURNAL OF ORGANIC CHEMISTRY, AMERICAN CHEMICAL SOCIETY, WASHINGTON, vol. 82, no. 8, 21 April 2017 (2017-04-21), Washington, pages 4226 - 4234, XP055774987, ISSN: 0022-3263, DOI: 10.1021/acs.joc.7b00200
CHOUDHURY SANTOSH KUMAR, ROUT PRAGATI, PARIDA BIBHUTI BHUSAN, FLORENT JEAN-CLAUDE, JOHANNES LUDGER, PHAOMEI GANNGAM, BERTOUNESQUE : "Metal-Free Activation of C(sp 3 )-H Bond, and a Practical and Rapid Synthesis of Privileged 1-Substituted 1,2,3,4-Tetrahydroisoquinolines", EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, WILEY-VCH, DE, vol. 2017, no. 35, 25 September 2017 (2017-09-25), DE, pages 5275 - 5292, XP055774990, ISSN: 1434-193X, DOI: 10.1002/ejoc.201700471
GOTO TATSUYA, IWATA TADAHISA, ABE HIDEKI: "Synthesis and Characterization of Biobased Polyesters Containing Anthraquinones Derived from Gallic Acid", BIOMACROMOLECULES, AMERICAN CHEMICAL SOCIETY, US, vol. 20, no. 1, 14 January 2019 (2019-01-14), US, pages 318 - 325, XP055774994, ISSN: 1525-7797, DOI: 10.1021/acs.biomac.8b01361
WANG, QIUAN, CHIEF EDITOR: "Calixarene Chemistry", PHYSICAL ORGANIC CHEMISTRY, 30 June 2010 (2010-06-30)
HIROSE TOMOYASU, KOJIMA YASUHIRO, MATSUI HIDEHITO, HANAKI HIDEAKI, IWATSUKI MASATO, SHIOMI KAZURO, ŌMURA SATOSHI, SUNAZUKA TOSHIAK: "Total synthesis of (±)-naphthacemycin A9, possessing both antibacterial activity against methicillin-resistant Staphylococcus aureus and circumventing effect of β-lactam resistance", THE JOURNAL OF ANTIBIOTICS, NATURE PUBLISHING GROUP, GB, vol. 70, no. 5, 1 May 2017 (2017-05-01), GB, pages 574 - 581, XP055774986, ISSN: 0021-8820, DOI: 10.1038/ja.2016.141
R. SHAH, J. ET AL.: "9-Aminomethyl-9, 10-dihydroanthracene (AMDA) Analogs as Structural Probes for Steric Tolerance in 5-HT2A and H1 Receptor Binding Sites", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 20, no. 3, 31 December 2009 (2009-12-31), XP026861837, ISSN: 0960-894X, DOI: 20200422153829Y
JANA ANUPAM, MISZTAL KASJAN, ŻAK ANNA, GRELA KAROL: "Synthesis of Selectively Substituted or Deuterated Indenes via Sequential Pd and Ru Catalysis", JOURNAL OF ORGANIC CHEMISTRY, AMERICAN CHEMICAL SOCIETY, WASHINGTON, vol. 82, no. 8, 21 April 2017 (2017-04-21), Washington, pages 4226 - 4234, XP055774987, ISSN: 0022-3263, DOI: 10.1021/acs.joc.7b00200
CHOUDHURY SANTOSH KUMAR, ROUT PRAGATI, PARIDA BIBHUTI BHUSAN, FLORENT JEAN-CLAUDE, JOHANNES LUDGER, PHAOMEI GANNGAM, BERTOUNESQUE : "Metal-Free Activation of C(sp 3 )-H Bond, and a Practical and Rapid Synthesis of Privileged 1-Substituted 1,2,3,4-Tetrahydroisoquinolines", EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, WILEY-VCH, DE, vol. 2017, no. 35, 25 September 2017 (2017-09-25), DE, pages 5275 - 5292, XP055774990, ISSN: 1434-193X, DOI: 10.1002/ejoc.201700471
GOTO TATSUYA, IWATA TADAHISA, ABE HIDEKI: "Synthesis and Characterization of Biobased Polyesters Containing Anthraquinones Derived from Gallic Acid", BIOMACROMOLECULES, AMERICAN CHEMICAL SOCIETY, US, vol. 20, no. 1, 14 January 2019 (2019-01-14), US, pages 318 - 325, XP055774994, ISSN: 1525-7797, DOI: 10.1021/acs.biomac.8b01361
Attorney, Agent or Firm:
TSINGYIHUA INTELLECTUAL PROPERTY LLC (CN)
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