Title:
INTERMEDIATE FOR COMPOUNDING 5-HYDROXYL-1,7-NAPHTHYRIDINE COMPOUND SUBSTITUTED BY ARYL OR HETEROARYL, AND PREPARATION METHOD THEREFOR
Document Type and Number:
WIPO Patent Application WO/2017/161555
Kind Code:
A1
Abstract:
The present invention relates to a compound represented by formula (IV), Ar being an aromatic ring or an heteroaromatic ring selected from a naphthalene ring, a pyridine ring, a thiophene ring, a furan ring and a substituted benzene ring, R3 being hydrogen or C1-3 alkyl. The present invention also relates a preparation method for the compound. The compound is an intermediate used for preparing a 5-hydroxyl-1,7-naphthyridine compound substituted by aryl or heteroaryl, used for inhibiting prolylhydroxylase.
Inventors:
ZHOU YUNLONG (CN)
CAI SUIXIONG (US)
JIAO LINGLING (CN)
JING YU (CN)
GUO MING (US)
WEN JIANFENG (CN)
CAI MINMIN (CN)
JI FENGHUA (CN)
CAI SUIXIONG (US)
JIAO LINGLING (CN)
JING YU (CN)
GUO MING (US)
WEN JIANFENG (CN)
CAI MINMIN (CN)
JI FENGHUA (CN)
Application Number:
PCT/CN2016/077327
Publication Date:
September 28, 2017
Filing Date:
March 25, 2016
Export Citation:
Assignee:
SHENYANG SUNSHINE PHARMACEUTICAL CO LTD (CN)
International Classes:
C07D213/80; C07D213/803
Foreign References:
CN105308023A | 2016-02-03 |
Attorney, Agent or Firm:
SHANGHAI PATENT & TRADEMARK LAW OFFICE, LLC (CN)
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