Title:
LIGHT SULFONAMIDE SYNTHESIS REACTION
Document Type and Number:
WIPO Patent Application WO/2023/120292
Kind Code:
A1
Abstract:
Provided is a method for producing a sulfonamide derivative, the method being characterized by including a step of causing a compound having a nitro group to react with a compound having a thiol group under light irradiation, and forming a sulfonamide derivative.
Inventors:
YUASA HIDEYA (JP)
KANAMORI TAKASHI (JP)
YUBE TOMOHIRO (JP)
KANAMORI TAKASHI (JP)
YUBE TOMOHIRO (JP)
Application Number:
PCT/JP2022/045786
Publication Date:
June 29, 2023
Filing Date:
December 13, 2022
Export Citation:
Assignee:
TOKYO INST TECH (JP)
International Classes:
C07C303/36; C07C205/06; C07C311/08; C07C319/12; C07C319/20; C07C323/36; C07C323/67; C07H15/203; C08G75/30
Domestic Patent References:
| WO2017061561A1 | 2017-04-13 | |||
| WO2017175598A1 | 2017-10-12 |
Foreign References:
| CN112939822A | 2021-06-11 | |||
| JP2014210754A | 2014-11-13 |
Other References:
FLEMING STEVEN A., RAWLINS DAVID B., SAMANO VICENTE, ROBINS MORRIS J.: "Photochemistry of nucleoside transport inhibitor 6-S-benzylated thiopurine ribonucleosides. Implications for a new class of photoaffinity labels", THE JOURNAL OF ORGANIC CHEMISTRY, AMERICAN CHEMICAL SOCIETY, vol. 57, no. 22, 1 October 1992 (1992-10-01), pages 5968 - 5976, XP093075562, ISSN: 0022-3263, DOI: 10.1021/jo00048a034
GOVINDARAJU THIMMAIAH, JONKHEIJM PASCAL, GOGOLIN LARS, SCHROEDER HENDRIK, BECKER CHRISTIAN F. W., NIEMEYER CHRISTOF M., WALDMANN H: "Surface immobilization of biomolecules by click sulfonamide reaction", CHEMICAL COMMUNICATIONS, ROYAL SOCIETY OF CHEMISTRY, UK, no. 32, 15 July 2008 (2008-07-15), UK , pages 3723, XP093075569, ISSN: 1359-7345, DOI: 10.1039/b806764c
BAO ZHAOWEI, ZOU JUAN, MOU CHENGLI, JIN ZHICHAO, REN SHI-CHAO, CHI YONGGUI ROBIN: "Direct Reaction of Nitroarenes and Thiols via Photodriven Oxygen Atom Transfer for Access to Sulfonamides", ORGANIC LETTERS, AMERICAN CHEMICAL SOCIETY, US, vol. 24, no. 48, 9 December 2022 (2022-12-09), US , pages 8907 - 8913, XP093075573, ISSN: 1523-7060, DOI: 10.1021/acs.orglett.2c03770
GOVINDARAJU THIMMAIAH, JONKHEIJM PASCAL, GOGOLIN LARS, SCHROEDER HENDRIK, BECKER CHRISTIAN F. W., NIEMEYER CHRISTOF M., WALDMANN H: "Surface immobilization of biomolecules by click sulfonamide reaction", CHEMICAL COMMUNICATIONS, ROYAL SOCIETY OF CHEMISTRY, UK, no. 32, 15 July 2008 (2008-07-15), UK , pages 3723, XP093075569, ISSN: 1359-7345, DOI: 10.1039/b806764c
BAO ZHAOWEI, ZOU JUAN, MOU CHENGLI, JIN ZHICHAO, REN SHI-CHAO, CHI YONGGUI ROBIN: "Direct Reaction of Nitroarenes and Thiols via Photodriven Oxygen Atom Transfer for Access to Sulfonamides", ORGANIC LETTERS, AMERICAN CHEMICAL SOCIETY, US, vol. 24, no. 48, 9 December 2022 (2022-12-09), US , pages 8907 - 8913, XP093075573, ISSN: 1523-7060, DOI: 10.1021/acs.orglett.2c03770
Attorney, Agent or Firm:
NOMURA, Kenichi et al. (JP)
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