Title:
LTA4 HYDROLASE INHIBITORS
Document Type and Number:
WIPO Patent Application WO2000017133
Kind Code:
A3
Abstract:
The invention concerns LTA4 hydrolase inhibiting compounds of formula (I). It also concerns their therapeutic, in particular anti-inflammatory, applications.
Inventors:
DANVY DENIS (FR)
MONTEIL THIERRY (FR)
PLAQUEVENT JEAN-CHRISTOPHE (FR)
DUHAMEL PIERRE (FR)
DUHAMEL LUCETTE (FR)
NOEL NADINE (FR)
GROS CLAUDE (FR)
CHAMARD OLIVIER (FR)
SCHWARTZ JEAN-CHARLES (FR)
LECOMTE JEANNE-MARIE (FR)
MONTEIL THIERRY (FR)
PLAQUEVENT JEAN-CHRISTOPHE (FR)
DUHAMEL PIERRE (FR)
DUHAMEL LUCETTE (FR)
NOEL NADINE (FR)
GROS CLAUDE (FR)
CHAMARD OLIVIER (FR)
SCHWARTZ JEAN-CHARLES (FR)
LECOMTE JEANNE-MARIE (FR)
Application Number:
PCT/FR1999/002240
Publication Date:
November 08, 2001
Filing Date:
September 21, 1999
Export Citation:
Assignee:
BIOPROJET SOC CIV (FR)
INST NAT SANTE RECH MED (FR)
DANVY DENIS (FR)
MONTEIL THIERRY (FR)
PLAQUEVENT JEAN CHRISTOPHE (FR)
DUHAMEL PIERRE (FR)
DUHAMEL LUCETTE (FR)
NOEL NADINE (FR)
GROS CLAUDE (FR)
CHAMARD OLIVIER (FR)
SCHWARTZ JEAN CHARLES (FR)
LECOMTE JEANNE MARIE (FR)
INST NAT SANTE RECH MED (FR)
DANVY DENIS (FR)
MONTEIL THIERRY (FR)
PLAQUEVENT JEAN CHRISTOPHE (FR)
DUHAMEL PIERRE (FR)
DUHAMEL LUCETTE (FR)
NOEL NADINE (FR)
GROS CLAUDE (FR)
CHAMARD OLIVIER (FR)
SCHWARTZ JEAN CHARLES (FR)
LECOMTE JEANNE MARIE (FR)
International Classes:
A61K31/085; A61K31/09; A61K31/10; A61K31/122; A61K31/135; A61K31/137; A61K31/138; A61K31/145; A61K31/165; A61K31/167; A61K31/192; A61K31/194; A61K31/195; A61K31/223; A61K31/225; A61K31/255; A61K31/265; A61K31/27; A61K31/277; A61K31/36; A61K31/4402; A61K31/695; A61P1/16; A61P17/06; A61P19/02; A61P29/00; A61P35/00; A61P43/00; C07B57/00; C07C43/225; C07C49/84; C07C57/34; C07C57/42; C07C69/732; C07C205/37; C07C215/28; C07C217/28; C07C229/22; C07C229/34; C07C233/19; C07C233/25; C07C255/54; C07C271/22; C07C309/66; C07C321/28; C07C323/25; C07C323/29; C07C323/32; C07C323/57; C07C327/30; C07D213/64; C07D317/64; C07F7/10; (IPC1-7): C07C323/25; C07C323/29; C07D317/54; C07D213/64; C07C327/30; A61K31/13; A61K31/36; A61K31/44
Domestic Patent References:
WO1996030014A1 | 1996-10-03 | |||
WO1994000420A1 | 1994-01-06 |
Foreign References:
FR2604434A1 | 1988-04-01 |
Other References:
Y. QIAN ET AL, J. MED. CHEM., vol. 39, no. 1, 1996, pages 217 - 223, XP002106492
M.C. FOURNIE-ZALUSKI ET AL, J. MED. CHEM., vol. 35, no. 7, 1992, pages 1259 - 1266, XP002106493
H. TOH ET AL, BIOCHEM. BIOPHYS. RES. COMMUN., vol. 171, no. 1, 1990, pages 216 - 221, XP002106870
M.C. FOURNIE-ZALUSKI ET AL, J. MED. CHEM., vol. 35, no. 7, 1992, pages 1259 - 1266, XP002106493
H. TOH ET AL, BIOCHEM. BIOPHYS. RES. COMMUN., vol. 171, no. 1, 1990, pages 216 - 221, XP002106870
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