Title:
MACROCYCLIC COMPOUND SERVING AS WEE1 INHIBITOR AND APPLICATIONS THEREOF
Document Type and Number:
WIPO Patent Application WO/2019/085933
Kind Code:
A1
Abstract:
Disclosed in the present invention are a macrocyclic compound serving as a Wee1 inhibitor, and applications thereof in the preparation of drugs for treating Wee1-related diseases. The present invention specifically relates to a compound represented by formula (II), an isomer thereof, and a pharmaceutically acceptable salt thereof.
Inventors:
QIAN WENYUAN (CN)
YANG CHUNDAO (CN)
LI ZHENGWEI (CN)
LI JIE (CN)
LI JIAN (CN)
CHEN SHUHUI (CN)
YANG CHUNDAO (CN)
LI ZHENGWEI (CN)
LI JIE (CN)
LI JIAN (CN)
CHEN SHUHUI (CN)
Application Number:
PCT/CN2018/112909
Publication Date:
May 09, 2019
Filing Date:
October 31, 2018
Export Citation:
Assignee:
MEDSHINE DISCOVERY INC (CN)
International Classes:
C07D471/04; A61P35/00; C07D487/04
Domestic Patent References:
WO2018171633A1 | 2018-09-27 | |||
WO2017075629A2 | 2017-05-04 | |||
WO2007126122A1 | 2007-11-08 | |||
WO2008133866A1 | 2008-11-06 | |||
WO2011034743A1 | 2011-03-24 | |||
WO2013126656A1 | 2013-08-29 | |||
WO2013012681A1 | 2013-01-24 | |||
WO2013059485A1 | 2013-04-25 | |||
WO2013013031A1 | 2013-01-24 | |||
WO2014167347A1 | 2014-10-16 | |||
WO2015019037A1 | 2015-02-12 | |||
WO2015092431A1 | 2015-06-25 |
Foreign References:
US20100221211A1 | 2010-09-02 | |||
US20050215556A1 | 2005-09-29 | |||
CN201711058653A | 2017-11-01 | |||
US20070254892A1 | 2007-11-01 | |||
EP2213673A1 | 2010-08-04 | |||
US20120220572A1 | 2012-08-30 |
Other References:
See also references of EP 3712150A4
Attorney, Agent or Firm:
SHANGHAI BESHINING LAW OFFICE (CN)
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