Title:
METHOD FOR MANUFACTURING BENZODIAZEPINE DERIVATIVE
Document Type and Number:
WIPO Patent Application WO/2010/113458
Kind Code:
A1
Abstract:
Disclosed is a commercially advantageous method for manufacturing a 1,5-benzodiazepine compound. A compound (5) is obtained from a reaction formula and used as an intermediate.
Inventors:
TERAUCHI MASARU (JP)
Application Number:
PCT/JP2010/002237
Publication Date:
October 07, 2010
Filing Date:
March 29, 2010
Export Citation:
Assignee:
ZERIA PHARM CO LTD (JP)
TERAUCHI MASARU (JP)
TERAUCHI MASARU (JP)
International Classes:
C07D243/12; C07C269/06; C07C271/20; C07C271/28; C07C303/36; C07C303/40; C07C311/16; A61K31/551; A61P1/04; A61P35/00; A61P35/02; A61P43/00; C07B61/00
Domestic Patent References:
WO1999064403A1 | 1999-12-16 | |||
WO1998025911A1 | 1998-06-18 | |||
WO2001040197A1 | 2001-06-07 | |||
WO2006077793A1 | 2006-07-27 | |||
WO1998025911A1 | 1998-06-18 | |||
WO1999064403A1 | 1999-12-16 | |||
WO2001040197A1 | 2001-06-07 | |||
WO2006077793A1 | 2006-07-27 | |||
WO1997005129A1 | 1997-02-13 |
Foreign References:
JPH08509237A | 1996-10-01 | |||
JP2008012873A | 2008-01-24 | |||
JPH10203987A | 1998-08-04 |
Other References:
BULL. CHEM. SOC. JPN., vol. 51, 1978, pages 1577
J. CHEM. SOC. PERKIN TRANS., vol. 1, 1997, pages 3219
J. CHEM. SOC., 1957, pages 4559
J. CHEM. SOC. CHEM. COMMUN., 1987, pages 153
J.CHEM. SOC., 1957, pages 4559
TETRAHEDRON ASYMMETRY, vol. 4, 1993, pages 903
See also references of EP 2415766A4
J. CHEM. SOC. PERKIN TRANS., vol. 1, 1997, pages 3219
J. CHEM. SOC., 1957, pages 4559
J. CHEM. SOC. CHEM. COMMUN., 1987, pages 153
J.CHEM. SOC., 1957, pages 4559
TETRAHEDRON ASYMMETRY, vol. 4, 1993, pages 903
See also references of EP 2415766A4
Attorney, Agent or Firm:
THE PATENT CORPORATE BODY ARUGA PATENT OFFICE (JP)
Patent business corporation Alga patent firm (JP)
Patent business corporation Alga patent firm (JP)
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