Title:
METHOD FOR TREATMENT AND PREVENTION OF DISTURBANCES OF THE CENTRAL NERVOUS SYSTEM ASSOCIATED WITH AN ALTERATION OF GLUTAMATERGIC NEUROTRANSMISSION BY ADMINISTRATION OF 2-AMINOBENZENESULFONAMIDE DERIVATIVES
Document Type and Number:
WIPO Patent Application WO2002089734
Kind Code:
A3
Abstract:
2-aminobenzenesulfonamide derivatives are used for the treatment or prevention of the disturbances of the central nervous system associated with a positive or negative modulation of glutamatergic neurotransmission, such as disturbances of memory and learning, schizophrenia, sexual disturbances, ischemic attacks, ictus, etc. For example, a compound according to formula (I): is administered to treat or prevent diseases of the central nervous system having a positive or negative modulation of AMPA/Kainate receptors and a negative modulation of NMDA receptors.
More Like This:
Inventors:
CANNAZZA GIUSEPPE (IT)
PARENTI CARLO (IT)
LINDNER WOLFGANG (IT)
PUIA GIULIA (IT)
BARALDI MARIO (IT)
BRAGHIROLI DANIELA (IT)
TAIT ANNALISA (IT)
PARENTI CARLO (IT)
LINDNER WOLFGANG (IT)
PUIA GIULIA (IT)
BARALDI MARIO (IT)
BRAGHIROLI DANIELA (IT)
TAIT ANNALISA (IT)
Application Number:
PCT/US2002/014262
Publication Date:
March 06, 2003
Filing Date:
May 07, 2002
Export Citation:
Assignee:
RETT CORP (US)
CANNAZZA GIUSEPPE (IT)
PARENTI CARLO (IT)
LINDNER WOLFGANG (IT)
PUIA GIULIA (IT)
BARALDI MARIO (IT)
BRAGHIROLI DANIELA (IT)
TAIT ANNALISA (IT)
CANNAZZA GIUSEPPE (IT)
PARENTI CARLO (IT)
LINDNER WOLFGANG (IT)
PUIA GIULIA (IT)
BARALDI MARIO (IT)
BRAGHIROLI DANIELA (IT)
TAIT ANNALISA (IT)
International Classes:
A61K31/136; A61K31/18; (IPC1-7): A61K31/04
Foreign References:
US6083947A | 2000-07-04 | |||
US5536719A | 1996-07-16 |
Other References:
See also references of EP 1435926A4
Download PDF: