METHODS OF PRODUCING C-ARYL GLUCOSIDE SGLT2 INHIBITORS

WIPO Patent Application WO2004063209

A3

Method for the production of C-aryl glucoside SGLT2 inhibitors useful for the treatment of diabetes and related diseases. and intermediates thereof. The C-aryl glucosides may be complexed with amino acid complex forming reagents.

JPH04217629	PRODUCTION OF SAPONIN FORM HYPOCOTYL OF SOYBEAN
JP2001526663	[Title of Invention] Medical Use of Pyruvate
JP3162465	INCLUSION COMPLEX AND PRODUCTION THEREOF

DESHPANDE PRASHANT P (US)
ELLSWORTH BRUCE A (US)
SINGH JANAK (US)
LAI CHIAJEN (US)
CRISPINO GERARD (US)
RANDAZZO MICHAEL E (US)
GOUGOUTAS JACK Z (US)
DENZEL THEODOR W (DE)

PCT/US2003/041373

May 12, 2005

December 23, 2003

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BRISTOL MYERS SQUIBB CO (US)
DESHPANDE PRASHANT P (US)
ELLSWORTH BRUCE A (US)
SINGH JANAK (US)
LAI CHIAJEN (US)
CRISPINO GERARD (US)
RANDAZZO MICHAEL E (US)
GOUGOUTAS JACK Z (US)
DENZEL THEODOR W (DE)

C07G3/00; C07H1/00; C07H5/04; C07H5/06; C07H7/00; C08B37/00; C07H; (IPC1-7): C07H1/00; C07G3/00

KURIBAYASHI ET AL.: "AgOTfa/SnCl4: a powerful new promoter combination in the Aryl C-glycosidation of a diverse range of sugar acetates and aromatic substrates", TETRAHEDRON LETTERS, vol. 39, no. 25, 1998, pages 4537 - 4540, XP004120733
KURIBAYASHI ET AL.: "C-glycosylated diphenylmethanes and benzophenones: the stille coupling reaction of C-glycosylated aryl tins with benzyl bromides and acid chlorides", JOURNAL OF CARBOHYDRATE CHEMISTRY, vol. 18, no. 4, 1999, pages 393 - 401, XP008044406

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